ME00376B - DIHIDROPTERIDINONI, POSTUPAK ZA NJlHOVO PRIPREMANJE I NJlHOVA PRIMJENA KAO LIJEK - Google Patents

DIHIDROPTERIDINONI, POSTUPAK ZA NJlHOVO PRIPREMANJE I NJlHOVA PRIMJENA KAO LIJEK

Info

Publication number
ME00376B
ME00376B MEP-2008-588A MEP58808A ME00376B ME 00376 B ME00376 B ME 00376B ME P58808 A MEP58808 A ME P58808A ME 00376 B ME00376 B ME 00376B
Authority
ME
Montenegro
Prior art keywords
dihydropteridinones
drugs
production
medicaments
isomers
Prior art date
Application number
MEP-2008-588A
Other languages
English (en)
Inventor
Trixi Brandl
Matthias Grauert
Flavio Solca
Anke Baum
Matthias Hoffmann
Steffen Breitfelder
Christian Eickmeier
Martin Steegmaier
Gisela Schnapp
Jens Juergen Quant
Florian Colbatzky
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Publication of MEP58808A publication Critical patent/MEP58808A/xx
Publication of ME00376B publication Critical patent/ME00376B/me

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D475/00—Heterocyclic compounds containing pteridine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Abstract

Ovaj pronalazak odnosi se, na nove dihidropteridinone, opšte formule (I), pri čemu ostaci L, R 1 , R 2 , R 3 , R 4  i R 5  imaju značenja navedena u patentnim zahtevima i u opisu, na njihove izomere, na postupak za pripremanje ovih dihidropteridinona, kao i na njihovu primenu kao lekova.
MEP-2008-588A 2003-02-26 2003-02-26 DIHIDROPTERIDINONI, POSTUPAK ZA NJlHOVO PRIPREMANJE I NJlHOVA PRIMJENA KAO LIJEK ME00376B (me)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/EP2003/001935 WO2004076454A1 (de) 2003-02-26 2003-02-26 Dihydropteridinone, verfahren zu deren herstellung und deren verwendung als arzneimittel

Publications (2)

Publication Number Publication Date
MEP58808A MEP58808A (en) 2011-05-10
ME00376B true ME00376B (me) 2011-10-10

Family

ID=32921552

Family Applications (1)

Application Number Title Priority Date Filing Date
MEP-2008-588A ME00376B (me) 2003-02-26 2003-02-26 DIHIDROPTERIDINONI, POSTUPAK ZA NJlHOVO PRIPREMANJE I NJlHOVA PRIMJENA KAO LIJEK

Country Status (27)

Country Link
EP (1) EP1599478B1 (me)
JP (1) JP3876265B2 (me)
KR (1) KR100983462B1 (me)
CN (2) CN101200457A (me)
AT (1) ATE361924T1 (me)
AU (1) AU2003215591B2 (me)
BR (1) BR0318145A (me)
CA (1) CA2517020C (me)
CY (1) CY1106752T1 (me)
DE (1) DE50307267D1 (me)
DK (1) DK1599478T3 (me)
EA (1) EA008778B1 (me)
ES (1) ES2287583T3 (me)
HK (1) HK1089444A1 (me)
HR (1) HRP20050735B1 (me)
IL (1) IL170419A (me)
ME (1) ME00376B (me)
MX (1) MXPA05009068A (me)
NO (1) NO332538B1 (me)
NZ (1) NZ542498A (me)
PL (1) PL226417B1 (me)
PT (1) PT1599478E (me)
RS (1) RS52386B (me)
SI (1) SI1599478T1 (me)
TW (1) TWI313600B (me)
UA (1) UA80743C2 (me)
WO (1) WO2004076454A1 (me)

Families Citing this family (112)

* Cited by examiner, † Cited by third party
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KR20050113198A (ko) 2005-12-01
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TW200417369A (en) 2004-09-16
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