MA35660B1 - Inhibiteurs de la protéine pak pour le traitement du syndrome de l'x fragile - Google Patents
Inhibiteurs de la protéine pak pour le traitement du syndrome de l'x fragileInfo
- Publication number
- MA35660B1 MA35660B1 MA37064A MA37064A MA35660B1 MA 35660 B1 MA35660 B1 MA 35660B1 MA 37064 A MA37064 A MA 37064A MA 37064 A MA37064 A MA 37064A MA 35660 B1 MA35660 B1 MA 35660B1
- Authority
- MA
- Morocco
- Prior art keywords
- fragile
- syndrome
- treatment
- inhibitors
- pak protein
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Abstract
Cette invention concerne des inhibiteurs de la protéine pak et des méthodes d'utilisation d'inhibiteurs de la protéine pak pour le traitement du syndrome de l'x fragile.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201161555902P | 2011-11-04 | 2011-11-04 | |
PCT/US2012/063426 WO2013067434A1 (fr) | 2011-11-04 | 2012-11-02 | Inhibiteurs de la protéine pak pour le traitement du syndrome de l'x fragile |
Publications (1)
Publication Number | Publication Date |
---|---|
MA35660B1 true MA35660B1 (fr) | 2014-11-01 |
Family
ID=48192852
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MA37064A MA35660B1 (fr) | 2011-11-04 | 2014-05-26 | Inhibiteurs de la protéine pak pour le traitement du syndrome de l'x fragile |
MA37065A MA35661B1 (fr) | 2011-11-04 | 2014-05-26 | Inhibiteurs de pak pour le traitement de troubles de prolifération cellulaire |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MA37065A MA35661B1 (fr) | 2011-11-04 | 2014-05-26 | Inhibiteurs de pak pour le traitement de troubles de prolifération cellulaire |
Country Status (20)
Country | Link |
---|---|
US (2) | US20130116263A1 (fr) |
EP (2) | EP2773643A4 (fr) |
JP (2) | JP2014532724A (fr) |
KR (2) | KR20140096098A (fr) |
CN (2) | CN104093717A (fr) |
AR (1) | AR089175A1 (fr) |
AU (2) | AU2012327187A1 (fr) |
BR (2) | BR112014010420A2 (fr) |
CA (2) | CA2854471A1 (fr) |
CL (2) | CL2014001131A1 (fr) |
CO (1) | CO7030960A2 (fr) |
CR (2) | CR20140250A (fr) |
EA (2) | EA201490925A1 (fr) |
IL (2) | IL232154A0 (fr) |
MA (2) | MA35660B1 (fr) |
MX (2) | MX2014005292A (fr) |
PH (1) | PH12014500995A1 (fr) |
SG (2) | SG11201401914WA (fr) |
TW (1) | TW201326169A (fr) |
WO (2) | WO2013067434A1 (fr) |
Families Citing this family (22)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2011156780A2 (fr) * | 2010-06-10 | 2011-12-15 | Afraxis, Inc. | 8-(sulfonylbenzyl)pyrido[2,3-d]pyrimidin-7(8h)-ones pour le traitement de troubles du snc |
JP6170060B2 (ja) | 2011-11-04 | 2017-07-26 | エフ.ホフマン−ラ ロシュ アーゲーF. Hoffmann−La Roche Aktiengesellschaft | 新規アリール−キノリン誘導体 |
CN111793068A (zh) | 2013-03-15 | 2020-10-20 | 西建卡尔有限责任公司 | 杂芳基化合物和其用途 |
US9321786B2 (en) | 2013-03-15 | 2016-04-26 | Celgene Avilomics Research, Inc. | Heteroaryl compounds and uses thereof |
EP3943087A1 (fr) | 2013-03-15 | 2022-01-26 | Celgene CAR LLC | Composés hétéroaryle et utilisations associées |
WO2015011252A1 (fr) * | 2013-07-26 | 2015-01-29 | F. Hoffmann-La Roche Ag | Inhibiteurs pyrimidine-pyridinone de sérine/thréonine kinase |
WO2015120049A1 (fr) * | 2014-02-07 | 2015-08-13 | Principia Biopharma, Inc. | Dérivés de quinolone utilisés en tant qu'inhibiteurs du récepteur du facteur de croissance des fibroblastes |
JP6631616B2 (ja) | 2014-07-26 | 2020-01-15 | ノース・アンド・サウス・ブラザー・ファーマシー・インベストメント・カンパニー・リミテッド | CDK阻害剤としての2−アミノ−ピリド[2,3−d]ピリミジン−7(8H)−オン誘導体及びその使用 |
EP3288556A4 (fr) | 2015-04-29 | 2018-09-19 | Dexcel Pharma Technologies Ltd. | Compositions à désintégration par voie orale |
US10694988B2 (en) * | 2016-02-17 | 2020-06-30 | Nuralogix Corporation | System and method for detecting physiological state |
US10076494B2 (en) | 2016-06-16 | 2018-09-18 | Dexcel Pharma Technologies Ltd. | Stable orally disintegrating pharmaceutical compositions |
JP7090037B2 (ja) * | 2016-06-23 | 2022-06-23 | エフ.ホフマン-ラ ロシュ アーゲー | 新規な[1,2,3]トリアゾロ[4,5-d]ピリミジン誘導体 |
WO2018013466A2 (fr) * | 2016-07-15 | 2018-01-18 | Dana-Farber Cancer Institute, Inc. | Biomarqueurs prédictifs de la résistance endocrinienne dans le cancer du sein |
CN106818805A (zh) * | 2016-12-27 | 2017-06-13 | 东莞市联洲知识产权运营管理有限公司 | 一种天然乙酰胆碱酯酶抑制剂及其杀虫应用 |
CN107083428B (zh) * | 2017-04-10 | 2020-09-25 | 徐州医科大学 | Pak5在癌症诊断预后治疗及药物筛选中的应用 |
US20220002429A1 (en) * | 2018-10-24 | 2022-01-06 | Northwestern University | Tumor cell aggregation inhibitors' for treating cancer |
TWI748317B (zh) * | 2019-01-03 | 2021-12-01 | 美商建南德克公司 | 吡啶并-嘧啶酮與喋啶酮化合物及使用方法 |
CN112213400B (zh) * | 2019-07-09 | 2022-06-07 | 四川弘合生物科技有限公司 | 一种β-榄香烯及其有关物质的检测方法 |
CN110496128B (zh) * | 2019-09-23 | 2022-09-30 | 吉林大学 | 利培酮或帕潘立酮在制备治疗弥漫性大b细胞淋巴瘤的药物中的应用 |
US11912668B2 (en) | 2020-11-18 | 2024-02-27 | Deciphera Pharmaceuticals, Llc | GCN2 and perk kinase inhibitors and methods of use thereof |
WO2022152259A1 (fr) * | 2021-01-15 | 2022-07-21 | 江苏先声药业有限公司 | Inhibiteur de cdk2/4/6, son procédé de préparation et son application |
CN113046323A (zh) * | 2021-04-02 | 2021-06-29 | 四川农业大学 | 一种基于miR-532-5p及其靶基因调控卵巢颗粒细胞的方法 |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1201765A3 (fr) * | 2000-10-16 | 2003-08-27 | Axxima Pharmaceuticals Aktiengesellschaft | Kinases cellulaires impliqués dans l'infection par cytomégalovirus et leur inhibition |
EP2094698A1 (fr) * | 2006-11-09 | 2009-09-02 | F. Hoffmann-Roche AG | Dérivés de 6-phényl-pyrido [2,3-d]pyrimidine-7-one substitués utilisés comme inhibiteurs de la kinase et méthodes d'utilisation de ceux-ci |
EP2112150B1 (fr) * | 2008-04-22 | 2013-10-16 | Forma Therapeutics, Inc. | Inhibiteurs Raf améliorés |
US8674095B2 (en) * | 2008-12-19 | 2014-03-18 | Afraxis Holdings, Inc. | Compounds for treating neuropsychiatric conditions |
US8372970B2 (en) * | 2009-10-09 | 2013-02-12 | Afraxis, Inc. | 8-ethyl-6-(aryl)pyrido[2,3-D]pyrimidin-7(8H)-ones for the treatment of CNS disorders |
WO2011156646A2 (fr) * | 2010-06-09 | 2011-12-15 | Afraxis, Inc. | 8-(sulfonylaryl)pyrido[2,3-d]pyrimidin-7(8h)-ones pour le traitement de troubles du snc |
WO2011156780A2 (fr) * | 2010-06-10 | 2011-12-15 | Afraxis, Inc. | 8-(sulfonylbenzyl)pyrido[2,3-d]pyrimidin-7(8h)-ones pour le traitement de troubles du snc |
-
2012
- 2012-11-02 EP EP12845870.0A patent/EP2773643A4/fr not_active Withdrawn
- 2012-11-02 BR BR112014010420A patent/BR112014010420A2/pt not_active Application Discontinuation
- 2012-11-02 EA EA201490925A patent/EA201490925A1/ru unknown
- 2012-11-02 WO PCT/US2012/063426 patent/WO2013067434A1/fr active Application Filing
- 2012-11-02 MX MX2014005292A patent/MX2014005292A/es not_active Application Discontinuation
- 2012-11-02 KR KR1020147014683A patent/KR20140096098A/ko not_active Application Discontinuation
- 2012-11-02 EP EP12844804.0A patent/EP2773642A1/fr not_active Ceased
- 2012-11-02 CA CA2854471A patent/CA2854471A1/fr not_active Abandoned
- 2012-11-02 SG SG11201401914WA patent/SG11201401914WA/en unknown
- 2012-11-02 AU AU2012327187A patent/AU2012327187A1/en not_active Abandoned
- 2012-11-02 SG SG11201401996TA patent/SG11201401996TA/en unknown
- 2012-11-02 MX MX2014005296A patent/MX2014005296A/es not_active Application Discontinuation
- 2012-11-02 EA EA201490927A patent/EA201490927A1/ru unknown
- 2012-11-02 US US13/668,079 patent/US20130116263A1/en not_active Abandoned
- 2012-11-02 KR KR1020147014685A patent/KR20140105451A/ko not_active Application Discontinuation
- 2012-11-02 JP JP2014540152A patent/JP2014532724A/ja active Pending
- 2012-11-02 CA CA2854462A patent/CA2854462A1/fr not_active Abandoned
- 2012-11-02 WO PCT/US2012/063413 patent/WO2013067423A1/fr active Application Filing
- 2012-11-02 US US14/356,118 patent/US20150031693A1/en not_active Abandoned
- 2012-11-02 CN CN201280066127.2A patent/CN104093717A/zh active Pending
- 2012-11-02 BR BR112014010631A patent/BR112014010631A2/pt not_active Application Discontinuation
- 2012-11-02 CN CN201280066130.4A patent/CN104039786A/zh active Pending
- 2012-11-02 AU AU2012327183A patent/AU2012327183A1/en not_active Abandoned
- 2012-11-02 JP JP2014540157A patent/JP2015501786A/ja active Pending
- 2012-11-05 TW TW101141080A patent/TW201326169A/zh unknown
- 2012-11-05 AR ARP120104155A patent/AR089175A1/es unknown
-
2014
- 2014-04-22 IL IL232154A patent/IL232154A0/en unknown
- 2014-04-24 IL IL232215A patent/IL232215A0/en unknown
- 2014-04-30 CL CL2014001131A patent/CL2014001131A1/es unknown
- 2014-04-30 CL CL2014001132A patent/CL2014001132A1/es unknown
- 2014-05-02 PH PH12014500995A patent/PH12014500995A1/en unknown
- 2014-05-26 MA MA37064A patent/MA35660B1/fr unknown
- 2014-05-26 MA MA37065A patent/MA35661B1/fr unknown
- 2014-05-26 CR CR20140250A patent/CR20140250A/es unknown
- 2014-05-26 CR CR20140251A patent/CR20140251A/es unknown
- 2014-06-04 CO CO14119704A patent/CO7030960A2/es unknown
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