MA33679B1 - Derives de 2-oxo-1-pyrrolidinyle imidazothiadiazole - Google Patents

Derives de 2-oxo-1-pyrrolidinyle imidazothiadiazole

Info

Publication number
MA33679B1
MA33679B1 MA34783A MA34783A MA33679B1 MA 33679 B1 MA33679 B1 MA 33679B1 MA 34783 A MA34783 A MA 34783A MA 34783 A MA34783 A MA 34783A MA 33679 B1 MA33679 B1 MA 33679B1
Authority
MA
Morocco
Prior art keywords
oxo
imidazothiadiazole
pyrrolidinyl derivatives
derivatives
pyrrolidinyl
Prior art date
Application number
MA34783A
Other languages
Arabic (ar)
English (en)
Inventor
Yannick Quesnel
Laurent Turet
Joël Mercier
Original Assignee
Ucb Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42034570&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA33679(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Ucb Pharma Sa filed Critical Ucb Pharma Sa
Publication of MA33679B1 publication Critical patent/MA33679B1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/433—Thidiazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

L'invention concerne des dérivés de 2-oxo-1-pyrrolidine imidazothiadiazole, leurs procédés de préparation, des compositions pharmaceutiques les contenant et leur utilisation comme produits pharmaceutiques.
MA34783A 2009-10-23 2012-04-19 Derives de 2-oxo-1-pyrrolidinyle imidazothiadiazole MA33679B1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP09173912 2009-10-23
PCT/EP2010/006434 WO2011047860A1 (fr) 2009-10-23 2010-10-21 Derives de 2-oxo-1-pyrrolidinyle imidazothiadiazole

Publications (1)

Publication Number Publication Date
MA33679B1 true MA33679B1 (fr) 2012-10-01

Family

ID=42034570

Family Applications (1)

Application Number Title Priority Date Filing Date
MA34783A MA33679B1 (fr) 2009-10-23 2012-04-19 Derives de 2-oxo-1-pyrrolidinyle imidazothiadiazole

Country Status (29)

Country Link
US (1) US8822508B2 (fr)
EP (1) EP2491045B1 (fr)
JP (1) JP5808020B2 (fr)
KR (1) KR20120102058A (fr)
CN (1) CN102574869A (fr)
AR (1) AR078722A1 (fr)
AU (1) AU2010310100B2 (fr)
BR (1) BR112012009310B8 (fr)
CA (1) CA2778194C (fr)
CL (1) CL2012001031A1 (fr)
CY (1) CY1117288T1 (fr)
DK (1) DK2491045T3 (fr)
EA (1) EA201200616A1 (fr)
ES (1) ES2565515T3 (fr)
HR (1) HRP20160263T1 (fr)
HU (1) HUE028668T2 (fr)
IL (1) IL218696A0 (fr)
IN (1) IN2012DN02793A (fr)
MA (1) MA33679B1 (fr)
ME (1) ME02355B (fr)
MX (1) MX347070B (fr)
PE (1) PE20121562A1 (fr)
PL (1) PL2491045T3 (fr)
RS (1) RS54595B1 (fr)
SI (1) SI2491045T1 (fr)
SM (1) SMT201600076B (fr)
TN (1) TN2012000147A1 (fr)
TW (1) TW201118103A (fr)
WO (1) WO2011047860A1 (fr)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK2699581T3 (en) * 2011-04-18 2016-01-11 Ucb Biopharma Sprl 2-oxo-1-IMIDAZOLIDINYLIMIDAZOTHIADIAZOLDERIVATIVER
US9581654B2 (en) 2013-02-12 2017-02-28 Johnson Controls Technology Company Vehicle battery monitoring system
WO2015110435A1 (fr) 2014-01-21 2015-07-30 Janssen Pharmaceutica Nv Combinaisons comprenant des modulateurs allostériques positifs ou des agonistes orthostériques de sous-type 2 de récepteur glutamatergique métabotrope, et leur utilisation
LT3096790T (lt) 2014-01-21 2019-10-10 Janssen Pharmaceutica, N.V. Deriniai, apimantys 2 potipio metabotropinio glutamaterginio receptoriaus teigiamus alosterinius moduliatorius arba ortosterinius agonistus, ir jų panaudojimas
TW201908324A (zh) * 2017-07-10 2019-03-01 比利時商優稀美生物醫藥公司 ２－側氧－１－咪唑啶基咪唑噻二唑衍生物
MA49559A (fr) * 2017-07-10 2021-05-05 UCB Biopharma SRL Dérivativés de 2-oxo-1,3-oxazolidinyl imidazothiadiazole
CN107827870B (zh) * 2017-10-24 2019-11-08 江苏仁明生物科技有限公司 一种正电子药物[18f]fpmmp及其制备方法与中间体
CA3083166A1 (fr) 2017-12-12 2019-06-20 UCB Biopharma SRL Derives de 2-oxo-1-pyrrolidinyl imidazothiadiazole
JP7340542B2 (ja) * 2018-05-08 2023-09-07 ユーシービー バイオファルマ エスアールエル １－イミダゾチアジアゾロ－２ｈ－ピロール－５－オン誘導体
CN113549052B (zh) * 2021-07-09 2022-09-02 首都医科大学脑重大疾病研究中心(北京脑重大疾病研究院) 4-苯基-1-（吡啶-4-基甲基）吡咯烷-2-酮衍生物及其制备方法和应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8412358D0 (en) 1984-05-15 1984-06-20 Ucb Sa Pharmaceutical composition
GB8412357D0 (en) 1984-05-15 1984-06-20 Ucb Sa Pharmaceutical composition
GB0004297D0 (en) 2000-02-23 2000-04-12 Ucb Sa 2-oxo-1 pyrrolidine derivatives process for preparing them and their uses
ES2323313T3 (es) * 2003-12-02 2009-07-13 Ucb Pharma, S.A. Derivados de imidazol, procedimientos para prepararlos y sus usos.
EP2308870A3 (fr) * 2005-06-01 2011-10-19 UCB Pharma S.A. Dérivés de 2-oxo-1-pyrrolidine, leurs procédés de préparation et leurs utilisations

Also Published As

Publication number Publication date
CN102574869A (zh) 2012-07-11
EP2491045A1 (fr) 2012-08-29
JP5808020B2 (ja) 2015-11-10
SMT201600076B (it) 2016-04-29
EP2491045B1 (fr) 2015-12-23
TN2012000147A1 (en) 2013-09-19
AR078722A1 (es) 2011-11-30
DK2491045T3 (en) 2016-03-14
CA2778194C (fr) 2016-07-12
WO2011047860A1 (fr) 2011-04-28
BR112012009310B8 (pt) 2021-05-25
JP2013508321A (ja) 2013-03-07
KR20120102058A (ko) 2012-09-17
AU2010310100B2 (en) 2015-09-10
MX347070B (es) 2017-04-11
IN2012DN02793A (fr) 2015-07-24
IL218696A0 (en) 2012-05-31
HUE028668T2 (en) 2016-12-28
CY1117288T1 (el) 2017-04-26
EA201200616A1 (ru) 2012-12-28
PL2491045T3 (pl) 2016-06-30
TW201118103A (en) 2011-06-01
CL2012001031A1 (es) 2012-09-14
US20120245208A1 (en) 2012-09-27
BR112012009310B1 (pt) 2021-01-12
SI2491045T1 (sl) 2016-04-29
MX2012003839A (es) 2012-05-08
AU2010310100A1 (en) 2012-05-17
US8822508B2 (en) 2014-09-02
BR112012009310A2 (pt) 2016-06-07
RS54595B1 (en) 2016-08-31
CA2778194A1 (fr) 2011-04-28
ME02355B (fr) 2016-06-20
HRP20160263T1 (hr) 2016-04-08
ES2565515T3 (es) 2016-04-05
PE20121562A1 (es) 2012-11-30

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