MA24511A1 - Inhibiteurs de l'enzyme de conversion de l'interleukine 1b - Google Patents

Inhibiteurs de l'enzyme de conversion de l'interleukine 1b

Info

Publication number
MA24511A1
MA24511A1 MA23932A MA23932A MA24511A1 MA 24511 A1 MA24511 A1 MA 24511A1 MA 23932 A MA23932 A MA 23932A MA 23932 A MA23932 A MA 23932A MA 24511 A1 MA24511 A1 MA 24511A1
Authority
MA
Morocco
Prior art keywords
interleukin
enzyme inhibitors
conversion enzyme
conversion
inhibitors
Prior art date
Application number
MA23932A
Other languages
English (en)
Inventor
W Bemis Guy
J Lauffer David
A Murcko Mark
M C Golec Julian
J Livingston David
D Mullican Michael
Original Assignee
Vertex Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US08/261,452 external-priority patent/US5756466A/en
Priority claimed from US08/440,898 external-priority patent/US5847135A/en
Application filed by Vertex Pharma filed Critical Vertex Pharma
Publication of MA24511A1 publication Critical patent/MA24511A1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/0202—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -NH-X-X-C(=0)-, X being an optionally substituted carbon atom or a heteroatom, e.g. beta-amino acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Genetics & Genomics (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Immunology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Peptides Or Proteins (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Paper (AREA)
MA23932A 1994-06-17 1995-06-16 Inhibiteurs de l'enzyme de conversion de l'interleukine 1b MA24511A1 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US08/261,452 US5756466A (en) 1994-06-17 1994-06-17 Inhibitors of interleukin-1β converting enzyme
US08/405,581 US5656627A (en) 1994-06-17 1995-03-17 Inhibitors of interleukin-1β converting enzyme
US08/440,898 US5847135A (en) 1994-06-17 1995-05-25 Inhibitors of interleukin-1β converting enzyme

Publications (1)

Publication Number Publication Date
MA24511A1 true MA24511A1 (fr) 1998-12-31

Family

ID=27401408

Family Applications (1)

Application Number Title Priority Date Filing Date
MA23932A MA24511A1 (fr) 1994-06-17 1995-06-16 Inhibiteurs de l'enzyme de conversion de l'interleukine 1b

Country Status (22)

Country Link
US (2) US5716929A (fr)
EP (1) EP0784628A1 (fr)
JP (1) JP4190029B2 (fr)
CN (1) CN1192035C (fr)
AP (1) AP797A (fr)
AU (1) AU709114B2 (fr)
BG (1) BG63634B1 (fr)
BR (1) BR9508051A (fr)
CA (1) CA2192089C (fr)
CZ (1) CZ298625B6 (fr)
FI (1) FI965036A (fr)
GE (1) GEP20012446B (fr)
HU (1) HUT76622A (fr)
IL (1) IL114015A0 (fr)
IS (1) IS4399A (fr)
MA (1) MA24511A1 (fr)
MX (1) MX9606546A (fr)
NZ (1) NZ289560A (fr)
PL (1) PL185693B1 (fr)
SK (1) SK287422B6 (fr)
TW (1) TW509698B (fr)
WO (1) WO1995035308A1 (fr)

Families Citing this family (138)

* Cited by examiner, † Cited by third party
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JPH10504285A (ja) 1998-04-28
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CN1159196A (zh) 1997-09-10
CZ369896A3 (en) 1997-06-11
IL114015A0 (en) 1995-10-31
AP797A (en) 2000-01-07
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TW509698B (en) 2002-11-11
EP0784628A1 (fr) 1997-07-23
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