LU86958A1 - Sels d'acide thiamorpholinone carboxylique et de derives de diamino-2,4 pyrimidine,leur utilisation en cosmetique et pharmacie - Google Patents

Sels d'acide thiamorpholinone carboxylique et de derives de diamino-2,4 pyrimidine,leur utilisation en cosmetique et pharmacie Download PDF

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Publication number
LU86958A1
LU86958A1 LU86958A LU86958A LU86958A1 LU 86958 A1 LU86958 A1 LU 86958A1 LU 86958 A LU86958 A LU 86958A LU 86958 A LU86958 A LU 86958A LU 86958 A1 LU86958 A1 LU 86958A1
Authority
LU
Luxembourg
Prior art keywords
thiamorpholinone
diamino
piperidino
carboxylate
pyrimidine
Prior art date
Application number
LU86958A
Other languages
English (en)
French (fr)
Inventor
Jean Maignan
Gerard Lang
Serge Restle
Original Assignee
Oreal
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Oreal filed Critical Oreal
Priority to LU86958A priority Critical patent/LU86958A1/fr
Priority to AT88112024T priority patent/ATE61801T1/de
Priority to EP88112024A priority patent/EP0304649B1/de
Priority to DE8888112024T priority patent/DE3862083D1/de
Priority to CA000573492A priority patent/CA1314884C/fr
Priority to JP63188534A priority patent/JPS6450867A/ja
Priority to US07/225,818 priority patent/US4970063A/en
Publication of LU86958A1 publication Critical patent/LU86958A1/fr
Priority to GR91400638T priority patent/GR3001965T3/el

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D279/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/101,4-Thiazines; Hydrogenated 1,4-thiazines
    • C07D279/121,4-Thiazines; Hydrogenated 1,4-thiazines not condensed with other rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/49Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/49Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
    • A61K8/494Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with more than one nitrogen as the only hetero atom
    • A61K8/4953Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with more than one nitrogen as the only hetero atom containing pyrimidine ring derivatives, e.g. minoxidil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61QSPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q7/00Preparations for affecting hair growth
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/50Three nitrogen atoms

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Birds (AREA)
  • Dermatology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Cosmetics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
LU86958A 1987-07-31 1987-07-31 Sels d'acide thiamorpholinone carboxylique et de derives de diamino-2,4 pyrimidine,leur utilisation en cosmetique et pharmacie LU86958A1 (fr)

Priority Applications (8)

Application Number Priority Date Filing Date Title
LU86958A LU86958A1 (fr) 1987-07-31 1987-07-31 Sels d'acide thiamorpholinone carboxylique et de derives de diamino-2,4 pyrimidine,leur utilisation en cosmetique et pharmacie
AT88112024T ATE61801T1 (de) 1987-07-31 1988-07-26 Salze von 6-piperidino-2,4-diaminopyrimidin-3oxyd und von derivaten der thiamorpholin-3-on-5- carbonsaeure und deren verwendung in kosmetischen stoffen und als heilmittel.
EP88112024A EP0304649B1 (de) 1987-07-31 1988-07-26 Salze von 6-Piperidino-2,4-diaminopyrimidin-3-oxyd und von Derivaten der Thiamorpholin-3-on-5-carbonsäure und deren Verwendung in kosmetischen Stoffen und als Heilmittel
DE8888112024T DE3862083D1 (de) 1987-07-31 1988-07-26 Salze von 6-piperidino-2,4-diaminopyrimidin-3-oxyd und von derivaten der thiamorpholin-3-on-5-carbonsaeure und deren verwendung in kosmetischen stoffen und als heilmittel.
CA000573492A CA1314884C (fr) 1987-07-31 1988-07-29 Sels d'acide thiamorpholinone carboxylique et de derives de diamino-2,4 pyrimidine, leur utilisation en cosmetique et pharmacie
JP63188534A JPS6450867A (en) 1987-07-31 1988-07-29 Salts of thiamorpholinonecarboxylic acid and 2,4-diaminopyrimidine derivative and use for cosmetic and pharmaceutical composition
US07/225,818 US4970063A (en) 1987-07-31 1988-07-29 Salts of thiamorpholinone carboxylic acid with 2,4-diaminopyrimidine derivatives and their use in cosmetics and pharmaceuticals
GR91400638T GR3001965T3 (en) 1987-07-31 1991-05-20 Salts of 6-piperidino-2,4-diaminopyrimidin-3-oxide and of derivatives of thiamorpholin-3-on-5-carboxylic acid, their cosmetical and medicinal use

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
LU86958 1987-07-31
LU86958A LU86958A1 (fr) 1987-07-31 1987-07-31 Sels d'acide thiamorpholinone carboxylique et de derives de diamino-2,4 pyrimidine,leur utilisation en cosmetique et pharmacie

Publications (1)

Publication Number Publication Date
LU86958A1 true LU86958A1 (fr) 1989-03-08

Family

ID=19730954

Family Applications (1)

Application Number Title Priority Date Filing Date
LU86958A LU86958A1 (fr) 1987-07-31 1987-07-31 Sels d'acide thiamorpholinone carboxylique et de derives de diamino-2,4 pyrimidine,leur utilisation en cosmetique et pharmacie

Country Status (8)

Country Link
US (1) US4970063A (de)
EP (1) EP0304649B1 (de)
JP (1) JPS6450867A (de)
AT (1) ATE61801T1 (de)
CA (1) CA1314884C (de)
DE (1) DE3862083D1 (de)
GR (1) GR3001965T3 (de)
LU (1) LU86958A1 (de)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
LU87304A1 (fr) * 1988-07-29 1990-02-07 Oreal Nouveaux derives d'ureylene triamino-2,4,6 pyrimidine oxyde-3,leur preparation et leur utilisation en cosmetique et dermopharmacie
JP2869168B2 (ja) * 1990-08-10 1999-03-10 鐘紡株式会社 育毛剤及びそれを含有する養毛化粧料
PT683659E (pt) * 1993-02-09 2003-01-31 Tulsa Forte Pharmacy Entpr Inc Um metodo para estimular o crescimento de cabelo com derivados cationicos do minoxidil usando iontoforese terapeutica
CN112811614A (zh) * 2020-12-03 2021-05-18 嘉兴沃特泰科环保科技股份有限公司 一种循环水无磷阻垢剂及其制备方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3382247A (en) * 1965-11-01 1968-05-07 Upjohn Co 6-amino-1, 2-dihydro-1-hydroxy-2-imino-4-phenoxypyrimidines
US4139619A (en) * 1976-05-24 1979-02-13 The Upjohn Company 6-Amino-4-(substituted amino)-1,2-dihydro-1-hydroxy-2-iminopyrimidine, topical compositions and process for hair growth
HU177601B (en) * 1978-10-27 1981-11-28 Egyt Gyogyszervegyeszeti Gyar New process for preparing 6-piperidino-2,4-diamino-pyrimidine-3-oxide
FR2525106B1 (fr) * 1982-04-15 1985-06-07 Oreal Composition cosmetique contenant en tant qu'agent actif sur l'elasticite et la souplesse de la peau, de la thiamorpholinone ou l'un de ses derives
FR2525220A1 (fr) * 1982-04-15 1983-10-21 Oreal Nouveaux derives substitues de la thiamorpholinone et leurs procedes de preparation
IT1201436B (it) * 1985-07-19 1989-02-02 Vincenzo Zappia Formulazioni topiche a lento rilascio

Also Published As

Publication number Publication date
CA1314884C (fr) 1993-03-23
EP0304649B1 (de) 1991-03-20
GR3001965T3 (en) 1992-11-23
JPS6450867A (en) 1989-02-27
EP0304649A1 (de) 1989-03-01
US4970063A (en) 1990-11-13
DE3862083D1 (de) 1991-04-25
ATE61801T1 (de) 1991-04-15

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