KR840009103A - 1-아졸릴-3-피라졸릴-2-프로판올 유도체의 제조방법 - Google Patents
1-아졸릴-3-피라졸릴-2-프로판올 유도체의 제조방법 Download PDFInfo
- Publication number
- KR840009103A KR840009103A KR1019840001928A KR840001928A KR840009103A KR 840009103 A KR840009103 A KR 840009103A KR 1019840001928 A KR1019840001928 A KR 1019840001928A KR 840001928 A KR840001928 A KR 840001928A KR 840009103 A KR840009103 A KR 840009103A
- Authority
- KR
- South Korea
- Prior art keywords
- formula
- carbon atoms
- phenyl
- optionally substituted
- alkyl
- Prior art date
Links
- CICQCPXOTVUFNW-UHFFFAOYSA-N 1-(1h-pyrazol-5-yl)-3-(1h-pyrrol-2-yl)propan-2-ol Chemical class C=1C=NNC=1CC(O)CC1=CC=CN1 CICQCPXOTVUFNW-UHFFFAOYSA-N 0.000 title 1
- 125000004432 carbon atom Chemical group C* 0.000 claims 8
- 125000000217 alkyl group Chemical group 0.000 claims 6
- 150000001875 compounds Chemical class 0.000 claims 6
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims 6
- 239000002253 acid Substances 0.000 claims 4
- 125000000304 alkynyl group Chemical group 0.000 claims 4
- 125000004353 pyrazol-1-yl group Chemical group [H]C1=NN(*)C([H])=C1[H] 0.000 claims 4
- 125000003626 1,2,4-triazol-1-yl group Chemical group [*]N1N=C([H])N=C1[H] 0.000 claims 3
- 125000003342 alkenyl group Chemical group 0.000 claims 3
- 239000003085 diluting agent Substances 0.000 claims 3
- 229910052736 halogen Inorganic materials 0.000 claims 3
- 150000002367 halogens Chemical class 0.000 claims 3
- 125000002962 imidazol-1-yl group Chemical group [*]N1C([H])=NC([H])=C1[H] 0.000 claims 3
- 125000001624 naphthyl group Chemical group 0.000 claims 3
- 125000003884 phenylalkyl group Chemical group 0.000 claims 3
- 150000003839 salts Chemical class 0.000 claims 3
- WTKZEGDFNFYCGP-UHFFFAOYSA-N Pyrazole Chemical compound C=1C=NNC=1 WTKZEGDFNFYCGP-UHFFFAOYSA-N 0.000 claims 2
- KAESVJOAVNADME-UHFFFAOYSA-N Pyrrole Chemical compound C=1C=CNC=1 KAESVJOAVNADME-UHFFFAOYSA-N 0.000 claims 2
- 229910052783 alkali metal Inorganic materials 0.000 claims 2
- 150000001340 alkali metals Chemical class 0.000 claims 2
- 239000011230 binding agent Substances 0.000 claims 2
- 238000004519 manufacturing process Methods 0.000 claims 2
- 229910052751 metal Inorganic materials 0.000 claims 2
- 239000002184 metal Substances 0.000 claims 2
- 125000001424 substituent group Chemical group 0.000 claims 2
- ZFOWEXGOKLKOFQ-UHFFFAOYSA-N 2-(oxiran-2-ylmethyl)-1h-pyrrole Chemical compound C=1C=CNC=1CC1CO1 ZFOWEXGOKLKOFQ-UHFFFAOYSA-N 0.000 claims 1
- ZAMOUSCENKQFHK-UHFFFAOYSA-N Chlorine atom Chemical compound [Cl] ZAMOUSCENKQFHK-UHFFFAOYSA-N 0.000 claims 1
- PXGOKWXKJXAPGV-UHFFFAOYSA-N Fluorine Chemical compound FF PXGOKWXKJXAPGV-UHFFFAOYSA-N 0.000 claims 1
- 125000004183 alkoxy alkyl group Chemical group 0.000 claims 1
- 125000003545 alkoxy group Chemical group 0.000 claims 1
- 125000004414 alkyl thio group Chemical group 0.000 claims 1
- 229910052801 chlorine Inorganic materials 0.000 claims 1
- 239000000460 chlorine Substances 0.000 claims 1
- 229910052731 fluorine Inorganic materials 0.000 claims 1
- 239000011737 fluorine Substances 0.000 claims 1
- 229910052739 hydrogen Inorganic materials 0.000 claims 1
- 239000001257 hydrogen Substances 0.000 claims 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 claims 1
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 claims 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims 1
- 229910052698 phosphorus Inorganic materials 0.000 claims 1
- 239000011574 phosphorus Substances 0.000 claims 1
- 239000001294 propane Substances 0.000 claims 1
- 125000005346 substituted cycloalkyl group Chemical group 0.000 claims 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
- A01N43/647—Triazoles; Hydrogenated triazoles
- A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Dentistry (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Agronomy & Crop Science (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
내용 없음
Description
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음
Claims (3)
- a) 일반식(Ⅱ))의 2-아졸릴메틸-옥시란을 일반식(Ⅲ)의 아졸과 알칼리 금속 알코올레이트 및 희석제 존재하에 반응시키거나,b) 일반식(Ⅳ)의 2-할로게노메틸-옥시란을 일반식(Ⅴ)의 피라졸과 희석제 및 바람직하게는 산결합제 존재하에 반응시키거나,c) 일반식(Ⅵ)의 디할로게노알칸올을 일반식(Ⅴ)의 피라졸과 희석제 및 바람직하게는 산결합체 존재하에 반응시키고, 만일 필요하면, 수득된 일반식(Ⅰ)의 화합물에 산 또는 금속염을 가함을 특징으로 하여 일반식(Ⅰ)의-아졸릴-3-피라졸릴-2-프로판을 유도체 및 그의 산부가염 및 금속염 착화합물을 제조하는 방법.상기식에서Az는 1,2,4-트리아졸-1일, 이미다졸-1-일 또는 피라졸-1-일이고R은 알킬, 알케닐, 알키닐, 임의로 치환된 페닐, 임의로 치환된 페닐알킬, 임의로 치환된 페닐알케닐, 임의로 치환된 페닐알키닐, 나프틸 또는 임의로 치환된 시클로알킬이며,Az′는 Az와 같은 의미이나 Az 및/또는 Az′는 피라졸-1-일이고,Hal은 할로겐이며,M은 수소 또는 알칼리금속이다.
- 제1항에 있어서, Ar은 1,2,4-트리아졸-1-일, 이미다졸-1-일 또는 피라졸-1-일이고, R은 탄소수 1 내지 12의 지쇄 또는 측쇄 알킬, 각 경우에 탄소수 2 내지 6의 지쇄 또는 측쇄 알케닐 또는 알키닐, 또는 페닐, 알킬부위가 탄소수 1 내지 4인 페닐알킬, 알케닐 부위가 탄소수 2 내지 4인 페닐 알케닐 또는 알키닐 부위가 탄소수 2 내지 4인 페닐 알키닐, (이때 페닐, 페닐알킬, 페닐알케닐 또는 페닐알키닐은 각각의 경우에 할로겐, 탄소수 1 내지 4의 알킬, 각 경우에 탄소수 1 또는 2인 알콕시 및 알킬티오, 각 알킬티위가 탄소수 1 또는 2인 알콕시알킬, 할로겐으로 임의로 치환된 페닐등의 같거나 또는 다른 치환체로 페닐상에서 임의로 일-, 이- 또는 삼-치환되어 있음)또는 나프틸 또는 나프틸 또는 탄소수 3 내지 7을 갖고, 탄소수 1내지 4의 알킬로 임의로 치환된 시클로알킬을 나타내는 일반식(Ⅰ)의 화합물을 제조하는 방법.
- 제1항에 있어서, Az가 1,2,4-트리아졸-1-일, 이미다졸-1-일 또는 피라졸-1-일이고 R은 불소, 염소, 메틸 및 메톡시의 같거나 또는 다른 치환체로 임의로 일- 또는 이치환된 페닐인 일반식(Ⅰ)의 화합물을 제조하는 방법.※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DEP3313073.6 | 1983-04-12 | ||
DE3313073A DE3313073A1 (de) | 1983-04-12 | 1983-04-12 | 1-azolyl-3-pyrazolyl-2-propanol-derivate, verfahren zu ihrer herstellung und ihre verwendung als fungizide |
Publications (2)
Publication Number | Publication Date |
---|---|
KR840009103A true KR840009103A (ko) | 1984-12-24 |
KR900008815B1 KR900008815B1 (ko) | 1990-11-30 |
Family
ID=6196058
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
KR1019840001928A KR900008815B1 (ko) | 1983-04-12 | 1984-04-12 | 1-아졸릴-3-피라졸릴-2-프로판올 유도체의 제조방법 |
Country Status (16)
Country | Link |
---|---|
US (1) | US4587239A (ko) |
EP (1) | EP0121888B1 (ko) |
JP (1) | JPS59196867A (ko) |
KR (1) | KR900008815B1 (ko) |
AT (1) | ATE34574T1 (ko) |
AU (1) | AU564060B2 (ko) |
BR (1) | BR8401701A (ko) |
CA (1) | CA1242444A (ko) |
DE (2) | DE3313073A1 (ko) |
DK (1) | DK187684A (ko) |
ES (1) | ES531513A0 (ko) |
GR (1) | GR81836B (ko) |
HU (1) | HU192005B (ko) |
IL (1) | IL71477A (ko) |
NZ (1) | NZ207775A (ko) |
ZA (1) | ZA842675B (ko) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8306351D0 (en) * | 1983-03-08 | 1983-04-13 | Ici Plc | Azole fungicides |
DE3513259A1 (de) * | 1985-04-13 | 1986-10-23 | Bayer Ag, 5090 Leverkusen | Heterocyclische amid-derivate |
GB8614712D0 (en) * | 1986-06-17 | 1986-07-23 | Ici Plc | Heterocyclic compounds |
DE3730871A1 (de) * | 1987-09-15 | 1989-03-23 | Bayer Ag | Bisazolyl-hydroxyalkyl-derivate |
WO1993012108A1 (en) * | 1991-12-18 | 1993-06-24 | Schering Corporation | Imidazolyl or imidazoylalkyl substituted with a four or five membered nitrogen containing heterocyclic ring |
WO1993014152A1 (en) * | 1992-01-16 | 1993-07-22 | Teijin Limited | Polyester film for metal sheet lamination and use thereof |
US20020068771A1 (en) * | 1997-02-21 | 2002-06-06 | Dentsply Detrey Gmbh. | Low shrinking polymerizable dental material |
JP5055263B2 (ja) * | 2005-03-30 | 2012-10-24 | ダエウン ファーマシューティカル カンパニー リミテッド | 抗真菌性トリアゾール誘導体 |
JP2009513698A (ja) * | 2005-10-31 | 2009-04-02 | デウン ファーマシューティカル カンパニー リミテッド | 新規な抗菌トリアゾール誘導体 |
KR20080062876A (ko) * | 2006-12-29 | 2008-07-03 | 주식회사 대웅제약 | 신규한 항진균성 트리아졸 유도체 |
EA024385B1 (ru) * | 2011-06-19 | 2016-09-30 | Ваймет Фармасьютикалс, Инк. | Соединения, ингибирующие металлоферменты |
KR101964195B1 (ko) * | 2011-06-23 | 2019-04-01 | 비아멧 파마슈티컬즈(엔씨), 인코포레이티드 | 금속효소 억제제 화합물 |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2979512A (en) * | 1961-04-11 | Pyrazole derivatives | ||
DE2448060A1 (de) * | 1974-10-09 | 1976-04-15 | Bayer Ag | Mittel zur regulierung des pflanzenwachstums |
DE2461406C2 (de) * | 1974-12-24 | 1984-06-14 | Bayer Ag, 5090 Leverkusen | Azolyl-(1)-methane und deren Salze, Verfahren zu ihrer Herstellung sowie diese enthaltende Arzneimittel |
DE2635883A1 (de) * | 1976-08-10 | 1978-02-16 | Bayer Ag | N-sulfenylierte oximcarbamate, verfahren zu ihrer herstellung und ihre verwendung als insektizide, akarizide und nematozide |
CH619931A5 (ko) * | 1976-08-12 | 1980-10-31 | Ciba Geigy Ag | |
US4229460A (en) * | 1977-01-31 | 1980-10-21 | Janssen Pharmaceutica N.V. | Heterocyclic derivatives of 1-(1,3-dioxolan-2-ylmethyl)-1H-1,2,4-triazoles having antifungal and antibacterial properties |
GB2078719B (en) * | 1980-06-02 | 1984-04-26 | Ici Ltd | Heterocyclic compounds |
DE3175673D1 (en) * | 1980-11-19 | 1987-01-15 | Ici Plc | Triazole compounds, a process for preparing them, their use as plant fungicides and fungicidal compositions containing them |
DE3262386D1 (en) * | 1981-06-06 | 1985-03-28 | Pfizer Ltd | Antifungal agents, processes for their preparation, and pharmaceutical compositions containing them |
-
1983
- 1983-04-12 DE DE3313073A patent/DE3313073A1/de not_active Withdrawn
-
1984
- 1984-03-22 US US06/592,162 patent/US4587239A/en not_active Expired - Fee Related
- 1984-04-02 EP EP84103627A patent/EP0121888B1/de not_active Expired
- 1984-04-02 AT AT84103627T patent/ATE34574T1/de not_active IP Right Cessation
- 1984-04-02 DE DE8484103627T patent/DE3471481D1/de not_active Expired
- 1984-04-06 AU AU26613/84A patent/AU564060B2/en not_active Expired - Fee Related
- 1984-04-09 NZ NZ207775A patent/NZ207775A/en unknown
- 1984-04-09 JP JP59069281A patent/JPS59196867A/ja active Pending
- 1984-04-09 IL IL71477A patent/IL71477A/xx not_active IP Right Cessation
- 1984-04-10 CA CA000451607A patent/CA1242444A/en not_active Expired
- 1984-04-11 GR GR74373A patent/GR81836B/el unknown
- 1984-04-11 DK DK187684A patent/DK187684A/da not_active Application Discontinuation
- 1984-04-11 HU HU841426A patent/HU192005B/hu not_active IP Right Cessation
- 1984-04-11 BR BR8401701A patent/BR8401701A/pt unknown
- 1984-04-11 ES ES531513A patent/ES531513A0/es active Granted
- 1984-04-11 ZA ZA842675A patent/ZA842675B/xx unknown
- 1984-04-12 KR KR1019840001928A patent/KR900008815B1/ko not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
US4587239A (en) | 1986-05-06 |
DK187684D0 (da) | 1984-04-11 |
ATE34574T1 (de) | 1988-06-15 |
AU564060B2 (en) | 1987-07-30 |
HUT34019A (en) | 1985-01-28 |
BR8401701A (pt) | 1984-11-20 |
DE3471481D1 (en) | 1988-06-30 |
JPS59196867A (ja) | 1984-11-08 |
AU2661384A (en) | 1984-10-18 |
ES8502112A1 (es) | 1984-12-16 |
KR900008815B1 (ko) | 1990-11-30 |
HU192005B (en) | 1987-04-28 |
CA1242444A (en) | 1988-09-27 |
ES531513A0 (es) | 1984-12-16 |
IL71477A (en) | 1987-01-30 |
EP0121888A2 (de) | 1984-10-17 |
EP0121888A3 (en) | 1986-03-19 |
DE3313073A1 (de) | 1984-10-18 |
IL71477A0 (en) | 1984-07-31 |
GR81836B (ko) | 1984-12-12 |
DK187684A (da) | 1984-10-13 |
NZ207775A (en) | 1986-06-11 |
ZA842675B (en) | 1984-11-28 |
EP0121888B1 (de) | 1988-05-25 |
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