JPS6039678B2 - 新規インド−ル誘導体の製法 - Google Patents

新規インド−ル誘導体の製法

Info

Publication number
JPS6039678B2
JPS6039678B2 JP49115686A JP11568674A JPS6039678B2 JP S6039678 B2 JPS6039678 B2 JP S6039678B2 JP 49115686 A JP49115686 A JP 49115686A JP 11568674 A JP11568674 A JP 11568674A JP S6039678 B2 JPS6039678 B2 JP S6039678B2
Authority
JP
Japan
Prior art keywords
formula
hydrogen
lower alkyl
ethyl
indolyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
JP49115686A
Other languages
English (en)
Japanese (ja)
Other versions
JPS5076076A (nl
Inventor
レヒアツプ ア−キボ−ルド ジヨン
ランバ−ト ジヤツクソン ジヨン
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
John Wyeth and Brother Ltd
Original Assignee
John Wyeth and Brother Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by John Wyeth and Brother Ltd filed Critical John Wyeth and Brother Ltd
Publication of JPS5076076A publication Critical patent/JPS5076076A/ja
Publication of JPS6039678B2 publication Critical patent/JPS6039678B2/ja
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
JP49115686A 1973-10-10 1974-10-09 新規インド−ル誘導体の製法 Expired JPS6039678B2 (ja)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
GB47208/73 1973-10-10
GB4720873 1973-10-10
GB3531/74 1974-01-25
GB353174*[A GB1425354A (en) 1973-10-10 1974-01-25 Indole derivatives
GB727774 1974-02-18
GB7277/74 1974-02-18

Publications (2)

Publication Number Publication Date
JPS5076076A JPS5076076A (nl) 1975-06-21
JPS6039678B2 true JPS6039678B2 (ja) 1985-09-06

Family

ID=27254287

Family Applications (1)

Application Number Title Priority Date Filing Date
JP49115686A Expired JPS6039678B2 (ja) 1973-10-10 1974-10-09 新規インド−ル誘導体の製法

Country Status (10)

Country Link
JP (1) JPS6039678B2 (nl)
CH (4) CH610323A5 (nl)
DE (1) DE2447947A1 (nl)
FR (1) FR2247239B1 (nl)
GB (1) GB1425354A (nl)
HK (1) HK36179A (nl)
IE (1) IE40052B1 (nl)
KE (1) KE2950A (nl)
MY (1) MY7900210A (nl)
NL (1) NL179731C (nl)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS62157297U (nl) * 1986-03-27 1987-10-06

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4147786A (en) 1976-02-02 1979-04-03 Ciba-Geigy Corporation 1-Indolylalkyl-3-or 4-trimethyleneurido-piperidines
GB1542137A (en) * 1976-03-12 1979-03-14 Wyeth John & Brother Ltd Process for preparing 3(piperidinoalkyl)indoles
JPS56158Y2 (nl) * 1976-06-28 1981-01-06
GB1586817A (en) * 1977-12-01 1981-03-25 Wyeth John & Brother Ltd Indole derivatives
US4242347A (en) 1979-06-18 1980-12-30 Ciba-Geigy Corporation Hypotensive indolylalkylpiperidyl guanidines and isoureas
DK733788A (da) * 1988-01-14 1989-07-15 Fujisawa Pharmaceutical Co Indolylpiperidinderivater og fremgangsmaade til fremstilling deraf
SE9902987D0 (sv) 1999-08-24 1999-08-24 Astra Pharma Prod Novel compounds
FR2802206B1 (fr) 1999-12-14 2005-04-22 Sod Conseils Rech Applic Derives de 4-aminopiperidine et leur utilisation en tant que medicament
GB0011838D0 (en) * 2000-05-17 2000-07-05 Astrazeneca Ab Chemical compounds
GB0104050D0 (en) 2001-02-19 2001-04-04 Astrazeneca Ab Chemical compounds
GB0107228D0 (en) 2001-03-22 2001-05-16 Astrazeneca Ab Chemical compounds
SE0103818D0 (sv) 2001-11-15 2001-11-15 Astrazeneca Ab Chemical compounds
SE0301369D0 (sv) 2003-05-09 2003-05-09 Astrazeneca Ab Chemical compounds

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS62157297U (nl) * 1986-03-27 1987-10-06

Also Published As

Publication number Publication date
CH611615A5 (en) 1979-06-15
NL179731B (nl) 1986-06-02
FR2247239A1 (nl) 1975-05-09
IE40052B1 (en) 1979-02-28
MY7900210A (en) 1979-12-31
KE2950A (en) 1979-04-27
FR2247239B1 (nl) 1978-07-21
JPS5076076A (nl) 1975-06-21
IE40052L (en) 1975-04-10
NL7413358A (nl) 1975-04-14
HK36179A (en) 1979-06-15
GB1425354A (en) 1976-02-18
CH610323A5 (en) 1979-04-12
CH612431A5 (en) 1979-07-31
DE2447947A1 (de) 1975-04-17
NL179731C (nl) 1986-11-03
CH613449A5 (en) 1979-09-28

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