JPS5239694A - Producing novel penicillins and cephalosporins - Google Patents

Producing novel penicillins and cephalosporins

Info

Publication number
JPS5239694A
JPS5239694A JP50104046A JP10404675A JPS5239694A JP S5239694 A JPS5239694 A JP S5239694A JP 50104046 A JP50104046 A JP 50104046A JP 10404675 A JP10404675 A JP 10404675A JP S5239694 A JPS5239694 A JP S5239694A
Authority
JP
Japan
Prior art keywords
cephalosporins
producing novel
penicillins
novel penicillins
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP50104046A
Other languages
Japanese (ja)
Other versions
JPS5310076B2 (en
Inventor
Isamu Saikawa
Shuntaro Takano
Chosaku Yoshida
Okuta Takashima
Kaishu Momoi
Chiaki Kutani
Hiroshi Kodama
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Toyama Chemical Co Ltd
Original Assignee
Toyama Chemical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Toyama Chemical Co Ltd filed Critical Toyama Chemical Co Ltd
Priority to JP50104046A priority Critical patent/JPS5239694A/en
Priority to GB32136/76A priority patent/GB1517098A/en
Priority to CY1030A priority patent/CY1030A/en
Priority to CH1072576A priority patent/CH618442A5/en
Priority to IN1558/CAL/76A priority patent/IN144093B/en
Priority to MX764854U priority patent/MX4341E/en
Priority to PT65518A priority patent/PT65518B/en
Priority to ES451053A priority patent/ES451053A1/en
Priority to AR264504A priority patent/AR212920A1/en
Priority to NL7609539A priority patent/NL7609539A/en
Priority to HU76TO1036A priority patent/HU173129B/en
Priority to SE7609558A priority patent/SE434156B/en
Priority to FI762464A priority patent/FI63584C/en
Priority to DK389276A priority patent/DK147235C/en
Priority to DD7600194498A priority patent/DD129215A5/en
Priority to CA260,041A priority patent/CA1077925A/en
Priority to AT643376A priority patent/AT347581B/en
Publication of JPS5239694A publication Critical patent/JPS5239694A/en
Publication of JPS5310076B2 publication Critical patent/JPS5310076B2/ja
Priority to KE299379A priority patent/KE2993A/en
Priority to HK715/79A priority patent/HK71579A/en
Priority to MY1980163A priority patent/MY8000163A/en
Priority to FI810164A priority patent/FI65622C/en
Priority to SE8205079A priority patent/SE446985B/en
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

PURPOSE: Penicillins and cephalosporins of formula I(R1 is H, carboxyl protective group, salt-forming cation; Z is radical of formula II or III ;R is amino acid radical ; n is 1, 2, 2;X is O, S;m is 4-n;R2 ,R3 are H, halogen, alkyl, cycloalkyl, aryl, acyl;R4 is H, CN, azide;A is H, CN, alkyl;Y is O, S)9 For example, D(-)α-(4-ethyl-2,3-dioxo-piperazinocarbonylamino) benzylpenicillin.
COPYRIGHT: (C)1977,JPO&Japio
JP50104046A 1975-08-29 1975-08-29 Producing novel penicillins and cephalosporins Granted JPS5239694A (en)

Priority Applications (22)

Application Number Priority Date Filing Date Title
JP50104046A JPS5239694A (en) 1975-08-29 1975-08-29 Producing novel penicillins and cephalosporins
GB32136/76A GB1517098A (en) 1975-08-29 1976-08-02 Process for producing penicillins and cephalosporins
CY1030A CY1030A (en) 1975-08-29 1976-08-02 Process for producing penicillins and cephalosporins
CH1072576A CH618442A5 (en) 1975-08-29 1976-08-24 Process for the preparation of new penicillins and of new cephalosporins
IN1558/CAL/76A IN144093B (en) 1975-08-29 1976-08-25
MX764854U MX4341E (en) 1975-08-29 1976-08-25 PROCEDURE FOR THE PREPARATION OF PENICILLINS AND CEPHALOSPORINS CONTAINING A MONO OXO GROUP OR DIOXO-PIPERAZINE (TIO) CARBONYLAMINE
PT65518A PT65518B (en) 1975-08-29 1976-08-26 Process for the preparation of novel penicillins and cephalosporins
SE7609558A SE434156B (en) 1975-08-29 1976-08-27 PROCEDURE FOR PENICILLIN PREPARATION
AR264504A AR212920A1 (en) 1975-08-29 1976-08-27 PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF THE 6- (DIOXO-PIPERAZINE-CARBONYLAMINE-ACETAMIDE) PENICILANIC ACID OR OF THE 7- (DIOXO-PIPERAZINE-CARBONYLAMINE-ACETAMIDE) -DELTA-3-CEFEM-4-CARBOXYL ACID
NL7609539A NL7609539A (en) 1975-08-29 1976-08-27 PROCESS FOR THE PREPARATION OF NEW PENICILLINS AND CEPHALOSSPORINS.
HU76TO1036A HU173129B (en) 1975-08-29 1976-08-27 Process for producing new, piperazino-substituted pename- and cepheme- derivatives
ES451053A ES451053A1 (en) 1975-08-29 1976-08-27 Process for producing penicillins and cephalosporins
FI762464A FI63584C (en) 1975-08-29 1976-08-27 PROCEDURE FOR THE FRAMEWORK OF THERAPEUTIC THERAPY
DK389276A DK147235C (en) 1975-08-29 1976-08-27 METHOD OF ANALOGUE FOR PREPARING PENICILLIN OR CEPHALOSPORIN COMPOUNDS OR PHARMACEUTICAL ACCEPTABLE SALTS THEREOF
DD7600194498A DD129215A5 (en) 1975-08-29 1976-08-27 PROCESS FOR THE PREPARATION OF NEW PENICILLIN AND CEPHALOSPORIN
CA260,041A CA1077925A (en) 1975-08-29 1976-08-27 Process for producing novel penicillins and cephalosporins
AT643376A AT347581B (en) 1975-08-29 1976-08-30 PROCESS FOR THE PRODUCTION OF NEW PENICILLINES AND CEPHALOSPORINES
KE299379A KE2993A (en) 1975-08-29 1979-09-25 A process for producing novel penicillins and cephalosporins
HK715/79A HK71579A (en) 1975-08-29 1979-10-11 A process for producing novel penicillins and cephalosporins
MY1980163A MY8000163A (en) 1975-08-29 1980-12-31 A process for producing novel penicillins and cephalosporins
FI810164A FI65622C (en) 1975-08-29 1981-01-21 FREQUENCY REQUIREMENT FOR THERAPEUTIC THERAPEUTIC PENICILLINER
SE8205079A SE446985B (en) 1975-08-29 1982-09-07 PROCEDURE FOR THE PREPARATION OF CEPHALOSPORINE COMPOUNDS

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP50104046A JPS5239694A (en) 1975-08-29 1975-08-29 Producing novel penicillins and cephalosporins

Publications (2)

Publication Number Publication Date
JPS5239694A true JPS5239694A (en) 1977-03-28
JPS5310076B2 JPS5310076B2 (en) 1978-04-11

Family

ID=14370263

Family Applications (1)

Application Number Title Priority Date Filing Date
JP50104046A Granted JPS5239694A (en) 1975-08-29 1975-08-29 Producing novel penicillins and cephalosporins

Country Status (19)

Country Link
JP (1) JPS5239694A (en)
AR (1) AR212920A1 (en)
AT (1) AT347581B (en)
CA (1) CA1077925A (en)
CH (1) CH618442A5 (en)
CY (1) CY1030A (en)
DD (1) DD129215A5 (en)
DK (1) DK147235C (en)
ES (1) ES451053A1 (en)
FI (1) FI63584C (en)
GB (1) GB1517098A (en)
HK (1) HK71579A (en)
HU (1) HU173129B (en)
IN (1) IN144093B (en)
MX (1) MX4341E (en)
MY (1) MY8000163A (en)
NL (1) NL7609539A (en)
PT (1) PT65518B (en)
SE (2) SE434156B (en)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS57121042A (en) * 1981-01-22 1982-07-28 Nippon Synthetic Chem Ind Co Ltd:The Resin composition
JPS57131240A (en) * 1981-02-06 1982-08-14 Nippon Synthetic Chem Ind Co Ltd:The Resin composition

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GR78166B (en) * 1981-05-04 1984-09-26 Chinoin Gyogyszer Es Vegyeszet
JPS5859420U (en) * 1981-10-16 1983-04-21 ヤンマーディーゼル株式会社 rotary mower device
CN111533758A (en) * 2020-05-11 2020-08-14 承德医学院 Piperacillin magnesium compound, composition, preparation method and application

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS57121042A (en) * 1981-01-22 1982-07-28 Nippon Synthetic Chem Ind Co Ltd:The Resin composition
JPH0317861B2 (en) * 1981-01-22 1991-03-11 Nippon Synthetic Chem Ind
JPS57131240A (en) * 1981-02-06 1982-08-14 Nippon Synthetic Chem Ind Co Ltd:The Resin composition
JPH0317862B2 (en) * 1981-02-06 1991-03-11 Nippon Synthetic Chem Ind

Also Published As

Publication number Publication date
SE434156B (en) 1984-07-09
FI63584B (en) 1983-03-31
PT65518B (en) 1978-07-04
HU173129B (en) 1979-02-28
ATA643376A (en) 1978-05-15
PT65518A (en) 1976-09-01
CA1077925A (en) 1980-05-20
DK147235C (en) 1986-10-06
FI63584C (en) 1983-07-11
MY8000163A (en) 1980-12-31
HK71579A (en) 1979-10-19
MX4341E (en) 1982-04-02
ES451053A1 (en) 1977-12-16
DK389276A (en) 1977-03-01
SE7609558L (en) 1977-03-01
IN144093B (en) 1978-03-25
AR212920A1 (en) 1978-11-15
CH618442A5 (en) 1980-07-31
CY1030A (en) 1980-08-01
JPS5310076B2 (en) 1978-04-11
SE446985B (en) 1986-10-20
AT347581B (en) 1979-01-10
SE8205079L (en) 1982-09-07
GB1517098A (en) 1978-07-12
SE8205079D0 (en) 1982-09-07
NL7609539A (en) 1977-03-02
DK147235B (en) 1984-05-21
FI762464A (en) 1977-03-01
DD129215A5 (en) 1978-01-04

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