JO3055B1 - Picolinamide derivatives as kinase inhibitors - Google Patents

Picolinamide derivatives as kinase inhibitors

Info

Publication number
JO3055B1
JO3055B1 JOP/2009/0326A JOP20090326A JO3055B1 JO 3055 B1 JO3055 B1 JO 3055B1 JO P20090326 A JOP20090326 A JO P20090326A JO 3055 B1 JO3055 B1 JO 3055B1
Authority
JO
Jordan
Prior art keywords
kinase
compositions
kinase inhibitors
new compounds
picolinamide derivatives
Prior art date
Application number
JOP/2009/0326A
Other languages
Arabic (ar)
Inventor
Lan Jiong
Nishiguchi Gisele
Burger Matthew
Han Wooseok
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Application granted granted Critical
Publication of JO3055B1 publication Critical patent/JO3055B1/en

Links

Abstract

New compounds, compositions and methods of inhibition of Provirus Integration of Maloney Kinase (PIM kinase) activity associated with tumorigenesis in a human or animal subject are provided. In certain embodiments, the compounds and compositions are effective to inhibit the activity of at least one PIM kinase. The new compounds and compositions may be used either alone or in combination with at least one additional agent for the treatment of a serine/threonine kinase or receptor tyrosine kinase mediated disorder, such as cancer.
JOP/2009/0326A 2008-09-02 2009-09-01 Picolinamide derivatives as kinase inhibitors JO3055B1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US9366608P 2008-09-02 2008-09-02

Publications (1)

Publication Number Publication Date
JO3055B1 true JO3055B1 (en) 2017-03-15

Family

ID=43566735

Family Applications (1)

Application Number Title Priority Date Filing Date
JOP/2009/0326A JO3055B1 (en) 2008-09-02 2009-09-01 Picolinamide derivatives as kinase inhibitors

Country Status (3)

Country Link
AR (1) AR073474A1 (en)
JO (1) JO3055B1 (en)
UA (1) UA103034C2 (en)

Also Published As

Publication number Publication date
AR073474A1 (en) 2010-11-10
UA103034C2 (en) 2013-09-10

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