ITMI20052008A1 - Nuovi antimalarici derivati della 4-aminochinolina - Google Patents
Nuovi antimalarici derivati della 4-aminochinolinaInfo
- Publication number
- ITMI20052008A1 ITMI20052008A1 IT002008A ITMI20052008A ITMI20052008A1 IT MI20052008 A1 ITMI20052008 A1 IT MI20052008A1 IT 002008 A IT002008 A IT 002008A IT MI20052008 A ITMI20052008 A IT MI20052008A IT MI20052008 A1 ITMI20052008 A1 IT MI20052008A1
- Authority
- IT
- Italy
- Prior art keywords
- aminochinolina
- antimalaric
- derivatives
- new
- new antimalaric
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D455/00—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine
- C07D455/02—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing not further condensed quinolizine ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- A61P33/06—Antimalarials
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Priority Applications (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT002008A ITMI20052008A1 (it) | 2005-10-21 | 2005-10-21 | Nuovi antimalarici derivati della 4-aminochinolina |
PCT/IB2006/002946 WO2007045987A1 (en) | 2005-10-21 | 2006-10-20 | New anti-malaria derivatives of 4-aminoquinoline |
EP06809083A EP1937686A1 (en) | 2005-10-21 | 2006-10-20 | New anti-malaria derivatives of 4-aminoquinoline |
CNA2006800486047A CN101346381A (zh) | 2005-10-21 | 2006-10-20 | 新颖的抗疟疾4-氨基喹啉衍生物 |
AP2008004444A AP2008004444A0 (en) | 2005-10-21 | 2008-04-26 | New anti-malaria derivatives of 4-aminoquinoline |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT002008A ITMI20052008A1 (it) | 2005-10-21 | 2005-10-21 | Nuovi antimalarici derivati della 4-aminochinolina |
Publications (1)
Publication Number | Publication Date |
---|---|
ITMI20052008A1 true ITMI20052008A1 (it) | 2007-04-22 |
Family
ID=37735214
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IT002008A ITMI20052008A1 (it) | 2005-10-21 | 2005-10-21 | Nuovi antimalarici derivati della 4-aminochinolina |
Country Status (5)
Country | Link |
---|---|
EP (1) | EP1937686A1 (it) |
CN (1) | CN101346381A (it) |
AP (1) | AP2008004444A0 (it) |
IT (1) | ITMI20052008A1 (it) |
WO (1) | WO2007045987A1 (it) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU2009316721A1 (en) | 2008-11-18 | 2010-05-27 | Oregon Health & Science University | Compounds for treating parasitic disease |
EP2680844B1 (en) | 2011-03-04 | 2016-10-19 | GlaxoSmithKline Intellectual Property Development Limited | Amino-quinolines as kinase inhibitors |
TWI547494B (zh) | 2011-08-18 | 2016-09-01 | 葛蘭素史克智慧財產發展有限公司 | 作為激酶抑制劑之胺基喹唑啉類 |
TW201425307A (zh) | 2012-09-13 | 2014-07-01 | Glaxosmithkline Llc | 作為激酶抑制劑之胺基-喹啉類 |
TWI592417B (zh) | 2012-09-13 | 2017-07-21 | 葛蘭素史克智慧財產發展有限公司 | 胺基喹唑啉激酶抑制劑之前藥 |
CN102898369A (zh) * | 2012-11-05 | 2013-01-30 | 上海书亚医药科技有限公司 | 3-氨基-7-溴喹啉-2-甲酸乙酯及其制备方法 |
RU2662810C2 (ru) | 2013-02-21 | 2018-07-31 | Глэксосмитклайн Интеллекчуал Проперти Дивелопмент Лимитед | Хиназолины в качестве ингибиторов киназы |
CN108191829B (zh) * | 2016-06-30 | 2020-07-03 | 珠海赛隆药业股份有限公司(长沙)医药研发中心 | 应用富马酸沃诺拉赞中间体ⅳ制备富马酸沃诺拉赞的方法 |
CN107915720B (zh) * | 2016-10-08 | 2020-09-11 | 常州市第四制药厂有限公司 | 沃诺拉赞的新制备方法 |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2002072554A1 (en) * | 2001-03-14 | 2002-09-19 | The University Of Liverpool | Anti-malarial compounds |
ITMI20032044A1 (it) * | 2003-10-21 | 2005-04-22 | Univ Degli Studi Milano | Chinolizidinil e chinolizidinilalchil-derivati della 4-ammino-chinolina ad attivita' antimalarica |
-
2005
- 2005-10-21 IT IT002008A patent/ITMI20052008A1/it unknown
-
2006
- 2006-10-20 WO PCT/IB2006/002946 patent/WO2007045987A1/en active Application Filing
- 2006-10-20 EP EP06809083A patent/EP1937686A1/en not_active Withdrawn
- 2006-10-20 CN CNA2006800486047A patent/CN101346381A/zh active Pending
-
2008
- 2008-04-26 AP AP2008004444A patent/AP2008004444A0/xx unknown
Also Published As
Publication number | Publication date |
---|---|
AP2008004444A0 (en) | 2008-04-30 |
CN101346381A (zh) | 2009-01-14 |
EP1937686A1 (en) | 2008-07-02 |
WO2007045987A1 (en) | 2007-04-26 |
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