IT8621734A0 - Processo per la preparazione dell'alfa-n-[(ipoxatin-9-il)pentilossicarbonil-]arginina - Google Patents

Processo per la preparazione dell'alfa-n-[(ipoxatin-9-il)pentilossicarbonil-]arginina

Info

Publication number
IT8621734A0
IT8621734A0 IT8621734A IT2173486A IT8621734A0 IT 8621734 A0 IT8621734 A0 IT 8621734A0 IT 8621734 A IT8621734 A IT 8621734A IT 2173486 A IT2173486 A IT 2173486A IT 8621734 A0 IT8621734 A0 IT 8621734A0
Authority
IT
Italy
Prior art keywords
pentihloxycarbonyl
ipoxatin
arginine
alpha
preparation
Prior art date
Application number
IT8621734A
Other languages
English (en)
Other versions
IT1213495B (it
Inventor
Riccardo Stradi
Original Assignee
Sigma Tau Ind Farmaceuti
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sigma Tau Ind Farmaceuti filed Critical Sigma Tau Ind Farmaceuti
Publication of IT8621734A0 publication Critical patent/IT8621734A0/it
Priority to IT8621734A priority Critical patent/IT1213495B/it
Priority to DE8787113168T priority patent/DE3764051D1/de
Priority to EP87113168A priority patent/EP0260588B1/en
Priority to ES87113168T priority patent/ES2017485B3/es
Priority to AT87113168T priority patent/ATE55130T1/de
Priority to PH35793A priority patent/PH25318A/en
Priority to IL83863A priority patent/IL83863A0/xx
Priority to JP62228206A priority patent/JPS6388184A/ja
Priority to IN669/MAS/87A priority patent/IN165609B/en
Priority to AR87308744A priority patent/AR242576A1/es
Priority to CA000547042A priority patent/CA1276148C/en
Priority to KR1019870010239A priority patent/KR950008971B1/ko
Priority to AU78471/87A priority patent/AU593136B2/en
Priority to ZA876961A priority patent/ZA876961B/xx
Priority to DK489087A priority patent/DK168570B1/da
Application granted granted Critical
Publication of IT1213495B publication Critical patent/IT1213495B/it
Priority to GR90400651T priority patent/GR3000796T3/el

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/26Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/28Oxygen atom
    • C07D473/30Oxygen atom attached in position 6, e.g. hypoxanthine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IT8621734A 1986-09-17 1986-09-17 Processo per la preparazione dell'alfa-n-[(ipoxatin-9-il)pentilossicarbonil-]arginina IT1213495B (it)

Priority Applications (16)

Application Number Priority Date Filing Date Title
IT8621734A IT1213495B (it) 1986-09-17 1986-09-17 Processo per la preparazione dell'alfa-n-[(ipoxatin-9-il)pentilossicarbonil-]arginina
DE8787113168T DE3764051D1 (de) 1986-09-17 1987-09-09 Verfahren zur herstellung von alpha-n-((hypoxanthin-9-yl)-pentyloxycarbonyl)-arginin.
EP87113168A EP0260588B1 (en) 1986-09-17 1987-09-09 Process for the preparation of alpha-N-[(hypoxanthin-9-yl)-pentyloxycarbonyl]-arginine
ES87113168T ES2017485B3 (es) 1986-09-17 1987-09-09 Proceso para la preparacion de alfa-n-(hipoxantin-9il)pentiloxi-carbonil-arginina.
AT87113168T ATE55130T1 (de) 1986-09-17 1987-09-09 Verfahren zur herstellung von alpha-n((hypoxanthin-9-yl)-pentyloxycarbonyl>-arginin.
PH35793A PH25318A (en) 1986-09-17 1987-09-10 Process for the preparation of (-n-£hypoxanthin-9-yl0 pentyloxycarbonyl|-arginine
IL83863A IL83863A0 (en) 1986-09-17 1987-09-10 Process for the preparation of alpha-n-(hypoxanthin-9-yl)-pentyloxycarbonyl)-arginine
JP62228206A JPS6388184A (ja) 1986-09-17 1987-09-11 α―N―〔(ハイポキサンチン―9―イル)―ペンチルオキシカルボニル〕―アルギニンの製造方法
IN669/MAS/87A IN165609B (it) 1986-09-17 1987-09-14
AR87308744A AR242576A1 (es) 1986-09-17 1987-09-16 Proceso para la preparacion de alfa-n-¡(hipoxantin-9-il)-pentiloxicarbonil¿-arginina.
CA000547042A CA1276148C (en) 1986-09-17 1987-09-16 Process for the preparation of -n-¬(hypoxanthin-9-yl)-pentyloxycarbonyl|-arginine
KR1019870010239A KR950008971B1 (ko) 1986-09-17 1987-09-16 α-N-[(히포크산틴-9-일)펜틸옥시카르보닐]알기닌의 제조방법
AU78471/87A AU593136B2 (en) 1986-09-17 1987-09-16 Process for the preparation of alpha-N- ((hypoxanthin -9-yl)- pentyloxycarbonyl)- arginine
ZA876961A ZA876961B (en) 1986-09-17 1987-09-16 Process for the preparation of alpha-n-((hypoxanthin-9-yl)-pentyloxy-carbonyl)-arginine
DK489087A DK168570B1 (da) 1986-09-17 1987-09-17 Fremgangsmåde til fremstilling af alfa-N-[(hypoxanthin-9-yl)-pentyloxycarbonyl]-arginin
GR90400651T GR3000796T3 (en) 1986-09-17 1990-09-14 Process for the preparation of alpha-n-û(hypoxanthin-9-yl)-pentyloxycarbonyl¨-arginine

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT8621734A IT1213495B (it) 1986-09-17 1986-09-17 Processo per la preparazione dell'alfa-n-[(ipoxatin-9-il)pentilossicarbonil-]arginina

Publications (2)

Publication Number Publication Date
IT8621734A0 true IT8621734A0 (it) 1986-09-17
IT1213495B IT1213495B (it) 1989-12-20

Family

ID=11186113

Family Applications (1)

Application Number Title Priority Date Filing Date
IT8621734A IT1213495B (it) 1986-09-17 1986-09-17 Processo per la preparazione dell'alfa-n-[(ipoxatin-9-il)pentilossicarbonil-]arginina

Country Status (16)

Country Link
EP (1) EP0260588B1 (it)
JP (1) JPS6388184A (it)
KR (1) KR950008971B1 (it)
AR (1) AR242576A1 (it)
AT (1) ATE55130T1 (it)
AU (1) AU593136B2 (it)
CA (1) CA1276148C (it)
DE (1) DE3764051D1 (it)
DK (1) DK168570B1 (it)
ES (1) ES2017485B3 (it)
GR (1) GR3000796T3 (it)
IL (1) IL83863A0 (it)
IN (1) IN165609B (it)
IT (1) IT1213495B (it)
PH (1) PH25318A (it)
ZA (1) ZA876961B (it)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1241452B (it) * 1990-06-28 1994-01-17 Sigma Tau Ind Farmaceuti Derivati oligopeptidici dell'ipoxantina dotati di attivita' immunomodulante e composizioni farmaceutiche che li contengono
IT1244501B (it) * 1991-03-22 1994-07-15 Sigma Tau Ind Farmaceuti Derivati amminoacilici e oligopeptidici dell'allopurinolo dotati di attivita' immunostimolante e composizioni farmaceutiche che li contengono
US5994361A (en) * 1994-06-22 1999-11-30 Biochem Pharma Substituted purinyl derivatives with immunomodulating activity
NZ506202A (en) 1998-03-19 2003-10-31 Bristol Myers Squibb Co Biphasic controlled release delivery system for high solubility pharmaceuticals and method
US10940159B2 (en) 2010-07-09 2021-03-09 James Trinca Green Combination immediate/delayed release delivery system for short half-life pharmaceuticals including remogliflozin

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4221910A (en) * 1978-09-15 1980-09-09 Newport Pharmaceuticals International, Inc. 9-(Hydroxy alkyl)purines
AU564576B2 (en) * 1981-09-24 1987-08-20 Sigma-Tau Industrie Farmaceutiche Riunite S.P.A. Purine derivatives

Also Published As

Publication number Publication date
AU593136B2 (en) 1990-02-01
CA1276148C (en) 1990-11-13
JPS6388184A (ja) 1988-04-19
KR880003944A (ko) 1988-06-01
IT1213495B (it) 1989-12-20
EP0260588B1 (en) 1990-08-01
DK168570B1 (da) 1994-04-25
AU7847187A (en) 1988-03-24
DE3764051D1 (de) 1990-09-06
PH25318A (en) 1991-04-30
ZA876961B (en) 1988-05-25
KR950008971B1 (ko) 1995-08-10
IN165609B (it) 1989-11-25
IL83863A0 (en) 1988-02-29
DK489087D0 (da) 1987-09-17
DK489087A (da) 1988-03-18
EP0260588A1 (en) 1988-03-23
AR242576A1 (es) 1993-04-30
GR3000796T3 (en) 1991-10-10
ES2017485B3 (es) 1991-02-16
ATE55130T1 (de) 1990-08-15

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Legal Events

Date Code Title Description
TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19950928