IT8068267A0 - Composti intermedi per la preparazione di derivati della morfina eprocedimento per la preparazione ditali composti - Google Patents

Composti intermedi per la preparazione di derivati della morfina eprocedimento per la preparazione ditali composti

Info

Publication number
IT8068267A0
IT8068267A0 IT8068267A IT6826780A IT8068267A0 IT 8068267 A0 IT8068267 A0 IT 8068267A0 IT 8068267 A IT8068267 A IT 8068267A IT 6826780 A IT6826780 A IT 6826780A IT 8068267 A0 IT8068267 A0 IT 8068267A0
Authority
IT
Italy
Prior art keywords
preparation
compounds
procedure
morphine derivatives
intermediate compounds
Prior art date
Application number
IT8068267A
Other languages
English (en)
Italian (it)
Inventor
Dennis J Malfer
Donald F Loncrini
Original Assignee
Mallinckrodt Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mallinckrodt Inc filed Critical Mallinckrodt Inc
Publication of IT8068267A0 publication Critical patent/IT8068267A0/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D489/00Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula:
    • C07D489/06Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: with a hetero atom directly attached in position 14
    • C07D489/08Oxygen atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IT8068267A 1979-08-09 1980-08-07 Composti intermedi per la preparazione di derivati della morfina eprocedimento per la preparazione ditali composti IT8068267A0 (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US6527579A 1979-08-09 1979-08-09

Publications (1)

Publication Number Publication Date
IT8068267A0 true IT8068267A0 (it) 1980-08-07

Family

ID=22061564

Family Applications (1)

Application Number Title Priority Date Filing Date
IT8068267A IT8068267A0 (it) 1979-08-09 1980-08-07 Composti intermedi per la preparazione di derivati della morfina eprocedimento per la preparazione ditali composti

Country Status (16)

Country Link
JP (1) JPS56501010A (no)
AU (1) AU6116580A (no)
BE (1) BE884671A (no)
DD (1) DD154541A5 (no)
DK (1) DK151781A (no)
ES (1) ES494122A0 (no)
FI (1) FI802479A (no)
FR (1) FR2465735A1 (no)
GB (1) GB2066256A (no)
IL (1) IL60783A0 (no)
IT (1) IT8068267A0 (no)
NL (1) NL8020319A (no)
NO (1) NO802139L (no)
PL (1) PL226162A1 (no)
SE (1) SE8102214L (no)
WO (1) WO1981000409A1 (no)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4795813A (en) * 1981-08-17 1989-01-03 The Florida Board Of Regents On Behalf Of The Florida State University Synthesis of derivatives of codeine and other 3-O-alkylmorphines
US5668285A (en) * 1986-10-31 1997-09-16 The United States Of America As Represented By The Department Of Health And Human Services Total synthesis of northebaine, normophine, noroxymorphone enantiomers and derivatives via N-Nor intermediates
ATE178329T1 (de) * 1989-10-16 1999-04-15 Us Health Totale synthese von northebain-, normorphin-, noroxymorphon-enantiomeren und -derivaten via n- nor-zwischenverbindungen

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3249616A (en) * 1966-05-03 Ix-dfflydroxy-g-oxo-n-phenethylmor- phinan (cis) and production thereof
CA913077A (en) * 1972-10-24 J. Pachter Irwin Process of preparing n-substituted 14-hydroxydihydronormorphines
US2772270A (en) * 1954-10-21 1956-11-27 M J Lewenstein 14-hydroxymorphinone and 8, 14-dihydroxydihydromorphinone
US2806033A (en) * 1955-08-03 1957-09-10 Lewenstein Morphine derivative
BE638369A (no) * 1962-10-10
US3332950A (en) * 1963-03-23 1967-07-25 Endo Lab 14-hydroxydihydronormorphinone derivatives
NL7106612A (en) * 1971-05-13 1972-11-15 N-cycloalkylalkyl-14-hydroxy-dihydronormorphines - - by o-demethylation of 14-methoxy cpds
US3775414A (en) * 1972-05-10 1973-11-27 Bristol Myers Co Process for the preparation of 14-hydroxymorphinan derivatives
US4161597A (en) * 1976-12-20 1979-07-17 Research Corporation N-alkyl-14-hydroxymorphinans and derivatives

Also Published As

Publication number Publication date
ES8104296A1 (es) 1981-04-16
AU6116580A (en) 1981-02-12
DK151781A (da) 1981-04-03
WO1981000409A1 (en) 1981-02-19
FR2465735A1 (fr) 1981-03-27
DD154541A5 (de) 1982-03-31
GB2066256A (en) 1981-07-08
PL226162A1 (no) 1981-04-24
NL8020319A (nl) 1981-07-01
SE8102214L (sv) 1981-04-07
BE884671A (fr) 1980-12-01
FI802479A (fi) 1981-02-10
JPS56501010A (no) 1981-07-23
NO802139L (no) 1981-02-10
IL60783A0 (en) 1980-10-26
ES494122A0 (es) 1981-04-16

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