IT1397212B1 - Derivati di amminoalcoli e loro attivita' terapeutica - Google Patents

Derivati di amminoalcoli e loro attivita' terapeutica

Info

Publication number
IT1397212B1
IT1397212B1 ITMI2009A002317A ITMI20092317A IT1397212B1 IT 1397212 B1 IT1397212 B1 IT 1397212B1 IT MI2009A002317 A ITMI2009A002317 A IT MI2009A002317A IT MI20092317 A ITMI20092317 A IT MI20092317A IT 1397212 B1 IT1397212 B1 IT 1397212B1
Authority
IT
Italy
Prior art keywords
aminoalks
derivatives
therapeutic activity
therapeutic
activity
Prior art date
Application number
ITMI2009A002317A
Other languages
English (en)
Inventor
Renato Canevotti
Marina Carini
Gian Paolo Negrisoli
Giancarlo Aldini
Marica Orioli
Giulio Vistoli
Massimo Previtali
Original Assignee
Flamma Spa
Univ Degli Studi Milano
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Flamma Spa, Univ Degli Studi Milano filed Critical Flamma Spa
Priority to ITMI2009A002317A priority Critical patent/IT1397212B1/it
Priority to JP2012546410A priority patent/JP5787899B2/ja
Priority to ES10799013.7T priority patent/ES2439322T3/es
Priority to PCT/EP2010/070238 priority patent/WO2011080139A1/en
Priority to EP10799013.7A priority patent/EP2519507B1/en
Priority to US13/519,645 priority patent/US8623900B2/en
Priority to CN201080059714.XA priority patent/CN102791696B/zh
Publication of ITMI20092317A1 publication Critical patent/ITMI20092317A1/it
Application granted granted Critical
Publication of IT1397212B1 publication Critical patent/IT1397212B1/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/12Ophthalmic agents for cataracts
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P39/00General protective or antinoxious agents
    • A61P39/06Free radical scavengers or antioxidants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Diabetes (AREA)
  • Ophthalmology & Optometry (AREA)
  • Obesity (AREA)
  • Biochemistry (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Rheumatology (AREA)
  • Emergency Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Toxicology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
ITMI2009A002317A 2009-12-29 2009-12-29 Derivati di amminoalcoli e loro attivita' terapeutica IT1397212B1 (it)

Priority Applications (7)

Application Number Priority Date Filing Date Title
ITMI2009A002317A IT1397212B1 (it) 2009-12-29 2009-12-29 Derivati di amminoalcoli e loro attivita' terapeutica
JP2012546410A JP5787899B2 (ja) 2009-12-29 2010-12-20 アミノアルコール誘導体およびそれらの治療活性
ES10799013.7T ES2439322T3 (es) 2009-12-29 2010-12-20 Derivados de amino alcohol y sus actividades terapéuticas
PCT/EP2010/070238 WO2011080139A1 (en) 2009-12-29 2010-12-20 Amino alcohol derivatives and their therapeutic activities
EP10799013.7A EP2519507B1 (en) 2009-12-29 2010-12-20 Amino alcohol derivatives and their therapeutic activities
US13/519,645 US8623900B2 (en) 2009-12-29 2010-12-20 Amino alcohol derivatives and their therapeutic activities
CN201080059714.XA CN102791696B (zh) 2009-12-29 2010-12-20 氨基醇衍生物及其治疗活性

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ITMI2009A002317A IT1397212B1 (it) 2009-12-29 2009-12-29 Derivati di amminoalcoli e loro attivita' terapeutica

Publications (2)

Publication Number Publication Date
ITMI20092317A1 ITMI20092317A1 (it) 2011-06-30
IT1397212B1 true IT1397212B1 (it) 2013-01-04

Family

ID=42238759

Family Applications (1)

Application Number Title Priority Date Filing Date
ITMI2009A002317A IT1397212B1 (it) 2009-12-29 2009-12-29 Derivati di amminoalcoli e loro attivita' terapeutica

Country Status (7)

Country Link
US (1) US8623900B2 (it)
EP (1) EP2519507B1 (it)
JP (1) JP5787899B2 (it)
CN (1) CN102791696B (it)
ES (1) ES2439322T3 (it)
IT (1) IT1397212B1 (it)
WO (1) WO2011080139A1 (it)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2015191533A1 (en) * 2014-06-13 2015-12-17 East Carolina University Methods of using carnosinol and analogs thereof
EP3732165B1 (en) * 2017-12-27 2022-08-17 Flamma S.P.A. Peptide derivatives and therapeutic activity thereof

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5969135A (en) * 1995-11-02 1999-10-19 Icn Pharmaceuticals, Inc. Oligonucleotide analogs with an amino acid or a modified amino alcohol residue
IT1311924B1 (it) * 1999-04-13 2002-03-20 Nicox Sa Composti farmaceutici.
ITMI20061219A1 (it) * 2006-06-23 2007-12-24 Flamma Spa Composti dipeptidici contenenti d-istidina
ITMI20061218A1 (it) * 2006-06-23 2007-12-24 Flamma Spa Derivati pepticidi e loro attivita' terapeutica

Also Published As

Publication number Publication date
EP2519507A1 (en) 2012-11-07
US20120316212A1 (en) 2012-12-13
WO2011080139A1 (en) 2011-07-07
JP2013515753A (ja) 2013-05-09
ITMI20092317A1 (it) 2011-06-30
CN102791696A (zh) 2012-11-21
US8623900B2 (en) 2014-01-07
EP2519507B1 (en) 2013-10-16
CN102791696B (zh) 2015-04-01
ES2439322T3 (es) 2014-01-22
JP5787899B2 (ja) 2015-09-30

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