IT1193529B - ADENOSINIC DERIVATIVES FOR ANTI-INFLAMMATORY AND ANALGESIC ACTIVITIES AND THERAPEUTIC COMPOSITIONS THAT CONTAIN THEM AS AN ACTIVE PRINCIPLE - Google Patents
ADENOSINIC DERIVATIVES FOR ANTI-INFLAMMATORY AND ANALGESIC ACTIVITIES AND THERAPEUTIC COMPOSITIONS THAT CONTAIN THEM AS AN ACTIVE PRINCIPLEInfo
- Publication number
- IT1193529B IT1193529B IT21550/80A IT2155080A IT1193529B IT 1193529 B IT1193529 B IT 1193529B IT 21550/80 A IT21550/80 A IT 21550/80A IT 2155080 A IT2155080 A IT 2155080A IT 1193529 B IT1193529 B IT 1193529B
- Authority
- IT
- Italy
- Prior art keywords
- adenosinic
- inflammatory
- derivatives
- contain
- active principle
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/16—Purine radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pain & Pain Management (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Rheumatology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Priority Applications (29)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT21550/80A IT1193529B (en) | 1980-04-22 | 1980-04-22 | ADENOSINIC DERIVATIVES FOR ANTI-INFLAMMATORY AND ANALGESIC ACTIVITIES AND THERAPEUTIC COMPOSITIONS THAT CONTAIN THEM AS AN ACTIVE PRINCIPLE |
BE0/204529A BE888472A (en) | 1980-04-22 | 1981-04-17 | PHARMACEUTICAL COMPOSITIONS BASED ON ADENOSINE DERIVATIVES AND THEIR PREPARATION, |
JP5930181A JPS56166117A (en) | 1980-04-22 | 1981-04-21 | Antiinflammatory and analgesic adenosine derivative and therapeutical composition containing it as effective component |
NO811346A NO150515C (en) | 1980-04-22 | 1981-04-21 | PROCEDURE FOR PREPARING 5`-DEOXY-5`-METHYLTHIOADENOSINE |
CA000375784A CA1198105A (en) | 1980-04-22 | 1981-04-21 | Adenosine derivatives of antiinflammatory and analgesic activity, and therapeutic compositions which contain them as their active principle |
LU83307A LU83307A1 (en) | 1980-04-22 | 1981-04-21 | ADENOSINE DERIVATIVES WITH ANTI-INFLAMMATORY AND ANALGESIC ACTIVITY, AS WELL AS THERAPEUTIC COMPOSITIONS CONTAINING THESE DERIVATIVES AS ACTIVE INGREDIENT |
ES501539A ES501539A0 (en) | 1980-04-22 | 1981-04-21 | A PROCEDURE FOR THE PREPARATION OF ADENOSINE DERIVATIVES |
SE8102489A SE460198B (en) | 1980-04-22 | 1981-04-21 | PROCEDURES FOR THE PREPARATION OF 5'-DEOXI-5'-METHYLTIOADENOSINE |
AR285020A AR231144A1 (en) | 1980-04-22 | 1981-04-21 | PROCEDURE FOR THE PREPARATION OF 5'-DESOXI-5'-METHYLTICADENOSINE WITH ANTI-INFLAMMATORY AND ANALGESIC ACTIVITY |
DK176481A DK159453C (en) | 1980-04-22 | 1981-04-21 | METHOD FOR PREPARING 5'-DEOXY-5'-METHYLTHIOADENOSINE |
MX10149781U MX6553E (en) | 1980-04-22 | 1981-04-22 | PROCEDURE FOR PREPARING 5'-DESOXI-5'-METHYLTHIOADENOSINE |
CH4716/84A CH650514A5 (en) | 1980-04-22 | 1981-04-22 | METHOD FOR PRODUCING 5'-DESOXY-5'-METHYLTHIOADENOSINE. |
CH263281A CH645544A5 (en) | 1980-04-22 | 1981-04-22 | THERAPEUTIC, ADENOSINE DERIVATIVES WITH ANTI-INFLAMMATORY, ANALGETIC AND ANTIPYRETIC EFFECTIVENESS. |
GB8112428A GB2074446B (en) | 1980-04-22 | 1981-04-22 | Adenosine derivatives of antiinflammatory and analgesic activity and therapeutic compositions containing them |
FR8107992A FR2491761A1 (en) | 1980-04-22 | 1981-04-22 | ADENOSINE DERIVATIVES WITH ANTI-INFLAMMATORY AND ANALGESIC ACTIVITY AND THERAPEUTIC COMPOSITIONS CONTAINING THE SAME AS ACTIVE INGREDIENTS |
FI811249A FI70227C (en) | 1980-04-22 | 1981-04-22 | ADJUSTMENT OF THERAPEUTIC ADJUSTMENT |
NL8101984A NL192111C (en) | 1980-04-22 | 1981-04-22 | Drug preparation with anti-inflammatory effect. |
DE19813116067 DE3116067A1 (en) | 1980-04-22 | 1981-04-22 | THERAPEUTIC COMPOSITIONS WITH PAIN-RELEASING AND ANTI-INFLAMMATORY PROPERTIES THAT CONTAIN ADENOS IN DERIVATIVES AS ACTIVE INGREDIENTS |
ES511039A ES8306378A1 (en) | 1980-04-22 | 1982-04-01 | Adenosine derivatives of antiinflammatory and analgesic activity and therapeutic compositions containing them |
GB08321947A GB2144409B (en) | 1980-04-22 | 1983-08-15 | Preparation of 5'-deoxy-5'-methylthioadenosine |
FI834113A FI68629C (en) | 1980-04-22 | 1983-11-09 | FOERFARANDE FOER FRAMSTAELLNING AV 5'-DEOXY-5'-METHYLTIOADENOSIN |
DK25184A DK163518C (en) | 1980-04-22 | 1984-01-20 | ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY EFFECTIVE ADENOSIN DERIVATIVES |
NO840343A NO157863C (en) | 1980-04-22 | 1984-01-30 | ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE ADENOSIN DERIVATIVES. |
GB08413454A GB2144038B (en) | 1980-04-22 | 1984-05-25 | Adenosine derivatives of anti-inflammatory and analgesic activity and therapeutic compositions containing them |
CA000490761A CA1209915A (en) | 1980-04-22 | 1985-09-13 | Adenosine derivatives of antiinflammatory and analgesic activity, and therapeutic compositions which contain them as their active principle |
SE8700914A SE464635B (en) | 1980-04-22 | 1987-03-04 | USE OF AN ADENOSIN DERIVATIVE FOR THE PREPARATION OF A MEDICINE FOR TREATMENT OF INFLAMMATION, PAIN AND FEBRUARY |
SE8700913A SE466238B (en) | 1980-04-22 | 1987-03-04 | THERAPEUTIC COMPOSITION CONTAINING ADENOSIN DERIVATIVES |
JP1022771A JPH01301692A (en) | 1980-04-22 | 1989-02-02 | Novel production of 5'-deoxy-5'- methylthioadenosine |
MX9203630A MX9203630A (en) | 1980-04-22 | 1992-06-26 | DERIVATIVES OF ADENOSINE AND THERAPEUTIC COMPOSITIONS THAT CONTAIN THEM AS AN ACTIVE PRINCIPLE OF ANALGESIC AND ANTI-INFLAMMATORY ACTIVITY. |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT21550/80A IT1193529B (en) | 1980-04-22 | 1980-04-22 | ADENOSINIC DERIVATIVES FOR ANTI-INFLAMMATORY AND ANALGESIC ACTIVITIES AND THERAPEUTIC COMPOSITIONS THAT CONTAIN THEM AS AN ACTIVE PRINCIPLE |
Publications (2)
Publication Number | Publication Date |
---|---|
IT8021550A0 IT8021550A0 (en) | 1980-04-22 |
IT1193529B true IT1193529B (en) | 1988-07-08 |
Family
ID=11183457
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IT21550/80A IT1193529B (en) | 1980-04-22 | 1980-04-22 | ADENOSINIC DERIVATIVES FOR ANTI-INFLAMMATORY AND ANALGESIC ACTIVITIES AND THERAPEUTIC COMPOSITIONS THAT CONTAIN THEM AS AN ACTIVE PRINCIPLE |
Country Status (17)
Country | Link |
---|---|
JP (2) | JPS56166117A (en) |
AR (1) | AR231144A1 (en) |
BE (1) | BE888472A (en) |
CA (1) | CA1198105A (en) |
CH (2) | CH645544A5 (en) |
DE (1) | DE3116067A1 (en) |
DK (1) | DK159453C (en) |
ES (2) | ES501539A0 (en) |
FI (1) | FI70227C (en) |
FR (1) | FR2491761A1 (en) |
GB (3) | GB2074446B (en) |
IT (1) | IT1193529B (en) |
LU (1) | LU83307A1 (en) |
MX (1) | MX9203630A (en) |
NL (1) | NL192111C (en) |
NO (1) | NO150515C (en) |
SE (3) | SE460198B (en) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IT1177373B (en) * | 1984-12-06 | 1987-08-26 | Bioresearch Spa | SALTS OF 5'-METHYLLIUM-5'-DEOXYDENOSINE WITH LONG ALCHYLIC CHAIN SULPHONIC ACIDS |
IT1227049B (en) * | 1988-07-29 | 1991-03-14 | Bioresearch Spa | USE OF ADENOSINIC DERIVATIVES FOR THE PREPARATION OF PHARMACEUTICAL COMPOSITIONS HAVING IMMUNOSTIMULATING ACTIVITIES. |
JPH0497287A (en) * | 1990-08-10 | 1992-03-30 | Nec Ic Microcomput Syst Ltd | Picture display integrated circuit |
ES2259552B1 (en) * | 2005-03-17 | 2007-06-16 | Proyecto De Biomedicina Cima, S.L. | EMPLOYMENT OF 5'-METHYLTIOENENINE (MTA) IN THE PREVENTION AND / OR TREATMENT OF AUTOIMMUNE DISEASES AND / OR REPLACEMENT OF TRANSPLANTS. |
WO2006097547A1 (en) * | 2005-03-17 | 2006-09-21 | Proyecto De Biomedicina Cima S.L. | Use of 5'-methylthioadenosine (mta) in the prevention and/or treatment of autoimmune diseases and/or transplant rejection |
DE102010027595A1 (en) * | 2010-07-23 | 2012-01-26 | Helmut Vorbrüggen | Clinical application of adenosine derivative, preferably (dihydroxyphenyl)ethyl-amino-purin-9-yl-(hydroxymethyl)oxolane-diol, for reducing body temperature during impending ischemia of brain vessels, which occur during heart attacks |
DE102011005232A1 (en) * | 2011-03-08 | 2012-09-13 | AristoCon GmbH & Co. KG | Adenosine and its derivatives for use in pain therapy |
WO2014163152A1 (en) * | 2013-04-05 | 2014-10-09 | ライオン株式会社 | Non-rem sleep-promoting agent, deep sleep-promoting agent and natural sleep-inducing agent |
CN105101974B (en) * | 2013-04-05 | 2018-07-03 | 狮王株式会社 | Internal composition |
WO2014163151A1 (en) * | 2013-04-05 | 2014-10-09 | ライオン株式会社 | Yeast culture, and composition for internal application |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE1259341B (en) * | 1962-12-22 | 1968-01-25 | Boehringer & Soehne Gmbh | Process for the preparation of new 5'-sulfoxides of nucleosides |
DE1545645A1 (en) * | 1965-12-06 | 1969-08-21 | Boehringer Mannheim Gmbh | Process for the preparation of disubstituted adenosine derivatives |
FR2252405B1 (en) * | 1973-11-27 | 1978-04-28 | Ajinomoto Kk | |
FR2313937A1 (en) * | 1975-06-09 | 1977-01-07 | Anvar | DRUG BASED ON 5 'THIOETHERS OF ADENOSINE |
FR2424027A1 (en) * | 1978-04-28 | 1979-11-23 | Merieux Inst | NEW MEDICINAL PRODUCT, IN PARTICULAR SEDATIVE AND SLEEP INDUCER AND PHARMACEUTICAL COMPOSITIONS CONTAINING IT |
-
1980
- 1980-04-22 IT IT21550/80A patent/IT1193529B/en active
-
1981
- 1981-04-17 BE BE0/204529A patent/BE888472A/en not_active IP Right Cessation
- 1981-04-21 JP JP5930181A patent/JPS56166117A/en active Granted
- 1981-04-21 SE SE8102489A patent/SE460198B/en not_active IP Right Cessation
- 1981-04-21 NO NO811346A patent/NO150515C/en unknown
- 1981-04-21 CA CA000375784A patent/CA1198105A/en not_active Expired
- 1981-04-21 LU LU83307A patent/LU83307A1/en unknown
- 1981-04-21 DK DK176481A patent/DK159453C/en not_active IP Right Cessation
- 1981-04-21 ES ES501539A patent/ES501539A0/en active Granted
- 1981-04-21 AR AR285020A patent/AR231144A1/en active
- 1981-04-22 CH CH263281A patent/CH645544A5/en not_active IP Right Cessation
- 1981-04-22 FR FR8107992A patent/FR2491761A1/en active Granted
- 1981-04-22 CH CH4716/84A patent/CH650514A5/en not_active IP Right Cessation
- 1981-04-22 FI FI811249A patent/FI70227C/en not_active IP Right Cessation
- 1981-04-22 GB GB8112428A patent/GB2074446B/en not_active Expired
- 1981-04-22 DE DE19813116067 patent/DE3116067A1/en active Granted
- 1981-04-22 NL NL8101984A patent/NL192111C/en not_active IP Right Cessation
-
1982
- 1982-04-01 ES ES511039A patent/ES8306378A1/en not_active Expired
-
1983
- 1983-08-15 GB GB08321947A patent/GB2144409B/en not_active Expired
-
1984
- 1984-05-25 GB GB08413454A patent/GB2144038B/en not_active Expired
-
1987
- 1987-03-04 SE SE8700914A patent/SE464635B/en not_active IP Right Cessation
- 1987-03-04 SE SE8700913A patent/SE466238B/en not_active IP Right Cessation
-
1989
- 1989-02-02 JP JP1022771A patent/JPH01301692A/en active Granted
-
1992
- 1992-06-26 MX MX9203630A patent/MX9203630A/en unknown
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
TA | Fee payment date (situation as of event date), data collected since 19931001 |
Effective date: 19960429 |