IT1142620B - Derivati piperazinici 1,4-bisostituiti e processo per la loro preparazione - Google Patents

Derivati piperazinici 1,4-bisostituiti e processo per la loro preparazione

Info

Publication number
IT1142620B
IT1142620B IT25742/81A IT2574281A IT1142620B IT 1142620 B IT1142620 B IT 1142620B IT 25742/81 A IT25742/81 A IT 25742/81A IT 2574281 A IT2574281 A IT 2574281A IT 1142620 B IT1142620 B IT 1142620B
Authority
IT
Italy
Prior art keywords
piperazinic
bisubstituted
derivatives
preparation
piperazinic derivatives
Prior art date
Application number
IT25742/81A
Other languages
English (en)
Other versions
IT8125742A0 (it
Inventor
Irikura Tsutomu
Nishino Keigo
Okamura Kyuya
Taga Fukutaro
Original Assignee
Kyorin Seiyaku Kk
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kyorin Seiyaku Kk filed Critical Kyorin Seiyaku Kk
Publication of IT8125742A0 publication Critical patent/IT8125742A0/it
Application granted granted Critical
Publication of IT1142620B publication Critical patent/IT1142620B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D263/00Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/56Benzoxazoles; Hydrogenated benzoxazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D235/14Radicals substituted by nitrogen atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Neurosurgery (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pain & Pain Management (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
IT25742/81A 1980-12-23 1981-12-21 Derivati piperazinici 1,4-bisostituiti e processo per la loro preparazione IT1142620B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP55182632A JPS57106663A (en) 1980-12-23 1980-12-23 1,4-disubstituted piperazine derivative and its preparation

Publications (2)

Publication Number Publication Date
IT8125742A0 IT8125742A0 (it) 1981-12-21
IT1142620B true IT1142620B (it) 1986-10-08

Family

ID=16121678

Family Applications (1)

Application Number Title Priority Date Filing Date
IT25742/81A IT1142620B (it) 1980-12-23 1981-12-21 Derivati piperazinici 1,4-bisostituiti e processo per la loro preparazione

Country Status (10)

Country Link
JP (1) JPS57106663A (it)
KR (1) KR830007608A (it)
AU (1) AU7877481A (it)
BE (1) BE891580A (it)
DE (1) DE3151123A1 (it)
FR (1) FR2496661A1 (it)
GB (1) GB2091255A (it)
IT (1) IT1142620B (it)
SE (1) SE8107680L (it)
ZA (1) ZA818900B (it)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4835154A (en) * 1987-06-01 1989-05-30 Smithkline Beckman Corporation 1-aralykyl-5-piperazinylmethyl-2-mercaptoimidazoles and 2-alkylthioimidazoles and their use as dopamine-βhydroxylase inhibitors
US5149700A (en) * 1990-05-30 1992-09-22 American Home Products Corporation Substituted arylsulfonamides and benzamides
AU3248600A (en) * 1999-03-03 2000-09-21 Merck & Co., Inc. Inhibitors of prenyl-protein transferases

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2297045A1 (fr) * 1975-01-10 1976-08-06 Delalande Sa Nouveaux (aroyl-2' eth-1' yl)-1 (acetamido-4'' piperazin-1'' yl methyl)-2 benzimidazoles a proprietes antisecretoire gastrique et antiulcereuse
YU39992B (en) * 1976-04-02 1985-06-30 Janssen Pharmaceutica Nv Process for obtaining new piperazine and piperidine derivatives

Also Published As

Publication number Publication date
JPS57106663A (en) 1982-07-02
KR830007608A (ko) 1983-11-04
IT8125742A0 (it) 1981-12-21
BE891580A (fr) 1982-04-16
FR2496661A1 (fr) 1982-06-25
SE8107680L (sv) 1982-06-24
DE3151123A1 (de) 1982-08-12
AU7877481A (en) 1982-07-01
ZA818900B (en) 1982-12-29
GB2091255A (en) 1982-07-28

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