IL148548A0 - Bicyclic vasopressin agonists - Google Patents

Bicyclic vasopressin agonists

Info

Publication number
IL148548A0
IL148548A0 IL14854800A IL14854800A IL148548A0 IL 148548 A0 IL148548 A0 IL 148548A0 IL 14854800 A IL14854800 A IL 14854800A IL 14854800 A IL14854800 A IL 14854800A IL 148548 A0 IL148548 A0 IL 148548A0
Authority
IL
Israel
Prior art keywords
alkyl
bicyclic
vasopressin agonists
agonists
independently
Prior art date
Application number
IL14854800A
Other languages
English (en)
Original Assignee
Ferring Bv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ferring Bv filed Critical Ferring Bv
Publication of IL148548A0 publication Critical patent/IL148548A0/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D223/00Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
    • C07D223/14Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D223/16Benzazepines; Hydrogenated benzazepines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/10Drugs for disorders of the urinary system of the bladder
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/04Antihaemorrhagics; Procoagulants; Haemostatic agents; Antifibrinolytic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/12Antidiuretics, e.g. drugs for diabetes insipidus
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D267/00Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D267/02Seven-membered rings
    • C07D267/08Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D267/12Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D267/14Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Diabetes (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
IL14854800A 1999-10-20 2000-10-20 Bicyclic vasopressin agonists IL148548A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB9924836A GB2355454A (en) 1999-10-20 1999-10-20 Antidiuretic agents
PCT/GB2000/004055 WO2001029005A1 (en) 1999-10-20 2000-10-20 Bicyclic vasopressin agonists

Publications (1)

Publication Number Publication Date
IL148548A0 true IL148548A0 (en) 2002-09-12

Family

ID=10863070

Family Applications (2)

Application Number Title Priority Date Filing Date
IL14854800A IL148548A0 (en) 1999-10-20 2000-10-20 Bicyclic vasopressin agonists
IL148548A IL148548A (en) 1999-10-20 2002-03-06 Vasopressin agonists and pharmaceutics containing them for the treatment of hyperuriaemia

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL148548A IL148548A (en) 1999-10-20 2002-03-06 Vasopressin agonists and pharmaceutics containing them for the treatment of hyperuriaemia

Country Status (22)

Country Link
US (1) US6664249B1 (de)
EP (1) EP1226122B1 (de)
JP (1) JP4694747B2 (de)
KR (1) KR100725555B1 (de)
CN (1) CN1144788C (de)
AT (1) ATE284871T1 (de)
AU (1) AU777092B2 (de)
CA (1) CA2387886A1 (de)
CZ (1) CZ304069B6 (de)
DE (1) DE60016786T2 (de)
ES (1) ES2234684T3 (de)
GB (1) GB2355454A (de)
HK (1) HK1044155B (de)
HU (1) HU229357B1 (de)
IL (2) IL148548A0 (de)
MX (1) MXPA02003779A (de)
NO (1) NO322920B1 (de)
NZ (1) NZ517611A (de)
PL (1) PL206211B1 (de)
PT (1) PT1226122E (de)
RU (1) RU2254332C2 (de)
WO (1) WO2001029005A1 (de)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0000079D0 (en) * 2000-01-05 2000-02-23 Ferring Bv Novel antidiuretic agents
GB0015601D0 (en) * 2000-06-26 2000-08-16 Ferring Bv Novel antidiuretic agents
GB0210397D0 (en) 2002-05-07 2002-06-12 Ferring Bv Pharmaceutical formulations
ES2260563T3 (es) * 2003-11-13 2006-11-01 Ferring B.V. Paquete de blister y forma farmaceutica solida para ello.
EP1632494A1 (de) * 2004-08-24 2006-03-08 Ferring B.V. Vasopressin v1a antagonisten
SE528446C2 (sv) * 2006-03-02 2006-11-14 Ferring Int Ct Sa Farmaceutisk sammansättning innefattande desmopressin, kiseldioxid och stärkelse
CA2695634C (en) 2007-08-06 2018-01-23 Serenity Pharmaceuticals Corporation Methods and devices for desmopressin drug delivery
DK3225250T3 (da) 2008-05-21 2019-11-04 Ferring Bv Orodispersibel desmopressin til forlængelse af den indledende søvnperiode, som ikke forstyrres af nykturi
US11963995B2 (en) 2008-05-21 2024-04-23 Ferring B.V. Methods comprising desmopressin
US20100286045A1 (en) 2008-05-21 2010-11-11 Bjarke Mirner Klein Methods comprising desmopressin
CN102942558B (zh) * 2012-05-18 2014-04-16 天津药物研究院 一种苯并氮杂卓衍生物的制备方法

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2905909B2 (ja) * 1991-04-19 1999-06-14 大塚製薬株式会社 バソプレシン拮抗剤
DE69026708T2 (de) * 1989-10-20 1997-04-03 Otsuka Pharma Co Ltd Benzoheterozyklische verbindungen
US5753677A (en) * 1989-10-20 1998-05-19 Otsuka Pharmaceutical Co., Ltd. Benzoheterocyclic compounds
TW198715B (de) * 1991-04-19 1993-01-21 Dtsuka Seiyaku Kk
JPH05320135A (ja) * 1992-05-19 1993-12-03 Yamanouchi Pharmaceut Co Ltd テトラヒドロベンズアゼピン誘導体
WO1994004525A1 (en) * 1992-08-20 1994-03-03 Otsuka Pharmaceutical Company, Limited Benzoheterocyclic compounds as oxytocin and vasopressin antagonists
TW270927B (de) 1992-10-16 1996-02-21 Otsuka Pharma Co Ltd
JP2913082B2 (ja) * 1992-10-16 1999-06-28 大塚製薬株式会社 バソプレシン拮抗剤及びオキシトシン拮抗剤
WO1994012476A1 (en) 1992-11-25 1994-06-09 Yamanouchi Pharmaceutical Co., Ltd. Benzanilide derivative
AU6219994A (en) 1993-03-11 1994-09-26 Yamanouchi Pharmaceutical Co., Ltd. Compound with vasopressin antagonism
JP2926335B2 (ja) * 1997-06-13 1999-07-28 大塚製薬株式会社 医薬組成物

Also Published As

Publication number Publication date
EP1226122B1 (de) 2004-12-15
KR20020029794A (ko) 2002-04-19
DE60016786D1 (de) 2005-01-20
HUP0203622A2 (hu) 2003-02-28
DE60016786T2 (de) 2005-12-22
KR100725555B1 (ko) 2007-06-08
PT1226122E (pt) 2005-04-29
NO20021879L (no) 2002-04-19
HU229357B1 (en) 2013-11-28
NO20021879D0 (no) 2002-04-19
HUP0203622A3 (en) 2005-01-28
NZ517611A (en) 2002-11-26
NO322920B1 (no) 2006-12-18
EP1226122A1 (de) 2002-07-31
CN1382125A (zh) 2002-11-27
HK1044155A1 (en) 2002-10-11
RU2254332C2 (ru) 2005-06-20
CZ20021339A3 (cs) 2002-09-11
PL354044A1 (en) 2003-12-15
CA2387886A1 (en) 2001-04-26
GB2355454A (en) 2001-04-25
ES2234684T3 (es) 2005-07-01
US6664249B1 (en) 2003-12-16
AU1037401A (en) 2001-04-30
HK1044155B (zh) 2005-05-06
AU777092B2 (en) 2004-09-30
ATE284871T1 (de) 2005-01-15
IL148548A (en) 2007-02-11
JP2003512356A (ja) 2003-04-02
GB9924836D0 (en) 1999-12-22
CZ304069B6 (cs) 2013-09-18
JP4694747B2 (ja) 2011-06-08
WO2001029005A1 (en) 2001-04-26
CN1144788C (zh) 2004-04-07
PL206211B1 (pl) 2010-07-30
MXPA02003779A (es) 2002-09-30

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Legal Events

Date Code Title Description
FF Patent granted
KB Patent renewed