IL133900A0 - Process for the preparation of intermediates for 3-amino-2-mercaptobenzoic acid derivatives - Google Patents

Process for the preparation of intermediates for 3-amino-2-mercaptobenzoic acid derivatives

Info

Publication number
IL133900A0
IL133900A0 IL13390000A IL13390000A IL133900A0 IL 133900 A0 IL133900 A0 IL 133900A0 IL 13390000 A IL13390000 A IL 13390000A IL 13390000 A IL13390000 A IL 13390000A IL 133900 A0 IL133900 A0 IL 133900A0
Authority
IL
Israel
Prior art keywords
substituted
unsubstituted
compounds
preparation
carbon atoms
Prior art date
Application number
IL13390000A
Other languages
English (en)
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Priority to IL13390000A priority Critical patent/IL133900A0/xx
Publication of IL133900A0 publication Critical patent/IL133900A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C319/00—Preparation of thiols, sulfides, hydropolysulfides or polysulfides
    • C07C319/02—Preparation of thiols, sulfides, hydropolysulfides or polysulfides of thiols
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C319/00—Preparation of thiols, sulfides, hydropolysulfides or polysulfides
    • C07C319/02—Preparation of thiols, sulfides, hydropolysulfides or polysulfides of thiols
    • C07C319/12—Preparation of thiols, sulfides, hydropolysulfides or polysulfides of thiols by reactions not involving the formation of mercapto groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
    • C07C323/62—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atom of at least one of the thio groups bound to a carbon atom of a six-membered aromatic ring of the carbon skeleton
    • C07C323/63—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atom of at least one of the thio groups bound to a carbon atom of a six-membered aromatic ring of the carbon skeleton the carbon skeleton being further substituted by nitrogen atoms, not being part of nitro or nitroso groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C327/00—Thiocarboxylic acids
    • C07C327/20—Esters of monothiocarboxylic acids
    • C07C327/26—Esters of monothiocarboxylic acids having carbon atoms of esterified thiocarboxyl groups bound to carbon atoms of six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C335/00—Thioureas, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
    • C07C335/04—Derivatives of thiourea
    • C07C335/16—Derivatives of thiourea having nitrogen atoms of thiourea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C335/22—Derivatives of thiourea having nitrogen atoms of thiourea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by carboxyl groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62—Benzothiazoles
    • C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D277/82—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/14—Thiadiazoles; Hydrogenated thiadiazoles condensed with carbocyclic rings or ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Cephalosporin Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
IL13390000A 1995-12-21 2000-01-06 Process for the preparation of intermediates for 3-amino-2-mercaptobenzoic acid derivatives IL133900A0 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
IL13390000A IL133900A0 (en) 1995-12-21 2000-01-06 Process for the preparation of intermediates for 3-amino-2-mercaptobenzoic acid derivatives

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
CH363795 1995-12-21
IL11981996A IL119819A (en) 1995-12-21 1996-12-12 Processes for the preparation of derivatives of acid 3 - amino - 2 - Mercaptobenzoic, their use in the preparation of microbial and plant-killing agents and a number of such new compounds
US08/770,353 US5770758A (en) 1995-12-21 1996-12-20 3-amino-2-mercaptobenzoic acid derivatives and processes for their preparation
IL13390000A IL133900A0 (en) 1995-12-21 2000-01-06 Process for the preparation of intermediates for 3-amino-2-mercaptobenzoic acid derivatives

Publications (1)

Publication Number Publication Date
IL133900A0 true IL133900A0 (en) 2001-04-30

Family

ID=25693502

Family Applications (3)

Application Number Title Priority Date Filing Date
IL13390096A IL133900A (en) 1995-12-21 1996-12-12 Derivatives of benzothiazole and the process for their preparation
IL11981996A IL119819A (en) 1995-12-21 1996-12-12 Processes for the preparation of derivatives of acid 3 - amino - 2 - Mercaptobenzoic, their use in the preparation of microbial and plant-killing agents and a number of such new compounds
IL13390000A IL133900A0 (en) 1995-12-21 2000-01-06 Process for the preparation of intermediates for 3-amino-2-mercaptobenzoic acid derivatives

Family Applications Before (2)

Application Number Title Priority Date Filing Date
IL13390096A IL133900A (en) 1995-12-21 1996-12-12 Derivatives of benzothiazole and the process for their preparation
IL11981996A IL119819A (en) 1995-12-21 1996-12-12 Processes for the preparation of derivatives of acid 3 - amino - 2 - Mercaptobenzoic, their use in the preparation of microbial and plant-killing agents and a number of such new compounds

Country Status (21)

Country Link
US (1) US5770758A (xx)
EP (1) EP0780372B3 (xx)
JP (1) JP4217924B2 (xx)
KR (1) KR100470887B1 (xx)
CN (2) CN1163491C (xx)
AT (1) ATE208760T1 (xx)
AU (1) AU713526B2 (xx)
BR (1) BR9606092A (xx)
CA (1) CA2193460C (xx)
CZ (1) CZ291857B6 (xx)
DE (1) DE69616956T3 (xx)
DK (1) DK0780372T3 (xx)
ES (1) ES2168121T7 (xx)
HU (1) HU221600B (xx)
IL (3) IL133900A (xx)
MX (2) MXPA02000515A (xx)
PL (1) PL187885B1 (xx)
PT (1) PT780372E (xx)
RU (1) RU2176241C2 (xx)
SK (1) SK283840B6 (xx)
ZA (1) ZA9610774B (xx)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6002013A (en) * 1995-12-21 1999-12-14 Novartis Corporation 3-amino-2-mercaptobenzoic acid derivatives and processes for their preparation
GB9724586D0 (en) * 1997-11-20 1998-01-21 Rhone Poulenc Agriculture New herbicides
WO2004029050A1 (en) 2002-09-25 2004-04-08 Memory Pharmaceuticals Corporation Indazoles, benzothiazoles, and benzoisothiazoles, and preparation and uses thereof
DE10313887A1 (de) * 2003-03-27 2004-10-28 Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. Verfahren zum selektiven Gewinnen von Gold aus goldhaltigen Materialien
EP2368554B1 (en) 2003-04-08 2014-12-24 Progenics Pharmaceuticals, Inc. Pharmaceutical formulations containing methylnaltrexone
KR20070007759A (ko) * 2003-07-10 2007-01-16 아칠리온 파르마세우티칼스 인코포레이티드 바이러스 복제 억제제로서 유용한 치환된 아릴티오우레아유도체
CA2560741C (en) 2004-03-25 2013-08-06 Memory Pharmaceuticals Corporation Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, and preparation and uses thereof
AR057325A1 (es) 2005-05-25 2007-11-28 Progenics Pharm Inc Sintesis de (s)-n-metilnaltrexona, composiciones farmaceuticas y usos
AR057035A1 (es) 2005-05-25 2007-11-14 Progenics Pharm Inc SíNTESIS DE (R)-N-METILNALTREXONA, COMPOSICIONES FARMACÉUTICAS Y USOS
JP2009528373A (ja) * 2006-03-02 2009-08-06 マリンクロッド・インコーポレイテッド チアジアゾール化合物および光線療法のためのその使用
EP3263571B2 (en) 2007-03-29 2023-08-23 Progenics Pharmaceuticals, Inc. Crystal form of (r)-n-methylnaltrexone bromide and uses thereof
PE20130480A1 (es) 2007-03-29 2013-05-08 Progenics Pharm Inc Compuestos heterociclicos como antagonistas del receptor opioide periferico
MX2009010515A (es) 2007-03-29 2009-10-19 Wyeth Corp Antagonistas del receptor opioide periferico y usos de los mismos.
CA2713568C (en) 2008-02-06 2016-09-20 Progenics Pharmaceuticals, Inc. Preparation and use of (r),(r)-2,2'-bis-methylnaltrexone
CA2676881C (en) 2008-09-30 2017-04-25 Wyeth Peripheral opioid receptor antagonists and uses thereof
CN101492429B (zh) * 2008-12-10 2010-12-15 上海泰禾(集团)有限公司 一种苯并-[1，2，3]-噻二唑-7-甲酸三氟乙酯的提纯方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4150140A (en) * 1976-12-23 1979-04-17 The Upjohn Company Benzothiazolyl oxanic acids, esters and salts
DE2757924A1 (de) * 1977-12-24 1979-07-05 Hoechst Ag Verfahren zur herstellung von vinylchlorid-polymerisaten
DE3601286A1 (de) * 1986-01-17 1987-07-23 Consiglio Nazionale Ricerche Sammelmittel fuer die selektive flotation von blei- und zinkerzen und verfahren zu deren herstellung
DE19775050I2 (de) * 1987-08-21 2010-12-16 Syngenta Participations Ag Benzothiadiazole und ihre Verwendung in Verfahren und Mitteln gegen Pflanzenkrankheiten.
DE59003043D1 (de) * 1989-02-21 1993-11-18 Ciba Geigy Mittel zum Schutz von Pflanzen gegen Krankheiten.
EP0529600B1 (de) 1991-08-30 1996-11-06 Hoechst Aktiengesellschaft Verfahren zur Herstellung von 2-Aminobenzthiazolen
JPH0690518A (ja) * 1992-09-09 1994-03-29 Toshiba Corp 地絡継電器
JP3310104B2 (ja) * 1994-04-04 2002-07-29 三新化学工業株式会社 ２−アミノチオフェノール類の製造方法
BR9509373A (pt) * 1994-10-17 1998-07-07 Novartis Ag Processo para a preparação de 3- aminobenzonitrilas substituídas

Also Published As

Publication number Publication date
JPH09235279A (ja) 1997-09-09
CN1156722A (zh) 1997-08-13
HU221600B (hu) 2002-11-28
DE69616956T2 (de) 2002-06-20
PL317601A1 (en) 1997-06-23
HUP9603527A3 (en) 1999-04-28
EP0780372B3 (en) 2013-05-22
EP0780372A3 (en) 1997-09-17
AU713526C (en) 1997-06-26
ZA9610774B (en) 1997-06-30
DE69616956T3 (de) 2014-01-30
SK283840B6 (sk) 2004-03-02
KR100470887B1 (ko) 2005-03-14
DK0780372T3 (da) 2002-03-11
ES2168121T3 (es) 2002-06-01
CZ291857B6 (cs) 2003-06-18
JP4217924B2 (ja) 2009-02-04
BR9606092A (pt) 1998-09-01
DE69616956D1 (de) 2001-12-20
EP0780372A2 (en) 1997-06-25
AU7640496A (en) 1997-06-26
US5770758A (en) 1998-06-23
CZ377396A3 (en) 1997-07-16
CN1078888C (zh) 2002-02-06
HU9603527D0 (en) 1997-02-28
SK163696A3 (en) 1997-10-08
IL119819A (en) 2004-07-25
PT780372E (pt) 2002-04-29
CA2193460C (en) 2007-03-27
MXPA02000515A (es) 2002-09-17
IL119819A0 (en) 1997-03-18
CN1163491C (zh) 2004-08-25
HUP9603527A2 (en) 1997-09-29
CN1392144A (zh) 2003-01-22
ES2168121T7 (es) 2013-09-24
EP0780372B1 (en) 2001-11-14
AU713526B2 (en) 1999-12-02
MX9606665A (es) 1997-06-28
CA2193460A1 (en) 1997-06-22
ATE208760T1 (de) 2001-11-15
RU2176241C2 (ru) 2001-11-27
IL133900A (en) 2004-07-25
PL187885B1 (pl) 2004-10-29

Similar Documents

Publication Publication Date Title
IL133900A0 (en) Process for the preparation of intermediates for 3-amino-2-mercaptobenzoic acid derivatives
EP0484094A3 (en) Azasteroid compounds for the treatment of prostatic hypertrophy, their preparation and use
HU9401943D0 (en) Process for producing amide and urea derivatives and compositions containing them
WO1988000042A1 (en) New 5-alkoxy-2,4-diamino-alkyl benzols, and hair tinting means using them
NZ243022A (en) Substituted pyrrolidinylthio carbapenem derivatives
IL103361A0 (en) Novel 17beta-substituted aza-androstane derivatives
AU3381389A (en) Derivative of caffeic acid and pharmaceutical composition containing the same
NZ226222A (en) Preparation of n-alkylated alpha-aminodiacids and esters thereof, and use of those compounds in the synthesis of n-heterocyclic dipeptides
AU627631B2 (en) Pyrimidone derivatives and analogs in the treatment of asthma or certain skin disorders
MX170732B (es) Composicion de derivados de succinimida y su uso
SG49692G (en) Phenylacetic acid amides having antiinflammatory and analgesic activity
EP0315996A3 (en) Optically active compound, process for producing same and liquid crystal composition containing same
DE2962829D1 (en) Isomerisation of 3-azabicyclo(3.1.0)hexane derivatives
HUT47923A (en) Process for production of new derivatives of naphtotiazephin and medical compositions containing these substances
EP0373881A3 (en) Process for preparing optically active 2-oxoimidazolidine derivatives

Legal Events

Date Code Title Description
HP Change in proprietorship
FF Patent granted