IL124908A - Processes for the preparation of 5-pyrimidinyl substituted imidazoles and aminoalkyl carbonyl imidazole intermediates thereor - Google Patents

Processes for the preparation of 5-pyrimidinyl substituted imidazoles and aminoalkyl carbonyl imidazole intermediates thereor

Info

Publication number: IL124908A
Authority: IL; Israel
Prior art keywords: thereor; processes; preparation; substituted imidazoles; pyrimidinyl substituted
Prior art date: 1995-12-22

Application number

IL12490896A

Other languages

English (en)

Other versions

IL124908A0 (en

Original Assignee

Smithkline Beecham Corp

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-12-22

Filing date

1996-12-20

Publication date

2003-05-29

1996-12-20 Application filed by Smithkline Beecham Corp filed Critical Smithkline Beecham Corp

1996-12-20 Priority to IL14351796A priority Critical patent/IL143517A/xx

1999-01-26 Publication of IL124908A0 publication Critical patent/IL124908A0/xx

2003-05-29 Publication of IL124908A publication Critical patent/IL124908A/xx

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Epoxy Resins (AREA)

IL12490896A 1995-12-22 1996-12-20 Processes for the preparation of 5-pyrimidinyl substituted imidazoles and aminoalkyl carbonyl imidazole intermediates thereor IL124908A (en)

Priority Applications (1)

Application Number	Priority Date	Filing Date	Title
IL14351796A IL143517A (en)	1995-12-22	1996-12-20	Imidazole compounds

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US909895P	1995-12-22	1995-12-22
PCT/US1996/020599 WO1997023479A1 (en)	1995-12-22	1996-12-20	Novel synthesis

Publications (2)

Publication Number	Publication Date
IL124908A0 IL124908A0 (en)	1999-01-26
IL124908A true IL124908A (en)	2003-05-29

Family

ID=21735553

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
IL12490896A IL124908A (en)	1995-12-22	1996-12-20	Processes for the preparation of 5-pyrimidinyl substituted imidazoles and aminoalkyl carbonyl imidazole intermediates thereor
IL14351796A IL143517A (en)	1995-12-22	1996-12-20	Imidazole compounds

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
IL14351796A IL143517A (en)	1995-12-22	1996-12-20	Imidazole compounds

Country Status (18)

Country	Link
US (3)	US5917043A (xx)
EP (1)	EP1019393A1 (xx)
JP (1)	JP3245175B2 (xx)
KR (1)	KR19990076625A (xx)
CN (1)	CN1209128A (xx)
AR (3)	AR004405A1 (xx)
AU (1)	AU704500B2 (xx)
BR (1)	BR9612187A (xx)
CZ (1)	CZ198598A3 (xx)
HU (1)	HUP9902466A3 (xx)
IL (2)	IL124908A (xx)
NO (1)	NO982850L (xx)
NZ (1)	NZ326574A (xx)
PL (1)	PL327311A1 (xx)
TR (1)	TR199801121T2 (xx)
TW (1)	TW434236B (xx)
WO (1)	WO1997023479A1 (xx)
ZA (1)	ZA9610687B (xx)

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HUP9902460A3 (en) *	1996-01-11	2000-03-28	Smithkline Beecham Corp	Novel substituted imidazole compounds, their use, method for their preparation and pharmaceutical compositions containing them
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US6514977B1 (en)	1997-05-22	2003-02-04	G.D. Searle & Company	Substituted pyrazoles as p38 kinase inhibitors
US6979686B1 (en)	2001-12-07	2005-12-27	Pharmacia Corporation	Substituted pyrazoles as p38 kinase inhibitors
AU7966198A (en)	1997-06-13	1998-12-30	Smithkline Beecham Corporation	Novel pyrazole and pyrazoline substituted compounds
WO1998057966A1 (en)	1997-06-19	1998-12-23	Smithkline Beecham Corporation	Novel aryloxy substituted pyrimidine imidazole compounds
US6489325B1 (en)	1998-07-01	2002-12-03	Smithkline Beecham Corporation	Substituted imidazole compounds
US7301021B2 (en)	1997-07-02	2007-11-27	Smithkline Beecham Corporation	Substituted imidazole compounds
US6562832B1 (en)	1997-07-02	2003-05-13	Smithkline Beecham Corporation	Substituted imidazole compounds
CA2306077A1 (en)	1997-10-08	1999-04-15	Smithkline Beecham Corporation	Novel cycloalkenyl substituted compounds
AU1924699A (en)	1997-12-19	1999-07-12	Smithkline Beecham Corporation	Compounds of heteroaryl substituted imidazole, their pharmaceutical compositionsand uses
US6858617B2 (en)	1998-05-26	2005-02-22	Smithkline Beecham Corporation	Substituted imidazole compounds
DE69917296T2 (de) *	1998-08-20	2005-05-25	Smithkline Beecham Corp.	Neue substituierte triazolverbindungen
AU1909200A (en)	1998-11-04	2000-05-22	Smithkline Beecham Corporation	Pyridin-4-yl or pyrimidin-4-yl substituted pyrazines
US6239279B1 (en) *	1998-12-16	2001-05-29	Smithkline Beecham Corporation	Synthesis for 4-aryl-5-pyrimidine imidazole substituted derivatives
US6857013B2 (en) *	1999-01-29	2005-02-15	Intermec Ip.Corp.	Remote anomaly diagnosis and reconfiguration of an automatic data collection device platform over a telecommunications network
US20050274801A1 (en) *	1999-01-29	2005-12-15	Intermec Ip Corp.	Method, apparatus and article for validating ADC devices, such as barcode, RFID and magnetic stripe readers
US7122666B2 (en)	1999-07-21	2006-10-17	Sankyo Company, Limited	Heteroaryl-substituted pyrrole derivatives, their preparation and their therapeutic uses
US6976062B1 (en) *	1999-09-22	2005-12-13	Intermec Ip Corp.	Automated software upgrade utility
EP1233950B1 (en)	1999-11-23	2005-10-05	Smithkline Beecham Corporation	3,4-DIHYDRO-(1H)QUINAZOLIN-2-ONE COMPOUNDS AS CSBP/P39 kINASE INHIBITORS
JP2003514900A (ja)	1999-11-23	2003-04-22	スミスクライン・ビーチャム・コーポレイション	ＣＳＢＰ／ｐ３８キナーゼ阻害剤としての３，４−ジヒドロ−（１Ｈ）−キナゾリン−２−オン化合物
WO2001038312A1 (en)	1999-11-23	2001-05-31	Smithkline Beecham Corporation	3,4-DIHYDRO-(1H)QUINAZOLIN-2-ONE COMPOUNDS AS CSBP/p38 KINASE INHIBITORS
US6759410B1 (en) *	1999-11-23	2004-07-06	Smithline Beecham Corporation	3,4-dihydro-(1H)-quinazolin-2-ones and their use as CSBP/p38 kinase inhibitors
US7235551B2 (en) *	2000-03-02	2007-06-26	Smithkline Beecham Corporation	1,5-disubstituted-3,4-dihydro-1h-pyrimido[4,5-d]pyrimidin-2-one compounds and their use in treating csbp/p38 kinase mediated diseases
ES2372028T3 (es) *	2000-10-23	2012-01-13	Glaxosmithkline Llc	Nuevo compuesto de 8h-pirido[2,3-d]pirimidin-7-ona trisustituida para el tratamiento de enfermedades mediadas por la csbp/p38 quinasa.
EP1361225B1 (en)	2001-01-22	2007-11-07	Sankyo Company, Limited	Compounds substituted with bicyclic amino groups
WO2002094267A1 (fr) *	2001-05-24	2002-11-28	Sankyo Company, Limited	Preparation pharmaceutique pour prevenir ou traiter l'arthrite
AR039241A1 (es) *	2002-04-04	2005-02-16	Biogen Inc	Heteroarilos trisustituidos y metodos para su produccion y uso de los mismos
UA80295C2 (en)	2002-09-06	2007-09-10	Biogen Inc	Pyrazolopyridines and using the same
CL2004000234A1 (es) *	2003-02-12	2005-04-15	Biogen Idec Inc	Compuestos derivados 3-(piridin-2-il)-4-heteroaril-pirazol sustituidos, antagonistas de aik5 y/o aik4; composicion farmaceutica y uso del compuesto en el tratamiento de desordenes fibroticos como esclerodermia, lupus nefritico, cicatrizacion de herid
CA2603163A1 (en) *	2005-03-25	2006-10-05	Glaxo Group Limited	Process for preparing pyrido[2,3-d]pyrimidin-7-one and 3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one derivatives
PE20061351A1 (es) *	2005-03-25	2007-01-14	Glaxo Group Ltd	COMPUESTOS 8H-PIRIDO[2,3-d]PIRIMIDIN-7-ONA 2,4,8-TRISUSTITUIDOS COMO INHIBIDORES DE LA QUINASA CSBP/RK/p38
US8944332B2 (en)	2006-08-04	2015-02-03	Intermec Ip Corp.	Testing automatic data collection devices, such as barcode, RFID and/or magnetic stripe readers
WO2019168874A1 (en)	2018-02-27	2019-09-06	The Research Foundation For The State University Of New York	Difluoromethoxylation and trifluoromethoxylation compositions and methods for synthesizing same

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US3557114A (en) *	1968-12-23	1971-01-19	Merck & Co Inc	1-substituted-3-(2-pyrimidinyl) imidazolium salts
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US5593991A (en) *	1993-07-16	1997-01-14	Adams; Jerry L.	Imidazole compounds, use and process of making
IL110296A (en) *	1993-07-16	1999-12-31	Smithkline Beecham Corp	Imidazole compounds process for their preparation and pharmaceutical compositions containing them
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US5670527A (en) *	1993-07-16	1997-09-23	Smithkline Beecham Corporation	Pyridyl imidazole compounds and compositions
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ATE325113T1 (de) *	1993-10-01	2006-06-15	Novartis Pharma Gmbh	Pharmacologisch wirksame pyrimidinderivate und verfahren zu deren herstellung
DE4337611A1 (de) *	1993-11-04	1995-05-11	Boehringer Ingelheim Kg	Neue Benzoylguanidine, ihre Herstellung und ihre Verwendung in Arzneimitteln
PL321292A1 (en) *	1995-01-12	1997-11-24	Smithkline Beecham Corp	Novel xchemical compounds
US5739143A (en) *	1995-06-07	1998-04-14	Smithkline Beecham Corporation	Imidazole compounds and compositions
IL118544A (en) *	1995-06-07	2001-08-08	Smithkline Beecham Corp	History of imidazole, the process for their preparation and the pharmaceutical preparations containing them
ZA9610687B (en) *	1995-12-22	1997-09-29	Smithkline Beecham Corp	Novel synthesis.
AP9700912A0 (en) *	1996-01-11	1997-01-31	Smithkline Beecham Corp	Novel cycloalkyl substituted imidazoles
HUP9902460A3 (en) *	1996-01-11	2000-03-28	Smithkline Beecham Corp	Novel substituted imidazole compounds, their use, method for their preparation and pharmaceutical compositions containing them
ZA97175B (en) *	1996-01-11	1997-11-04	Smithkline Beecham Corp	Novel substituted imidazole compounds.
WO1997025047A1 (en) *	1996-01-11	1997-07-17	Smithkline Beecham Corporation	Novel cycloalkyl substituded imidazoles
US6096739A (en) *	1996-03-25	2000-08-01	Smithkline Beecham Corporation	Treatment for CNS injuries
EP0889887A4 (en) *	1996-03-25	2003-06-11	Smithkline Beecham Corp	TREATMENT OF CENTRAL NERVOUS SYSTEM INJURIES

1996
- 1996-12-19 ZA ZA9610687A patent/ZA9610687B/xx unknown
- 1996-12-20 WO PCT/US1996/020599 patent/WO1997023479A1/en not_active Application Discontinuation
- 1996-12-20 IL IL12490896A patent/IL124908A/xx not_active IP Right Cessation
- 1996-12-20 TR TR1998/01121T patent/TR199801121T2/xx unknown
- 1996-12-20 BR BR9612187A patent/BR9612187A/pt not_active Application Discontinuation
- 1996-12-20 IL IL14351796A patent/IL143517A/xx not_active IP Right Cessation
- 1996-12-20 KR KR1019980704729A patent/KR19990076625A/ko not_active Application Discontinuation
- 1996-12-20 AU AU14681/97A patent/AU704500B2/en not_active Ceased
- 1996-12-20 US US08/771,320 patent/US5917043A/en not_active Expired - Fee Related
- 1996-12-20 CN CN96180018A patent/CN1209128A/zh active Pending
- 1996-12-20 EP EP96945272A patent/EP1019393A1/en not_active Withdrawn
- 1996-12-20 JP JP52385597A patent/JP3245175B2/ja not_active Expired - Fee Related
- 1996-12-20 PL PL96327311A patent/PL327311A1/xx unknown
- 1996-12-20 AR ARP960105842A patent/AR004405A1/es unknown
- 1996-12-20 HU HU9902466A patent/HUP9902466A3/hu unknown
- 1996-12-20 US US09/091,799 patent/US6100399A/en not_active Expired - Fee Related
- 1996-12-20 NZ NZ326574A patent/NZ326574A/xx unknown
- 1996-12-20 CZ CZ981985A patent/CZ198598A3/cs unknown
1997
- 1997-08-22 TW TW086112050A patent/TW434236B/zh not_active IP Right Cessation
1998
- 1998-03-30 AR ARP980101441A patent/AR012567A1/es not_active Application Discontinuation
- 1998-03-30 AR ARP980101440A patent/AR015579A1/es not_active Application Discontinuation
- 1998-06-19 NO NO982850A patent/NO982850L/no not_active Application Discontinuation
1999
- 1999-01-20 US US09/233,511 patent/US6255491B1/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
AU1468197A (en)	1997-07-17
AR004405A1 (es)	1998-11-04
US5917043A (en)	1999-06-29
IL143517A0 (en)	2002-04-21
NZ326574A (en)	2000-01-28
BR9612187A (pt)	1999-07-13
CZ198598A3 (cs)	1998-10-14
AR012567A1 (es)	2000-11-08
JP2000502683A (ja)	2000-03-07
AU704500B2 (en)	1999-04-22
EP1019393A4 (en)	2000-07-19
WO1997023479A1 (en)	1997-07-03
NO982850D0 (no)	1998-06-19
HUP9902466A3 (en)	2002-11-28
TR199801121T2 (xx)	1998-08-21
AR015579A1 (es)	2001-05-16
CN1209128A (zh)	1999-02-24
PL327311A1 (en)	1998-12-07
KR19990076625A (ko)	1999-10-15
IL124908A0 (en)	1999-01-26
JP3245175B2 (ja)	2002-01-07
US6255491B1 (en)	2001-07-03
ZA9610687B (en)	1997-09-29
HUP9902466A2 (hu)	2000-05-28
NO982850L (no)	1998-06-19
IL143517A (en)	2003-09-17
US6100399A (en)	2000-08-08
TW434236B (en)	2001-05-16
EP1019393A1 (en)	2000-07-19

Legal Events

Date	Code	Title
2003-11-23	FF	Patent granted
2003-12-10	KB	Patent renewed
2004-12-15	NP	Permission for amending the patent specification granted (section 66, patents law 1967)
2007-02-12	KB	Patent renewed
2011-07-31	MM9K	Patent not in force due to non-payment of renewal fees

Publication	Publication Date	Title
IL124908A (en)	2003-05-29	Processes for the preparation of 5-pyrimidinyl substituted imidazoles and aminoalkyl carbonyl imidazole intermediates thereor
AU5750796A (en)	1996-12-11	System for the treatment of insomnia
GB9400965D0 (en)	1994-03-16	Audio conferencing system
TW300689U (en)	1997-03-11	Speaker system for television set
AU4237896A (en)	1996-06-06	Method and intermediates for the synthesis of korupensamines
GB2302231B (en)	1999-01-13	Speaker system
AU4247593A (en)	1993-12-13	Imidazoles for the treatment of atherosclerosis
GB2294214B (en)	1998-07-15	Metallic coating
AU3734193A (en)	1993-09-13	Ultrasonic spray coating system and method
GB9515336D0 (en)	1995-09-20	Multi-media services system
GB2305263B (en)	1998-03-11	System for simplifying the implementation of specified functions
GB2313847B (en)	1998-12-09	Member having composite coating and process for producing the same
GB9624854D0 (en)	1997-01-15	Structural part of hf-tight housings
SG44742A1 (en)	1997-12-19	Intermediates and process for the preparation of an antiviral agent
AU2352295A (en)	1995-11-16	Imidazole derivative and process for producing the same
AU6425696A (en)	1997-03-06	Method of operating an inductor and inductor for carrying out the method
HUP9600320A3 (en)	1999-03-29	Process and new intermediates for the preparation of triazolinon-derivatives
GB2302384B (en)	1999-08-11	Impregnation of liners
GB2270595B (en)	1995-12-06	An audio system
ZA966438B (en)	1997-02-19	Method of operationg an inductor and inductor for carrying out the method.
GB2294216B (en)	1998-07-15	Method of metallic painting
GB9416237D0 (en)	1994-10-05	Sound distribution system
AU3374595A (en)	1996-05-02	Vehicle powder coating system
AU2028797A (en)	1997-10-22	Use of substituted aryl imidazoles
GB9622465D0 (en)	1997-01-08	Method of transforming pyrazole compounds and compounds prepared using the method