HUP9904107A3 - 3-substituted pyrido[4',3':4,5]thieno[2,3-d]pyrimidine derivatives,their preparation and their use - Google Patents

3-substituted pyrido[4',3':4,5]thieno[2,3-d]pyrimidine derivatives,their preparation and their use

Info

Publication number: HUP9904107A3
Authority: HU; Hungary
Prior art keywords: thieno; preparation; pyrimidine derivatives; substituted pyrido; pyrido
Prior art date: 1996-09-10

Application number

HU9904107A

Other languages

English (en)

Original Assignee

Basf Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1996-09-10

Filing date

1997-08-22

Publication date

2001-10-29

1997-08-22 Application filed by Basf Ag filed Critical Basf Ag

2000-05-28 Publication of HUP9904107A2 publication Critical patent/HUP9904107A2/hu

2001-10-29 Publication of HUP9904107A3 publication Critical patent/HUP9904107A3/hu

Links

-1 3-substituted pyrido[4',3':4,5]thieno[2,3-d]pyrimidine Chemical class 0.000 title 1
229940083082 pyrimidine derivative acting on arteriolar smooth muscle Drugs 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D495/14—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pain & Pain Management (AREA)
Psychiatry (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

HU9904107A 1996-09-10 1997-08-22 3-substituted pyrido[4',3':4,5]thieno[2,3-d]pyrimidine derivatives,their preparation and their use HUP9904107A3 (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE19636769A DE19636769A1 (de)	1996-09-10	1996-09-10	3-Substituierte Pyrido [4',3':4,5]thieno[2,3-d]pyrimidin-Derivate, ihre Herstellung und Verwendung

Publications (2)

Publication Number	Publication Date
HUP9904107A2 HUP9904107A2 (hu)	2000-05-28
HUP9904107A3 true HUP9904107A3 (en)	2001-10-29

Family

ID=7805168

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
HU9904107A HUP9904107A3 (en)	1996-09-10	1997-08-22	3-substituted pyrido[4',3':4,5]thieno[2,3-d]pyrimidine derivatives,their preparation and their use

Country Status (32)

Country	Link
US (1)	US6222034B1 (hu)
EP (1)	EP0927184B1 (hu)
JP (1)	JP2001500138A (hu)
KR (1)	KR20000035987A (hu)
CN (2)	CN1230962A (hu)
AR (1)	AR009572A1 (hu)
AT (1)	ATE252587T1 (hu)
AU (1)	AU736678B2 (hu)
BG (1)	BG63602B1 (hu)
BR (1)	BR9711724A (hu)
CA (1)	CA2265509A1 (hu)
CO (1)	CO4900071A1 (hu)
CZ (1)	CZ288896B6 (hu)
DE (2)	DE19636769A1 (hu)
DK (1)	DK0927184T3 (hu)
ES (1)	ES2210570T3 (hu)
HK (1)	HK1043593A1 (hu)
HR (1)	HRP970484A2 (hu)
HU (1)	HUP9904107A3 (hu)
ID (1)	ID18260A (hu)
IL (1)	IL128142A0 (hu)
NO (1)	NO991132L (hu)
NZ (1)	NZ334350A (hu)
PL (1)	PL332144A1 (hu)
PT (1)	PT927184E (hu)
RU (1)	RU2198888C2 (hu)
SK (1)	SK283039B6 (hu)
TR (1)	TR199900503T2 (hu)
TW (1)	TW480264B (hu)
UA (1)	UA54449C2 (hu)
WO (1)	WO1998011110A1 (hu)
ZA (1)	ZA978081B (hu)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE19724980A1 (de) *	1997-06-13	1998-12-17	Basf Ag	3-Substituierte 3,4-Dihydro-thieno[2,3-d]pyrimidin-Derivate, ihre Herstellung und Verwendung
DE19724979A1 (de) *	1997-06-13	1998-12-17	Basf Ag	3-substituierte Pyrido [3,4,5]thieno[2,3-d]pyrimidin-Derivate, ihre Herstellung und Verwendung
DE19734444A1 (de)	1997-08-08	1999-02-11	Basf Ag	3-Substituierte 3,4,5,7-Tetrahydro-pyrrolo(3',4':4,5) thieno (2,3-d) pyrimidin-Derivate, ihre Herstellung und Verwendung
DE19900545A1 (de) *	1999-01-11	2000-07-13	Basf Ag	Verwendung von Pyrimidinderivaten zur Prophylaxe und Therapie der zerebralen Ischämie
DE19900673A1 (de) *	1999-01-11	2000-07-13	Basf Ag	Verwendung von Bindungspartnern für 5-HT5-Rezeptoren zur Behandlung neurodegenerativer und neuropsychiatrischer Störungen
FR2791980B1 (fr) *	1999-04-09	2001-07-06	Sod Conseils Rech Applic	Pyrido-thieno-diazepines, leur procede de preparation, et les compositions pharmaceutiques les contenant
DE10031390A1 (de) *	2000-07-03	2002-01-17	Knoll Ag	Pyrimidinderivate und ihre Verwendung zur Prophylaxe und Therapie der zerebralen Ischämie
DE10031389A1 (de) *	2000-07-03	2002-01-17	Knoll Ag	Pyrimidinderivate und ihre Verwendung zur Prophylaxe und Therapie der zerebralen Ischämie
AU2001269540A1 (en)	2000-07-18	2002-01-30	Sumitomo Pharmaceuticals Co. Ltd.	Serotonin reuptake inhibitors
DE10259382A1 (de) *	2002-12-18	2004-07-01	Abbott Gmbh & Co. Kg	3-Substituierte 3,4-Dihydro-thieno[2,3-d]pyrimidin-4-on-Derivate, ihre Herstellung und Verwendung
US20050222175A1 (en) *	2004-03-31	2005-10-06	Dhanoa Dale S	New piperidinylamino-thieno[2,3-D] pyrimidine compounds
BRPI0408988A (pt) *	2003-03-31	2006-03-28	Predix Pharmaceuticals Holding	composto de piperidinilamino-tieno[2,3-d]pirimidina
US7612078B2 (en) *	2003-03-31	2009-11-03	Epix Delaware, Inc.	Piperidinylamino-thieno[2,3-D] pyrimidine compounds
US20050165025A1 (en) *	2004-01-22	2005-07-28	Recordati Ireland Ltd.	Combination therapy with 5HT 1A and 5HT 1B-receptor antagonists
US7488736B2 (en) *	2004-05-17	2009-02-10	Epix Delaware, Inc.	Thienopyridinone compounds and methods of treatment
US7407966B2 (en) *	2004-10-07	2008-08-05	Epix Delaware, Inc.	Thienopyridinone compounds and methods of treatment
US7598265B2 (en) *	2004-09-30	2009-10-06	Epix Delaware, Inc.	Compositions and methods for treating CNS disorders
US7576211B2 (en) *	2004-09-30	2009-08-18	Epix Delaware, Inc.	Synthesis of thienopyridinone compounds and related intermediates
US8114894B2 (en) *	2008-12-03	2012-02-14	Nanotherapeutics, Inc.	Bicyclic compounds and methods of making and using same
DK2558473T3 (da) *	2010-04-14	2016-12-19	Bayer Ip Gmbh	Fremgangsmåde til fremstilling af dithiin-tetracarboximider

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE272079C (hu) *
DE272088C (hu) *
DE272086C (hu) *
DE1937459A1 (de) *	1968-08-02	1970-02-05	Ciba Geigy	Neue Pyrimidinderivate und Verfahren zu ihrer Herstellung
US3823151A (en) *	1968-08-02	1974-07-09	Ciba Geigy Corp	4,5,6,7-tetrahydrothieno(2,3-d)pyridines
JPS60146891A (ja) *	1984-01-05	1985-08-02	Mitsubishi Chem Ind Ltd	〔２，３−ｄ〕チエノピリミジン誘導体およびその塩
EP0799617A3 (en) *	1986-02-24	1997-11-12	Mitsui Petrochemical Industries, Ltd.	Therapeutic agent for neurological diseases
US5001130A (en)	1988-02-18	1991-03-19	Bristol-Myers Company	Psychotropic heterobicycloalkylpiperazine derivatives
US4835157A (en) *	1988-03-15	1989-05-30	Ortho Pharmaceutical Corporation	Thieno- and furopyrimidine-2,4-dione piperidine derivatives as serotonin antagonists and alpha adrenergic blocking agents

1996
- 1996-09-10 DE DE19636769A patent/DE19636769A1/de not_active Withdrawn
1997
- 1997-08-22 CZ CZ1999759A patent/CZ288896B6/cs not_active IP Right Cessation
- 1997-08-22 HU HU9904107A patent/HUP9904107A3/hu unknown
- 1997-08-22 EP EP97940118A patent/EP0927184B1/de not_active Expired - Lifetime
- 1997-08-22 NZ NZ334350A patent/NZ334350A/xx unknown
- 1997-08-22 AT AT97940118T patent/ATE252587T1/de not_active IP Right Cessation
- 1997-08-22 CN CN97197765A patent/CN1230962A/zh active Pending
- 1997-08-22 DK DK97940118T patent/DK0927184T3/da active
- 1997-08-22 SK SK230-99A patent/SK283039B6/sk unknown
- 1997-08-22 PL PL97332144A patent/PL332144A1/xx unknown
- 1997-08-22 AU AU42071/97A patent/AU736678B2/en not_active Ceased
- 1997-08-22 UA UA99042039A patent/UA54449C2/uk unknown
- 1997-08-22 US US09/254,449 patent/US6222034B1/en not_active Expired - Lifetime
- 1997-08-22 TR TR1999/00503T patent/TR199900503T2/xx unknown
- 1997-08-22 JP JP10513191A patent/JP2001500138A/ja active Pending
- 1997-08-22 KR KR1019997001939A patent/KR20000035987A/ko not_active Application Discontinuation
- 1997-08-22 BR BR9711724A patent/BR9711724A/pt not_active Application Discontinuation
- 1997-08-22 RU RU99106781/04A patent/RU2198888C2/ru not_active IP Right Cessation
- 1997-08-22 WO PCT/EP1997/004593 patent/WO1998011110A1/de not_active Application Discontinuation
- 1997-08-22 IL IL12814297A patent/IL128142A0/xx unknown
- 1997-08-22 CA CA002265509A patent/CA2265509A1/en not_active Abandoned
- 1997-08-22 ES ES97940118T patent/ES2210570T3/es not_active Expired - Lifetime
- 1997-08-22 PT PT97940118T patent/PT927184E/pt unknown
- 1997-08-22 DE DE59710902T patent/DE59710902D1/de not_active Expired - Fee Related
- 1997-09-02 TW TW086112642A patent/TW480264B/zh not_active IP Right Cessation
- 1997-09-09 ZA ZA978081A patent/ZA978081B/xx unknown
- 1997-09-09 CO CO97052337A patent/CO4900071A1/es unknown
- 1997-09-09 AR ARP970104118A patent/AR009572A1/es unknown
- 1997-09-10 HR HR19636769.7A patent/HRP970484A2/xx not_active Application Discontinuation
- 1997-09-10 ID IDP973146A patent/ID18260A/id unknown
1999
- 1999-01-27 BG BG103122A patent/BG63602B1/bg unknown
- 1999-03-09 NO NO991132A patent/NO991132L/no not_active Application Discontinuation
2001
- 2001-05-18 CN CN01116979A patent/CN1332168A/zh active Pending
2002
- 2002-07-17 HK HK02105304.8A patent/HK1043593A1/zh unknown

Also Published As

Publication number	Publication date
DE19636769A1 (de)	1998-03-12
SK283039B6 (sk)	2003-02-04
SK23099A3 (en)	1999-08-06
KR20000035987A (ko)	2000-06-26
CA2265509A1 (en)	1998-03-19
UA54449C2 (uk)	2003-03-17
PL332144A1 (en)	1999-08-30
DE59710902D1 (de)	2003-11-27
ES2210570T3 (es)	2004-07-01
RU2198888C2 (ru)	2003-02-20
BG63602B1 (bg)	2002-06-28
CN1332168A (zh)	2002-01-23
EP0927184A1 (de)	1999-07-07
NZ334350A (en)	2000-07-28
CZ288896B6 (cs)	2001-09-12
ID18260A (id)	1998-03-19
NO991132D0 (no)	1999-03-09
ATE252587T1 (de)	2003-11-15
WO1998011110A1 (de)	1998-03-19
US6222034B1 (en)	2001-04-24
HK1043593A1 (zh)	2002-09-20
TW480264B (en)	2002-03-21
IL128142A0 (en)	1999-11-30
BR9711724A (pt)	1999-08-24
PT927184E (pt)	2004-03-31
CN1230962A (zh)	1999-10-06
AU736678B2 (en)	2001-08-02
NO991132L (no)	1999-03-09
AU4207197A (en)	1998-04-02
CO4900071A1 (es)	2000-03-27
BG103122A (en)	1999-09-30
EP0927184B1 (de)	2003-10-22
ZA978081B (en)	1999-03-09
AR009572A1 (es)	2000-04-26
DK0927184T3 (da)	2004-03-01
JP2001500138A (ja)	2001-01-09
HRP970484A2 (en)	1998-10-31
HUP9904107A2 (hu)	2000-05-28
CZ75999A3 (cs)	1999-06-16
TR199900503T2 (xx)	1999-07-21

Publication	Publication Date	Title
HUP9904107A3 (en)	2001-10-29	3-substituted pyrido[4',3':4,5]thieno[2,3-d]pyrimidine derivatives,their preparation and their use
IL134081A0 (en)	2001-04-30	1,2,4-triazolo [4,3-b]pyrido[3,2-d]pyridazine derivatives and pharmaceutical compositions containing them
HK1045510A1 (en)	2002-11-29	Imidazo[1,2-a]pyridine and pyrazolo[2,3-a]pyridine derivatives
HUP0002902A3 (en)	2002-09-30	3-substituted 3,4 dyhydro-thieno[2,3-d]pyrimidine derivatives and their use for the preparation of pharmaceutical compositions
HUP9900607A3 (en)	1999-11-29	Pyrido[2,3-d]pyrimidine derivatives and medicinal compositions thereof
IL128225A0 (en)	1999-11-30	Pyridazino [4,5-b]-quinoline 5-oxide derivatives their preparation and their use as glycine antagonists
HK1023338A1 (en)	2000-09-08	1h-pyrido [3,4-b] indole-4-carboxamide derivatives, preparation and application thereof in therapeutics
ZA987114B (en)	2000-02-07	3-substituted 3,4,5,7-tetrahydropyrrolol[3',4':4,5] thieno[2,3-D]pyrimidine derivatives, their preparation and use.
ZA985120B (en)	1999-12-13	3-Substituted pyrido[3',4':4,5]thieno[2,3-d]pyrimidine derivatives, their preparation and use.
HUP0003394A3 (en)	2003-04-28	Pyrido[2,3-b][1,5]benzodiazepine derivatives, their use, process for their preparation and pharmaceutical compositions containing them
GB2316072B (en)	2000-05-10	Pyrrolo[3,2-c]quinoline derivatives
ZA9811642B (en)	1999-06-24	Pyrido 1,2,4-thiadiazine derivatives their preparation and use
EP0904271A4 (en)	2002-01-23	5,6,7,8-tetrahydropyrido [2,3-d] PYRIMIDINE
HUP9902614A3 (en)	2001-12-28	Novel n-7-heterocyclyl pyrrolo[2,3-d]pyridines and their use