HUP0401776A2 - Intraorálisan széteső valdekoxib készítmények porlasztásos szárítási eljárással előállítva - Google Patents

Intraorálisan széteső valdekoxib készítmények porlasztásos szárítási eljárással előállítva

Info

Publication number
HUP0401776A2
HUP0401776A2 HU0401776A HUP0401776A HUP0401776A2 HU P0401776 A2 HUP0401776 A2 HU P0401776A2 HU 0401776 A HU0401776 A HU 0401776A HU P0401776 A HUP0401776 A HU P0401776A HU P0401776 A2 HUP0401776 A2 HU P0401776A2
Authority
HU
Hungary
Prior art keywords
valdecoxid
drying process
spray drying
compositions prepared
intraorally disintegrating
Prior art date
Application number
HU0401776A
Other languages
English (en)
Inventor
Joseph P. Reo
Uday J. Shah
Ken Yamamoto
Original Assignee
Pharmacia Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia Corporation filed Critical Pharmacia Corporation
Publication of HUP0401776A2 publication Critical patent/HUP0401776A2/hu

Links

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
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    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
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    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Virology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Diabetes (AREA)
  • Pulmonology (AREA)
  • Dermatology (AREA)
  • Communicable Diseases (AREA)
  • Immunology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Rheumatology (AREA)
  • Endocrinology (AREA)
  • Oncology (AREA)
  • Molecular Biology (AREA)
  • Neurosurgery (AREA)
  • Epidemiology (AREA)
  • Reproductive Health (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hematology (AREA)
  • Pain & Pain Management (AREA)
  • Gynecology & Obstetrics (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pregnancy & Childbirth (AREA)
  • Cardiology (AREA)
  • Urology & Nephrology (AREA)
  • Zoology (AREA)

Abstract

A találmány orálisan széteső, gyorsan szétmálló valdekoxib tablettákraés ilyen dózisformák előállítására alkalmas eljárásra vonatkozik. Akészítmények ciklooxigenáz-2 által közvetített betegségállapotok ésrendellenességek kezelésére vagy megelőzésére használhatók. Ó
HU0401776A 2001-10-10 2002-10-10 Intraorálisan széteső valdekoxib készítmények porlasztásos szárítási eljárással előállítva HUP0401776A2 (hu)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US32808801P 2001-10-10 2001-10-10
PCT/US2002/032333 WO2003030876A1 (en) 2001-10-10 2002-10-10 Intraorally disintegrating valdecoxib compositions prepared by spray drying process

Publications (1)

Publication Number Publication Date
HUP0401776A2 true HUP0401776A2 (hu) 2004-12-28

Family

ID=23279455

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0401776A HUP0401776A2 (hu) 2001-10-10 2002-10-10 Intraorálisan széteső valdekoxib készítmények porlasztásos szárítási eljárással előállítva

Country Status (28)

Country Link
EP (1) EP1450769A1 (hu)
JP (1) JP2005508348A (hu)
KR (1) KR20050035138A (hu)
CN (1) CN1602187A (hu)
AP (1) AP2004003022A0 (hu)
BG (1) BG108675A (hu)
BR (1) BR0213152A (hu)
CA (1) CA2462881A1 (hu)
CO (1) CO5570687A2 (hu)
CZ (1) CZ2004456A3 (hu)
EA (1) EA200400423A1 (hu)
EC (1) ECSP045056A (hu)
GE (1) GEP20063857B (hu)
HR (1) HRP20040331A2 (hu)
HU (1) HUP0401776A2 (hu)
IL (1) IL161253A0 (hu)
IS (1) IS7211A (hu)
MA (1) MA27543A1 (hu)
MX (1) MXPA04003404A (hu)
NO (1) NO20041894L (hu)
NZ (1) NZ532184A (hu)
OA (1) OA12666A (hu)
PL (1) PL370136A1 (hu)
SK (1) SK1662004A3 (hu)
TN (1) TNSN04056A1 (hu)
WO (1) WO2003030876A1 (hu)
YU (1) YU37104A (hu)
ZA (1) ZA200402728B (hu)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7815937B2 (en) 1998-10-27 2010-10-19 Biovail Laboratories International Srl Quick dissolve compositions and tablets based thereon
WO2012087113A1 (en) * 2010-12-24 2012-06-28 N.V. Nutricia Improved nutritional tablet

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5576014A (en) * 1994-01-31 1996-11-19 Yamanouchi Pharmaceutical Co., Ltd Intrabuccally dissolving compressed moldings and production process thereof
CN1140267C (zh) * 1996-05-17 2004-03-03 麦克公司 治疗环加氧酶-2介导的疾病的每天一次的组合物
JP2003516353A (ja) * 1999-12-08 2003-05-13 ファルマシア コーポレイション ヴァルデコキシブ組成物
US6316029B1 (en) * 2000-05-18 2001-11-13 Flak Pharma International, Ltd. Rapidly disintegrating solid oral dosage form
DK1309315T3 (da) * 2000-08-18 2006-10-09 Pharmacia Corp Hurtigt disintegrerende oral valdecoxib-formulering
CN1638739A (zh) * 2000-08-18 2005-07-13 法玛西雅厄普约翰美国公司 治疗成瘾性障碍的化合物

Also Published As

Publication number Publication date
NZ532184A (en) 2005-12-23
EP1450769A1 (en) 2004-09-01
AP2004003022A0 (en) 2004-06-30
ZA200402728B (en) 2005-03-17
TNSN04056A1 (fr) 2006-06-01
MXPA04003404A (es) 2004-06-18
BG108675A (en) 2005-03-31
YU37104A (sh) 2006-08-17
MA27543A1 (fr) 2005-10-03
PL370136A1 (en) 2005-05-16
CO5570687A2 (es) 2005-10-31
SK1662004A3 (sk) 2005-07-01
OA12666A (en) 2006-06-19
IL161253A0 (en) 2004-09-27
BR0213152A (pt) 2004-10-19
CN1602187A (zh) 2005-03-30
EA200400423A1 (ru) 2004-10-28
JP2005508348A (ja) 2005-03-31
CA2462881A1 (en) 2003-04-17
KR20050035138A (ko) 2005-04-15
CZ2004456A3 (cs) 2005-03-16
WO2003030876A1 (en) 2003-04-17
GEP20063857B (en) 2006-06-26
IS7211A (is) 2004-04-07
HRP20040331A2 (en) 2005-12-31
ECSP045056A (es) 2004-08-27
NO20041894D0 (no) 2004-05-07
NO20041894L (no) 2004-07-07

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