HK1251221A1 - 用於治療和預防乙型肝炎病毒感染的新的三環4-吡啶酮-3-甲酸衍生物 - Google Patents

用於治療和預防乙型肝炎病毒感染的新的三環4-吡啶酮-3-甲酸衍生物

Info

Publication number
HK1251221A1
HK1251221A1 HK18110504.8A HK18110504A HK1251221A1 HK 1251221 A1 HK1251221 A1 HK 1251221A1 HK 18110504 A HK18110504 A HK 18110504A HK 1251221 A1 HK1251221 A1 HK 1251221A1
Authority
HK
Hong Kong
Prior art keywords
pyridone
prophylaxis
hepatitis
treatment
carboxylic acid
Prior art date
Application number
HK18110504.8A
Other languages
English (en)
Inventor
Zhanling Cheng
Xingchun Han
Chungen Liang
Song Yang
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of HK1251221A1 publication Critical patent/HK1251221A1/zh

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/20—Antivirals for DNA viruses

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  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biotechnology (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
HK18110504.8A 2015-07-21 2018-08-15 用於治療和預防乙型肝炎病毒感染的新的三環4-吡啶酮-3-甲酸衍生物 HK1251221A1 (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CN2015084601 2015-07-21
PCT/EP2016/067002 WO2017013046A1 (en) 2015-07-21 2016-07-18 Novel tricyclic 4-pyridone-3-carboxylic acid derivatives for the treatment and prophylaxis of hepatitis b virus infection

Publications (1)

Publication Number Publication Date
HK1251221A1 true HK1251221A1 (zh) 2019-01-25

Family

ID=56418520

Family Applications (1)

Application Number Title Priority Date Filing Date
HK18110504.8A HK1251221A1 (zh) 2015-07-21 2018-08-15 用於治療和預防乙型肝炎病毒感染的新的三環4-吡啶酮-3-甲酸衍生物

Country Status (6)

Country Link
US (1) US10336751B2 (zh)
EP (1) EP3325477B1 (zh)
JP (1) JP6598974B2 (zh)
CN (1) CN107849037B (zh)
HK (1) HK1251221A1 (zh)
WO (1) WO2017013046A1 (zh)

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Also Published As

Publication number Publication date
EP3325477B1 (en) 2019-05-01
US20180134705A1 (en) 2018-05-17
JP6598974B2 (ja) 2019-10-30
EP3325477A1 (en) 2018-05-30
US10336751B2 (en) 2019-07-02
WO2017013046A1 (en) 2017-01-26
JP2018524374A (ja) 2018-08-30
CN107849037B (zh) 2020-04-17
CN107849037A (zh) 2018-03-27

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