FR2981933B1 - Derives d'oxoazetidine, leur procede de preparation et leur utilisation en medecine humaine ainsi qu'en cosmetique - Google Patents

Derives d'oxoazetidine, leur procede de preparation et leur utilisation en medecine humaine ainsi qu'en cosmetique

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Publication number
FR2981933B1
FR2981933B1 FR1159911A FR1159911A FR2981933B1 FR 2981933 B1 FR2981933 B1 FR 2981933B1 FR 1159911 A FR1159911 A FR 1159911A FR 1159911 A FR1159911 A FR 1159911A FR 2981933 B1 FR2981933 B1 FR 2981933B1
Authority
FR
France
Prior art keywords
compounds
cosmetics
preparation
human medicine
general formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR1159911A
Other languages
English (en)
Other versions
FR2981933A1 (fr
Inventor
Claire Bouix-Peter
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Galderma Research and Development SNC
Original Assignee
Galderma Research and Development SNC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to FR1159911A priority Critical patent/FR2981933B1/fr
Application filed by Galderma Research and Development SNC filed Critical Galderma Research and Development SNC
Priority to BR112013033861-0A priority patent/BR112013033861B1/pt
Priority to RU2014102966A priority patent/RU2624011C2/ru
Priority to ES12730549.8T priority patent/ES2620476T3/es
Priority to PCT/EP2012/062622 priority patent/WO2013001030A1/fr
Priority to JP2014517715A priority patent/JP5898310B2/ja
Priority to KR1020147002462A priority patent/KR101946085B1/ko
Priority to AU2012277838A priority patent/AU2012277838B2/en
Priority to CA2840606A priority patent/CA2840606A1/fr
Priority to US14/130,282 priority patent/US9353083B2/en
Priority to MX2014000170A priority patent/MX2014000170A/es
Priority to EP12730549.8A priority patent/EP2726478B1/fr
Priority to CN201280032433.4A priority patent/CN103827106B/zh
Priority to ARP120102343A priority patent/AR086803A1/es
Publication of FR2981933A1 publication Critical patent/FR2981933A1/fr
Application granted granted Critical
Publication of FR2981933B1 publication Critical patent/FR2981933B1/fr
Priority to IN711CHN2014 priority patent/IN2014CN00711A/en
Priority to US15/139,018 priority patent/US9981952B2/en
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
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    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
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    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
    • A61K8/494—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with more than one nitrogen as the only hetero atom
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  • Psychiatry (AREA)
  • Gynecology & Obstetrics (AREA)
  • Endocrinology (AREA)
FR1159911A 2011-06-30 2011-11-02 Derives d'oxoazetidine, leur procede de preparation et leur utilisation en medecine humaine ainsi qu'en cosmetique Expired - Fee Related FR2981933B1 (fr)

Priority Applications (16)

Application Number Priority Date Filing Date Title
FR1159911A FR2981933B1 (fr) 2011-11-02 2011-11-02 Derives d'oxoazetidine, leur procede de preparation et leur utilisation en medecine humaine ainsi qu'en cosmetique
MX2014000170A MX2014000170A (es) 2011-06-30 2012-06-28 Derivados de oxazetidina, proceso para su preparacion y uso de los mismos en medicina humana y en cosmetica.
ES12730549.8T ES2620476T3 (es) 2011-06-30 2012-06-28 Derivados de oxazetidina, procedimiento para su preparación y su utilización en medicina humana y en cosméticos
PCT/EP2012/062622 WO2013001030A1 (fr) 2011-06-30 2012-06-28 Dérivés d'oxazétidine, leur procédé de préparation et leur utilisation en médecine humaine et en cosmétique
JP2014517715A JP5898310B2 (ja) 2011-06-30 2012-06-28 オキサゼチジン誘導体、それらの調製方法並びにヒト医療及び化粧品におけるそれらの使用
KR1020147002462A KR101946085B1 (ko) 2011-06-30 2012-06-28 옥사제티딘 유도체, 그의 제조 방법 및 인간 의약 및 화장품에서의 그의 용도
AU2012277838A AU2012277838B2 (en) 2011-06-30 2012-06-28 Oxazetidine derivatives, process for preparing them and use thereof in human medicine and in cosmetics
CA2840606A CA2840606A1 (fr) 2011-06-30 2012-06-28 Derives d'oxazetidine, leur procede de preparation et leur utilisation en medecine humaine et en cosmetique
BR112013033861-0A BR112013033861B1 (pt) 2011-06-30 2012-06-28 Compostos agonistas do receptor de mc1r, usos de ditos compostos, composição farmacêutica, composição cosmética e usos cosméticos de compostos agonistas do receptor de mc1r
RU2014102966A RU2624011C2 (ru) 2011-06-30 2012-06-28 Производные оксазетидина, способ для их получения и их применение в медицине и косметике
EP12730549.8A EP2726478B1 (fr) 2011-06-30 2012-06-28 Dérivés d'oxazétidine, leur procédé de préparation et leur utilisation en médecine humaine et en cosmétique
CN201280032433.4A CN103827106B (zh) 2011-06-30 2012-06-28 氧氮杂环丁烷衍生物、其制备方法及其在人用药物和化妆品中的用途
US14/130,282 US9353083B2 (en) 2011-06-30 2012-06-28 Oxazetidine derivatives, process for preparing them and use in human medicine and in cosmetics
ARP120102343A AR086803A1 (es) 2011-06-30 2012-06-29 Derivados de oxazetidinas, composiciones farmaceuticas y cosmeticas que los contienen y uso de los mismos para tratar enfermedades dermatologicas fundamentalmente, y del aparato respiratorio, digestivo y cardiovascular, entre otras
IN711CHN2014 IN2014CN00711A (fr) 2011-06-30 2014-01-28
US15/139,018 US9981952B2 (en) 2011-06-30 2016-04-26 Oxazetidine derivatives, process for preparing them and use in human medicine and in cosmetics

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WO2013135880A1 (fr) * 2012-03-15 2013-09-19 Galderma Research & Development Combinaison d'un agoniste du récepteur mc1r et d'uvb dans le traitement et/ou la prévention de troubles de la pigmentation
CA2968836A1 (fr) 2016-06-13 2017-12-13 Gilead Sciences, Inc. Composes modulant fxr (nr1h4)
AU2018215619A1 (en) * 2017-02-01 2019-08-08 Clinuvel Pharmaceuticals Ltd Alpha-MSH analogues used in the treatment of xeroderma pigmentosum
CN110461328A (zh) 2017-03-28 2019-11-15 吉利德科学公司 治疗肝疾病的治疗组合
US11524005B2 (en) 2019-02-19 2022-12-13 Gilead Sciences, Inc. Solid forms of FXR agonists
BR112022025115A2 (pt) * 2020-06-10 2023-02-07 Mitsubishi Tanabe Pharma Corp Agente profilático ou terapêutico para fotodermatose

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MY128261A (en) * 1992-10-27 2007-01-31 Merck Sharp & Dohme New substituted azetidinones as anti-inflammatory and antidegenerative agents
JP2004532838A (ja) * 2001-03-02 2004-10-28 ブリストル−マイヤーズ スクイブ カンパニー メラノコルチン受容体のモデュレーターとして有用な化合物及びそれを含む製薬組成物
KR100661118B1 (ko) * 2003-11-12 2006-12-26 주식회사 엘지생명과학 멜라노코틴 수용체의 항진제
FR2937973B1 (fr) * 2008-11-04 2010-11-05 Galderma Res & Dev Modulateurs des recepteurs de la melanocortine, leur procede de preparation et leur utilisation en medecine humaine ainsi qu'en cosmetique
FR2937972B1 (fr) * 2008-11-04 2013-03-29 Galderma Res & Dev Derives d'oxoazetidine, leur procede de preparation et leur utilisation en medecine humaine ainsi qu'en cosmetique

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KR101946085B1 (ko) 2019-02-08
JP2014518238A (ja) 2014-07-28
CA2840606A1 (fr) 2013-01-03
BR112013033861A2 (pt) 2017-12-19
MX2014000170A (es) 2014-02-19
ES2620476T3 (es) 2017-06-28
KR20140050019A (ko) 2014-04-28
AU2012277838A1 (en) 2014-01-23
US9981952B2 (en) 2018-05-29
AU2012277838B2 (en) 2017-04-13
AR086803A1 (es) 2014-01-22
IN2014CN00711A (fr) 2015-04-03
US20160237065A1 (en) 2016-08-18
EP2726478B1 (fr) 2017-01-11
US20140228342A1 (en) 2014-08-14
RU2014102966A (ru) 2015-08-10
FR2981933A1 (fr) 2013-05-03
RU2624011C2 (ru) 2017-06-30
US9353083B2 (en) 2016-05-31
CN103827106A (zh) 2014-05-28
WO2013001030A1 (fr) 2013-01-03
EP2726478A1 (fr) 2014-05-07
JP5898310B2 (ja) 2016-04-06
BR112013033861B1 (pt) 2021-11-09

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