FR2792318B1 - INDAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION - Google Patents
INDAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATIONInfo
- Publication number
- FR2792318B1 FR2792318B1 FR9905013A FR9905013A FR2792318B1 FR 2792318 B1 FR2792318 B1 FR 2792318B1 FR 9905013 A FR9905013 A FR 9905013A FR 9905013 A FR9905013 A FR 9905013A FR 2792318 B1 FR2792318 B1 FR 2792318B1
- Authority
- FR
- France
- Prior art keywords
- preparation
- therapeutic application
- indazole derivatives
- indazole
- derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
- C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
- C07D451/06—Oxygen atoms
- C07D451/12—Oxygen atoms acylated by aromatic or heteroaromatic carboxylic acids, e.g. ***e
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
Priority Applications (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9905013A FR2792318B1 (en) | 1999-04-16 | 1999-04-16 | INDAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
AU39715/00A AU3971500A (en) | 1999-04-16 | 2000-04-11 | Indazole derivatives, preparation and therapeutic application thereof |
PCT/FR2000/000923 WO2000063215A2 (en) | 1999-04-16 | 2000-04-11 | Indazole derivatives, preparation and therapeutic application thereof |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9905013A FR2792318B1 (en) | 1999-04-16 | 1999-04-16 | INDAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2792318A1 FR2792318A1 (en) | 2000-10-20 |
FR2792318B1 true FR2792318B1 (en) | 2001-06-15 |
Family
ID=9544676
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR9905013A Expired - Fee Related FR2792318B1 (en) | 1999-04-16 | 1999-04-16 | INDAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
Country Status (3)
Country | Link |
---|---|
AU (1) | AU3971500A (en) |
FR (1) | FR2792318B1 (en) |
WO (1) | WO2000063215A2 (en) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TW200533348A (en) | 2004-02-18 | 2005-10-16 | Theravance Inc | Indazole-carboxamide compounds as 5-ht4 receptor agonists |
US7728006B2 (en) | 2004-04-07 | 2010-06-01 | Theravance, Inc. | Quinolinone-carboxamide compounds as 5-HT4 receptor agonists |
US8309575B2 (en) | 2004-04-07 | 2012-11-13 | Theravance, Inc. | Quinolinone-carboxamide compounds as 5-HT4 receptor agonists |
TWI351282B (en) | 2004-04-07 | 2011-11-01 | Theravance Inc | Quinolinone-carboxamide compounds as 5-ht4 recepto |
DE602005016446D1 (en) | 2004-11-05 | 2009-10-15 | Theravance Inc | 5-HT4 receptor agonist compounds |
ATE431824T1 (en) | 2004-11-05 | 2009-06-15 | Theravance Inc | QUINOLINONE-CARBOXAMIDE COMPOUNDS |
ES2347265T3 (en) | 2004-12-22 | 2010-10-27 | Theravance, Inc. | INDAZOL-CARBOXAMIDA COMPOUNDS. |
KR20070107807A (en) | 2005-03-02 | 2007-11-07 | 세라밴스 인코포레이티드 | Quinolinone compounds as 5-ht4 receptor agonists |
WO2007120599A2 (en) * | 2006-04-12 | 2007-10-25 | Wyeth | Dihydro[1,4]oxazino[2,3,4-hi]indazole derivatives as 5-hydroxytryptamine-6 ligands |
GB201511382D0 (en) | 2015-06-29 | 2015-08-12 | Imp Innovations Ltd | Novel compounds and their use in therapy |
EP3663723A1 (en) | 2018-12-04 | 2020-06-10 | Renishaw PLC | Encoder apparatus |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4950759A (en) * | 1988-07-07 | 1990-08-21 | Duphar International Research B.V. | Substituted 1,7-annelated 1H-indazoles |
GB8916682D0 (en) * | 1989-07-21 | 1989-09-06 | Beecham Group Plc | Pharmaceutical compounds |
CA2160420A1 (en) * | 1994-10-20 | 1996-04-21 | Haruhiko Kikuchi | 5-ht4 receptor agonists |
FR2769915B1 (en) * | 1997-10-21 | 2000-10-13 | Synthelabo | TRICYCLIC INDAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
-
1999
- 1999-04-16 FR FR9905013A patent/FR2792318B1/en not_active Expired - Fee Related
-
2000
- 2000-04-11 AU AU39715/00A patent/AU3971500A/en not_active Abandoned
- 2000-04-11 WO PCT/FR2000/000923 patent/WO2000063215A2/en active Application Filing
Also Published As
Publication number | Publication date |
---|---|
AU3971500A (en) | 2000-11-02 |
WO2000063215A2 (en) | 2000-10-26 |
FR2792318A1 (en) | 2000-10-20 |
WO2000063215A3 (en) | 2001-02-01 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
TP | Transmission of property | ||
ST | Notification of lapse |