FR2574793B1 - INDOLE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESS FOR THEIR PREPARATION - Google Patents

INDOLE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESS FOR THEIR PREPARATION

Info

Publication number
FR2574793B1
FR2574793B1 FR8518416A FR8518416A FR2574793B1 FR 2574793 B1 FR2574793 B1 FR 2574793B1 FR 8518416 A FR8518416 A FR 8518416A FR 8518416 A FR8518416 A FR 8518416A FR 2574793 B1 FR2574793 B1 FR 2574793B1
Authority
FR
France
Prior art keywords
preparation
pharmaceutical compositions
compositions containing
indole derivatives
indole
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
FR8518416A
Other languages
French (fr)
Other versions
FR2574793A1 (en
Inventor
David Edmund Bays
Colin Frederick Webb
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Glaxo Group Ltd
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of FR2574793A1 publication Critical patent/FR2574793A1/en
Application granted granted Critical
Publication of FR2574793B1 publication Critical patent/FR2574793B1/en
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • C07D209/16Tryptamines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
FR8518416A 1984-12-13 1985-12-12 INDOLE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESS FOR THEIR PREPARATION Expired FR2574793B1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB848431426A GB8431426D0 (en) 1984-12-13 1984-12-13 Chemical compounds

Publications (2)

Publication Number Publication Date
FR2574793A1 FR2574793A1 (en) 1986-06-20
FR2574793B1 true FR2574793B1 (en) 1988-10-14

Family

ID=10571103

Family Applications (1)

Application Number Title Priority Date Filing Date
FR8518416A Expired FR2574793B1 (en) 1984-12-13 1985-12-12 INDOLE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESS FOR THEIR PREPARATION

Country Status (11)

Country Link
JP (1) JPS61151172A (en)
AU (1) AU579687B2 (en)
BE (1) BE903846A (en)
CH (1) CH667454A5 (en)
DE (1) DE3543982A1 (en)
FR (1) FR2574793B1 (en)
GB (2) GB8431426D0 (en)
IT (1) IT1182089B (en)
NL (1) NL8503424A (en)
SE (1) SE8505887L (en)
ZA (1) ZA859520B (en)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8530507D0 (en) * 1985-12-11 1986-01-22 Glaxo Group Plc Chemical compounds
GB8607824D0 (en) * 1986-03-27 1986-04-30 Glaxo Group Ltd Chemical compounds
GB8614287D0 (en) * 1986-06-12 1986-07-16 Glaxo Group Ltd Chemical compounds
US4894386A (en) * 1987-04-15 1990-01-16 Ici Americas Inc. Aliphatic carboxamides
GB8719167D0 (en) * 1987-08-13 1987-09-23 Glaxo Group Ltd Chemical compounds
US5225431A (en) * 1987-10-23 1993-07-06 Burroughs Wellcome Co. Therapeutic substituted indole compounds and compositions thereof
SK281621B6 (en) * 1990-06-07 2001-05-10 Astrazeneca Ab Therapeutic heterocyclic compounds
GB9209882D0 (en) * 1992-05-07 1992-06-24 Glaxo Lab Sa Compositions
GB9211277D0 (en) 1992-05-28 1992-07-15 Glaxo Group Inc Pharmaceutical compositions
GB9216009D0 (en) * 1992-07-28 1992-09-09 Almirall Lab New indol derivatives
ES2056025B1 (en) * 1992-10-08 1995-05-01 Almirall Lab NEW DERIVATIVES OF INDOL.
FR2707639B1 (en) * 1993-06-30 1995-10-13 Pf Medicament New indole compounds derived from arylamines as selective ligands for the 5HT1D and 5HT1B receptors.
CA2508290C (en) 2002-12-20 2017-02-28 Ciba Specialty Chemicals Holding Inc. Synthesis of amines and intermediates for the synthesis thereof
WO2005118551A2 (en) 2004-05-28 2005-12-15 Ligand Pharmaceuticals Inc. Thrombopoietin activity modulating compounds and methods
WO2006047344A1 (en) * 2004-10-25 2006-05-04 Ligand Pharmaceuticals, Inc. Thrombopoietin activity modulating compounds and methods
EP2141148B1 (en) 2007-03-29 2013-07-03 Daiichi Sankyo Company, Limited Indole derivative having cpla2 inhibitory activity, use of the same and method for producing the same

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA795239B (en) * 1978-10-12 1980-11-26 Glaxo Group Ltd Heterocyclic compounds
GB2082175B (en) * 1980-08-12 1984-05-02 Glaxo Group Ltd Heterocyclic compounds
SE8505715L (en) * 1984-12-04 1986-06-05 Glaxo Group Ltd indole derivatives
GB8530507D0 (en) * 1985-12-11 1986-01-22 Glaxo Group Plc Chemical compounds

Also Published As

Publication number Publication date
GB8431426D0 (en) 1985-01-23
BE903846A (en) 1986-06-12
JPS61151172A (en) 1986-07-09
SE8505887D0 (en) 1985-12-12
IT8548921A0 (en) 1985-12-12
SE8505887L (en) 1986-06-14
FR2574793A1 (en) 1986-06-20
CH667454A5 (en) 1988-10-14
AU5115185A (en) 1986-06-19
ZA859520B (en) 1986-08-27
GB2168347A (en) 1986-06-18
DE3543982A1 (en) 1986-06-19
AU579687B2 (en) 1988-12-01
IT1182089B (en) 1987-09-30
NL8503424A (en) 1986-07-01
GB2168347B (en) 1988-02-03
GB8530591D0 (en) 1986-01-22

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Legal Events

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