FR2383941A1 - Nouveaux derives pyrimidinyliques et leur procede de preparation - Google Patents
Nouveaux derives pyrimidinyliques et leur procede de preparationInfo
- Publication number
- FR2383941A1 FR2383941A1 FR7820654A FR7820654A FR2383941A1 FR 2383941 A1 FR2383941 A1 FR 2383941A1 FR 7820654 A FR7820654 A FR 7820654A FR 7820654 A FR7820654 A FR 7820654A FR 2383941 A1 FR2383941 A1 FR 2383941A1
- Authority
- FR
- France
- Prior art keywords
- preparation process
- pyrimidinyl derivatives
- new
- new pyrimidinyl
- derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
La présente invention concerne de nouveaux dérivés pyrimidinyliques et leur procédé de préparation. Les composés de l'invention répondent à la formule générale :
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
AT73877A AT351036B (de) | 1977-02-04 | 1977-02-04 | Verfahren zur herstellung von neuen oxadiazolopyrimidinderivaten und von deren salzen |
LU7778639A LU78639A1 (fr) | 1977-02-04 | 1977-12-05 |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2383941A1 true FR2383941A1 (fr) | 1978-10-13 |
FR2383941B1 FR2383941B1 (fr) | 1980-07-25 |
Family
ID=25593772
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR7802908A Granted FR2379538A1 (fr) | 1977-02-04 | 1978-02-02 | Nouveaux derives d'oxadiazolopyrimidine, leur preparation et leur application en tant que medicaments |
FR7820654A Granted FR2383941A1 (fr) | 1977-02-04 | 1978-07-11 | Nouveaux derives pyrimidinyliques et leur procede de preparation |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR7802908A Granted FR2379538A1 (fr) | 1977-02-04 | 1978-02-02 | Nouveaux derives d'oxadiazolopyrimidine, leur preparation et leur application en tant que medicaments |
Country Status (22)
Country | Link |
---|---|
US (1) | US4150132A (fr) |
JP (1) | JPS6024794B2 (fr) |
AR (1) | AR223642A1 (fr) |
CA (1) | CA1092108A (fr) |
CH (1) | CH638215A5 (fr) |
DE (1) | DE2804518C2 (fr) |
DK (1) | DK50878A (fr) |
ES (2) | ES466589A1 (fr) |
FI (1) | FI62309C (fr) |
FR (2) | FR2379538A1 (fr) |
GB (2) | GB1563888A (fr) |
GR (1) | GR72280B (fr) |
IE (1) | IE46318B1 (fr) |
IL (2) | IL53925A (fr) |
IT (1) | IT1092334B (fr) |
MC (1) | MC1183A1 (fr) |
NL (1) | NL179585C (fr) |
NO (2) | NO780396L (fr) |
NZ (1) | NZ186334A (fr) |
PH (3) | PH14637A (fr) |
PT (1) | PT67614B (fr) |
SE (1) | SE7801311L (fr) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA1103245A (fr) * | 1978-07-21 | 1981-06-16 | Jean-Claude Muller | Procede de production de nouveaux derives de l'oxadiazolopyrimidine |
NZ190915A (en) * | 1978-07-31 | 1984-07-31 | Hoffmann La Roche | Oxadiazolotriazine derivatives and pharmaceutical compositions |
US4307093A (en) * | 1980-06-23 | 1981-12-22 | The Upjohn Company | Animal feed and process |
DK148826C (da) * | 1980-12-19 | 1986-03-24 | Hoffmann La Roche | Analogifremgangsmaade til fremstilling af oxadiazolopyrimidinderivater eller salte deraf med baser og pyrimidinderivat til anvendelse som mellemprodukt ved denne fremgangsmaade |
CA1179344A (fr) * | 1981-07-15 | 1984-12-11 | Jean-Claude Muller | Procede de preparation de 6-¬3,6-dihydro-1(2h)- pyridyl|pyrimidine-3-oxydes |
CH649291A5 (de) * | 1982-03-16 | 1985-05-15 | Hoffmann La Roche | Dicarbamate. |
WO1986000616A1 (fr) * | 1984-07-13 | 1986-01-30 | Gail Sansone Bazzano | Oxydes de pyrimidine substitues utiles pour favoriser la croissance des cheveux |
JPH04249875A (ja) * | 1991-01-08 | 1992-09-04 | Yazaki Corp | 電線を端子化するための成形用電極及び端子化電線 |
Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3382248A (en) * | 1965-11-01 | 1968-05-07 | Upjohn Co | 6-amino-4, 5-di(substituted amino)-1, 2-dihydro-1-hydroxy-2-iminopyrimidines |
FR2132726A1 (fr) * | 1971-04-07 | 1972-11-24 | Upjohn Co |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2118261A1 (de) * | 1971-04-15 | 1972-11-02 | C.H. Boehringer Sohn, 6507 Ingelheim | Neue N-haltige Bicyclen, deren Säureadditionssalze sowie Verfahren zu deren Herstellung |
BE786028A (fr) * | 1971-07-08 | 1973-01-08 | Boehringer Sohn Ingelheim | 2,3-dihydro-oxo-imidazo(1,2-a)-pyrimidines, leurs sels d'addition avec des acides et procedes pour les fabriquer |
BE790008A (fr) * | 1971-10-15 | 1973-04-12 | Fmc Corp | Nouveaux composes herbicides |
DE2210633C2 (de) * | 1972-03-06 | 1983-09-22 | Bayer Ag, 5090 Leverkusen | Kondensierte Pyridinderivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel |
DE2252122A1 (de) * | 1972-10-24 | 1974-04-25 | Hoechst Ag | Oxazolo-chinazoline und verfahren zu ihrer herstellung |
DE2253555A1 (de) * | 1972-11-02 | 1974-05-09 | Hoechst Ag | Oxazolo-pyrimidine und verfahren zu ihrer herstellung |
US3901928A (en) * | 1973-01-10 | 1975-08-26 | Robert Henry Hesse | 1' ,3' -dihydroxy steroid-5-enes method of preparing same and their use for preparing 1' -hydroxy-25-hydrogen vitamin d compounds |
-
1978
- 1978-01-10 CH CH22778A patent/CH638215A5/de not_active IP Right Cessation
- 1978-01-23 CA CA295,438A patent/CA1092108A/fr not_active Expired
- 1978-01-27 NZ NZ186334A patent/NZ186334A/xx unknown
- 1978-01-27 US US05/873,182 patent/US4150132A/en not_active Expired - Lifetime
- 1978-01-30 IT IT19786/78A patent/IT1092334B/it active
- 1978-01-30 IL IL53925A patent/IL53925A/xx unknown
- 1978-01-30 IE IE197/78A patent/IE46318B1/en unknown
- 1978-02-02 JP JP53009964A patent/JPS6024794B2/ja not_active Expired
- 1978-02-02 MC MC781280A patent/MC1183A1/fr unknown
- 1978-02-02 GR GR55335A patent/GR72280B/el unknown
- 1978-02-02 DE DE2804518A patent/DE2804518C2/de not_active Expired
- 1978-02-02 FR FR7802908A patent/FR2379538A1/fr active Granted
- 1978-02-02 FI FI780343A patent/FI62309C/fi not_active IP Right Cessation
- 1978-02-03 DK DK50878A patent/DK50878A/da not_active Application Discontinuation
- 1978-02-03 NL NLAANVRAGE7801288,A patent/NL179585C/xx not_active IP Right Cessation
- 1978-02-03 AR AR270966A patent/AR223642A1/es active
- 1978-02-03 GB GB2536/79A patent/GB1563888A/en not_active Expired
- 1978-02-03 GB GB4450/78A patent/GB1563887A/en not_active Expired
- 1978-02-03 ES ES466589A patent/ES466589A1/es not_active Expired
- 1978-02-03 SE SE7801311A patent/SE7801311L/xx unknown
- 1978-02-03 PT PT67614A patent/PT67614B/pt unknown
- 1978-02-03 NO NO780396A patent/NO780396L/no unknown
- 1978-02-06 PH PH20749A patent/PH14637A/en unknown
- 1978-02-06 PH PH20750A patent/PH13962A/en unknown
- 1978-07-11 FR FR7820654A patent/FR2383941A1/fr active Granted
- 1978-08-28 ES ES472875A patent/ES472875A1/es not_active Expired
- 1978-11-19 PH PH21786A patent/PH15009A/en unknown
-
1980
- 1980-03-14 IL IL59627A patent/IL59627A0/xx unknown
- 1980-10-23 NO NO803160A patent/NO803160L/no unknown
Patent Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3382248A (en) * | 1965-11-01 | 1968-05-07 | Upjohn Co | 6-amino-4, 5-di(substituted amino)-1, 2-dihydro-1-hydroxy-2-iminopyrimidines |
FR2132726A1 (fr) * | 1971-04-07 | 1972-11-24 | Upjohn Co |
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
FR2430412A1 (fr) | Derives substitues de propanolamine utiles comme medicaments et procede de leur preparation | |
FR2430419A1 (fr) | Nouveaux derives de l'indole, leur preparation et leur application comme medicaments | |
FR2357541A1 (fr) | Composes polyeniques et leur procede de preparation | |
FR2383171A1 (fr) | Derives de thiopropanoylaminoacides utiles comme hypotenseurs | |
FR2405937A1 (fr) | Nouveaux derives de dihydropyridine, leur procede de preparation et leur application | |
FR2403989A1 (fr) | Nouveaux derives a-halogenomethyles d'amines utiles comme medicaments et procedes de leur preparation | |
FR2374307A1 (fr) | Derives de la 1,4-dihydropyridine, leur procede d'obtention et composition pharmaceutique les contenant | |
FR2416892A1 (fr) | Derives de pyrido(1,2-a)pyrimidines, procede pour leur preparation et compositions pharmaceutiques qui les contiennent | |
FR2383165A1 (fr) | Nouveaux derives d'acides phenoxy-a-phenoxy-alcanecarboxyliques, leur preparation et leur application comme herbicides | |
FR2398065A1 (fr) | ||
FR2383183A1 (fr) | Derives de benzodiazepine | |
FR2363559A1 (fr) | Nouveaux derives de perhydro-aza-heterocycles utiles comme medicaments et procede pour leur preparation | |
FR2403330A1 (fr) | Nouveaux derives de benzoyl-2-chloro-4-glycinanilides substitues, leur procede de preparation et leur application en tant que medicaments | |
FR2386544A1 (fr) | Procede pour la preparation de derives d'imidazodiazepine | |
FR2363563A1 (fr) | Nouveaux derives de 1-acyloxymethyl-5-fluorouracile utiles notamment comme agents antitumoraux, et leur procede de preparation | |
FR2398058A1 (fr) | Nouveaux derives de l'indole, leur preparation et leur application comme medicaments | |
FR2418240A1 (fr) | Procede de preparation de composes de glucopyranose-nitrosouree et nouveaux composes ainsi obtenus | |
FR2383941A1 (fr) | Nouveaux derives pyrimidinyliques et leur procede de preparation | |
FR2377367A1 (fr) | Procede de preparation d'alcoxy-cetones | |
FR2383931A1 (fr) | Derives d'oxadiazolopyrimidine | |
FR2355020A1 (fr) | Antibiotiques de b-lactames et leur procede de preparation | |
FR2374291A1 (fr) | ||
FR2394514A1 (fr) | Nouvel acide cyclohexanecarboxylique et ses derives | |
FR2361352A1 (fr) | Derives acylamino (alkyl)-benzeniques, leur procede de preparation et leur application | |
FR2388789A1 (fr) | Derives d'acide benzoique, leur procede de preparation et leur application therapeutique |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
TP | Transmission of property | ||
ST | Notification of lapse |