FR2362141A1 - N- (6- (R3R4N) -4 (OR 5) -R5-3-PYRIDAZINYL) THERAPEUTIC ALKYLIDENYL AMINOMETHYLENEMALONATES - Google Patents

N- (6- (R3R4N) -4 (OR 5) -R5-3-PYRIDAZINYL) THERAPEUTIC ALKYLIDENYL AMINOMETHYLENEMALONATES

Info

Publication number
FR2362141A1
FR2362141A1 FR7725414A FR7725414A FR2362141A1 FR 2362141 A1 FR2362141 A1 FR 2362141A1 FR 7725414 A FR7725414 A FR 7725414A FR 7725414 A FR7725414 A FR 7725414A FR 2362141 A1 FR2362141 A1 FR 2362141A1
Authority
FR
France
Prior art keywords
aminomethylenemalonates
alkylidenyl
r3r4n
pyridazinyl
therapeutic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7725414A
Other languages
French (fr)
Other versions
FR2362141B1 (en
Inventor
Y Lesher
Chester J Opalka Jr
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
STWB Inc
Original Assignee
Sterling Drug Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/805,419 external-priority patent/US4104385A/en
Application filed by Sterling Drug Inc filed Critical Sterling Drug Inc
Publication of FR2362141A1 publication Critical patent/FR2362141A1/en
Application granted granted Critical
Publication of FR2362141B1 publication Critical patent/FR2362141B1/fr
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D237/00Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/02Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
    • C07D237/06Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D237/10Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D237/20Nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Abstract

Nouveaux composés à activité chimiothérapeutique. N-16-(R3 R4 N)-4 (ou 5)-R5 -3-pyfidazinylõ aminométhylènemalonates d'alkylidényle cyclique de formule :New compounds with chemotherapeutic activity. Cyclic alkylidenyl N-16- (R3 R4 N) -4 (or 5) -R5 -3-pyfidazinylõ aminomethylenemalonates of the formula:

FR7725414A 1976-08-19 1977-08-19 N- (6- (R3R4N) -4 (OR 5) -R5-3-PYRIDAZINYL) THERAPEUTIC ALKYLIDENYL AMINOMETHYLENEMALONATES Granted FR2362141A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US71569976A 1976-08-19 1976-08-19
US05/805,419 US4104385A (en) 1976-08-19 1977-06-10 Cyclic alkylidenyl N-[6-(amino)-3-pyridazinyl]aminomethylenemalonates

Publications (2)

Publication Number Publication Date
FR2362141A1 true FR2362141A1 (en) 1978-03-17
FR2362141B1 FR2362141B1 (en) 1981-07-17

Family

ID=27109402

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7725414A Granted FR2362141A1 (en) 1976-08-19 1977-08-19 N- (6- (R3R4N) -4 (OR 5) -R5-3-PYRIDAZINYL) THERAPEUTIC ALKYLIDENYL AMINOMETHYLENEMALONATES

Country Status (14)

Country Link
JP (1) JPS5334782A (en)
AR (1) AR221687A1 (en)
AU (1) AU515629B2 (en)
DE (1) DE2737542A1 (en)
DK (1) DK368177A (en)
EG (1) EG12733A (en)
FR (1) FR2362141A1 (en)
GB (1) GB1542030A (en)
IL (1) IL52681A (en)
LU (1) LU77976A1 (en)
NL (1) NL7709162A (en)
NZ (1) NZ184875A (en)
PH (1) PH12796A (en)
PT (1) PT66928B (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH03133573A (en) * 1989-07-26 1991-06-06 Sanso Aaku Kogyo Kk Melt-cutting electrode
HU226859B1 (en) * 1997-10-27 2009-12-28 Neurosearch As Phenyl- or heteroaryl-homopiperazines, their use and medicaments containing them

Also Published As

Publication number Publication date
NL7709162A (en) 1978-02-21
FR2362141B1 (en) 1981-07-17
GB1542030A (en) 1979-03-14
DE2737542A1 (en) 1978-02-23
PT66928A (en) 1977-09-01
NZ184875A (en) 1979-03-28
IL52681A0 (en) 1977-10-31
DK368177A (en) 1978-02-20
JPS5334782A (en) 1978-03-31
PH12796A (en) 1979-08-17
AR221687A1 (en) 1981-03-13
AU515629B2 (en) 1981-04-16
LU77976A1 (en) 1978-04-27
AU2770477A (en) 1979-02-15
IL52681A (en) 1981-06-29
PT66928B (en) 1979-02-05
EG12733A (en) 1979-09-30

Similar Documents

Publication Publication Date Title
FR2369266A1 (en) N-BENZO NEWS
FR2364210A1 (en) HETEROCYCLIC PHENYL ETHERS AND HERBICIDAL PRODUCTS CONTAINING THEM
FR2416891A1 (en) 6-N-PROPYL-8-METHOXYMETHYL OR METHYLMERCAPTOMETHYLERGOLINES AND RELATED COMPOUNDS, AND THEIR THERAPEUTIC USE
FR2386588A1 (en) PIGMENTS DERIVED FROM ISO-INDOLINE, THEIR PREPARATION AND THEIR APPLICATIONS
FR2400517A1 (en) TRIAZOLO-2,4-BENZODIAZEPINES AND THEIR THERAPEUTIC USE
FR2359810A1 (en) ALKYLENE OR CYCLOALKYLENE-AMMONIUM BIS-TETRAHALOGENOPHTHALATES, THEIR PREPARATION AND THEIR APPLICATION TO THE PREPARATION OF CORRESPONDING IMIDES
FR2356651A1 (en) NEW PENICILLANIC ACID DERIVATIVES AND THEIR THERAPEUTIC USE
FR2446283A1 (en) PHENOXYPHENYLPIPERIDINES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATIONS
FR2391199A1 (en) ALKYLENE DIAMINE DERIVATIVES AND MEDICINAL PRODUCTS CONTAINING THEM
FR2375234A1 (en) 1,2-DIHYDRO-3H-PYRROLO (1,2-A) PYRROLE-1-CARBOXYLATES AND THEIR OBTAINING
FR2362122A1 (en) NEWS 3- (2-ARYL-2-PROPYL) UREES, AND THEIR USE AS HERBICIDES
FR2357558A1 (en) 2,6-METHANO-2H-1-BENZOXOCINS
FR2391182A1 (en) DICARBONYL CHELATES AND MOISTURE-CURING EPOXIDE COMPOSITIONS
FR2362141A1 (en) N- (6- (R3R4N) -4 (OR 5) -R5-3-PYRIDAZINYL) THERAPEUTIC ALKYLIDENYL AMINOMETHYLENEMALONATES
FR2368474A1 (en)
FR2363541A1 (en) ACYLOXY-N, N 'DIACYLMALONAMIDES AND THEIR METHOD OF PREPARATION
FR2453167A1 (en) FURANS CARRYING AN ARYL SUBSTITUTE, THEIR PREPARATION AND THE MEDICINAL PRODUCTS CONTAINING SAME
FR2381030A1 (en) 2-PHENYLAMINOMETHYL IMIDAZOLINES AND THEIR PREPARATION
BE857979A (en) N- (6- (R3R4N) -4 (OR 5) - R5 - 3 - PYRIDAZINYL) THERAPEUTIC ALKYLIDENYL AMINOMETHYLENEMALONATES
FR2444044A1 (en) NOVEL DERIVATIVES OF N-PHENYL PHOSPHATES, N- (ALCOXY CARBONYLALCOYL) -ACETAMIDES AND FUNGICIDAL COMPOSITIONS CONTAINING THEM
FR2357613A2 (en) CATIONIC DYES, THEIR OBTAINING AND THEIR APPLICATION
FR2377406A1 (en) TETRATHIAPENTALENE AND TETRASELENAPENTALENE COMPOUNDS
FR2373524A1 (en) N1-CHLORO-3,5-DINITROSULFANILAMIDES HERBICIDES AND FUNGICIDES
FR2361364A1 (en) NEW DERIVATIVES OF AZETIDINE
FR2366292A1 (en) NEW TETRACYCLIC COMPOUNDS DERIVED FROM DIAZEPINE-1,4 WITH BIOLOGICAL ACTIVITY

Legal Events

Date Code Title Description
ST Notification of lapse