FR2351112A1 - Derive de prostaglandine et medicament contenant ce derive - Google Patents

Derive de prostaglandine et medicament contenant ce derive

Info

Publication number
FR2351112A1
FR2351112A1 FR7714201A FR7714201A FR2351112A1 FR 2351112 A1 FR2351112 A1 FR 2351112A1 FR 7714201 A FR7714201 A FR 7714201A FR 7714201 A FR7714201 A FR 7714201A FR 2351112 A1 FR2351112 A1 FR 2351112A1
Authority
FR
France
Prior art keywords
cpds
healing
alpha
derivs
prostaglandin
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7714201A
Other languages
English (en)
Other versions
FR2351112B1 (fr
Inventor
Salvador Moncada
Norman Whittake
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Wellcome Foundation Ltd
Original Assignee
Wellcome Foundation Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/624,486 external-priority patent/US3984400A/en
Priority claimed from FR7631769A external-priority patent/FR2361871A1/fr
Priority claimed from FR7710593A external-priority patent/FR2351111A1/fr
Application filed by Wellcome Foundation Ltd filed Critical Wellcome Foundation Ltd
Publication of FR2351112A1 publication Critical patent/FR2351112A1/fr
Application granted granted Critical
Publication of FR2351112B1 publication Critical patent/FR2351112B1/fr
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/93Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems condensed with a ring other than six-membered
    • C07D307/935Not further condensed cyclopenta [b] furans or hydrogenated cyclopenta [b] furans
    • C07D307/937Not further condensed cyclopenta [b] furans or hydrogenated cyclopenta [b] furans with hydrocarbon or substituted hydrocarbon radicals directly attached in position 2, e.g. prostacyclins

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FR7714201A 1975-10-21 1977-05-10 Derive de prostaglandine et medicament contenant ce derive Granted FR2351112A1 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US05/624,486 US3984400A (en) 1975-10-21 1975-10-21 11-Desoxy-16-aryl-ω-tetranorprostaglandins
FR7631769A FR2361871A1 (fr) 1975-10-21 1976-10-21 11-desoxy-16-arylprostaglandines 13-acetyleniques
FR7710593A FR2351111A1 (fr) 1976-05-11 1977-04-07 Methylacetals de 2-(2b-ethynyl-cyclopent-1a-yl) acetaldehydes et leur preparation

Publications (2)

Publication Number Publication Date
FR2351112A1 true FR2351112A1 (fr) 1977-12-09
FR2351112B1 FR2351112B1 (fr) 1981-05-29

Family

ID=27250686

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7714201A Granted FR2351112A1 (fr) 1975-10-21 1977-05-10 Derive de prostaglandine et medicament contenant ce derive

Country Status (1)

Country Link
FR (1) FR2351112A1 (fr)

Cited By (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2359125A1 (fr) * 1976-02-04 1978-02-17 Upjohn Co Nouveaux derives de prostaglandine, leur procede de preparation et medicament les contenant
FR2378777A1 (fr) * 1977-01-31 1978-08-25 Ono Pharmaceutical Co Nouveaux analogues de prostaglandines
FR2401141A1 (fr) * 1977-03-07 1979-03-23 Upjohn Co Nouveaux derives halogenes de prostaglandines et medicaments les contenant
FR2401921A1 (fr) * 1977-07-28 1979-03-30 Upjohn Co Derives de prostaglandines
EP0001270A1 (fr) * 1977-09-27 1979-04-04 Hoechst Aktiengesellschaft Analogues de la prostacycline, leurs procédés de préparation et leur utilisation pour le traitement des maladies de la circulation
EP0005768A1 (fr) * 1978-05-17 1979-12-12 The Wellcome Foundation Limited Formulations pharmaceutiques contenant des composés de prostaglandine et méthode pour leur fabrication
EP0013955A1 (fr) * 1979-01-25 1980-08-06 Hoechst Aktiengesellschaft Analogues de prostacycline, leurs intermédiaires, procédé pour leur préparation et des médicaments les contenant
EP0052204A1 (fr) * 1980-11-13 1982-05-26 American Cyanamid Company Analogues de prostacyclines de la série 1 et analogues apparentés
FR2513639A1 (fr) * 1981-09-25 1983-04-01 Squibb & Sons Inc Nouvelles prostacyclines dioxatricycliques utiles comme medicaments cardio-vasculaires et produits nouveaux utiles comme intermediaires pour leur synthese
EP0084775A1 (fr) * 1982-01-21 1983-08-03 MERCK PATENT GmbH 13-Thia-prostacyclines
WO2013024051A1 (fr) * 2011-08-12 2013-02-21 Ascendis Pharma A/S Composition à libération prolongée de prostacycline

Cited By (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2359125A1 (fr) * 1976-02-04 1978-02-17 Upjohn Co Nouveaux derives de prostaglandine, leur procede de preparation et medicament les contenant
FR2362833A1 (fr) * 1976-02-04 1978-03-24 Upjohn Co Nouveaux derives 5 de prostaglandine, leur procede de preparation et medicament les contenant
FR2378777A1 (fr) * 1977-01-31 1978-08-25 Ono Pharmaceutical Co Nouveaux analogues de prostaglandines
FR2401141A1 (fr) * 1977-03-07 1979-03-23 Upjohn Co Nouveaux derives halogenes de prostaglandines et medicaments les contenant
FR2401139A2 (fr) * 1977-03-07 1979-03-23 Upjohn Co Nouveaux derives d5 de prostaglandines, leur procede de preparation et medicaments les contenant
FR2401921A1 (fr) * 1977-07-28 1979-03-30 Upjohn Co Derives de prostaglandines
FR2401920A1 (fr) * 1977-07-28 1979-03-30 Upjohn Co Derives de prostaglandines
EP0001270A1 (fr) * 1977-09-27 1979-04-04 Hoechst Aktiengesellschaft Analogues de la prostacycline, leurs procédés de préparation et leur utilisation pour le traitement des maladies de la circulation
EP0005768A1 (fr) * 1978-05-17 1979-12-12 The Wellcome Foundation Limited Formulations pharmaceutiques contenant des composés de prostaglandine et méthode pour leur fabrication
FR2425856A1 (fr) * 1978-05-17 1979-12-14 Wellcome Found Medicament a base de prostaglandines
EP0013955A1 (fr) * 1979-01-25 1980-08-06 Hoechst Aktiengesellschaft Analogues de prostacycline, leurs intermédiaires, procédé pour leur préparation et des médicaments les contenant
EP0052204A1 (fr) * 1980-11-13 1982-05-26 American Cyanamid Company Analogues de prostacyclines de la série 1 et analogues apparentés
FR2513639A1 (fr) * 1981-09-25 1983-04-01 Squibb & Sons Inc Nouvelles prostacyclines dioxatricycliques utiles comme medicaments cardio-vasculaires et produits nouveaux utiles comme intermediaires pour leur synthese
EP0084775A1 (fr) * 1982-01-21 1983-08-03 MERCK PATENT GmbH 13-Thia-prostacyclines
WO2013024051A1 (fr) * 2011-08-12 2013-02-21 Ascendis Pharma A/S Composition à libération prolongée de prostacycline
US9872864B2 (en) 2011-08-12 2018-01-23 Ascendis Pharma A/S Sustained release composition of prostacyclin

Also Published As

Publication number Publication date
FR2351112B1 (fr) 1981-05-29

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