FR2258172A1 - 1-(2-Benzylaminoethyl) piperidines - with coronary vasodilator, spasmolytic, local anaesthetic, tranquillizing and uricosuric activity - Google Patents
1-(2-Benzylaminoethyl) piperidines - with coronary vasodilator, spasmolytic, local anaesthetic, tranquillizing and uricosuric activityInfo
- Publication number
- FR2258172A1 FR2258172A1 FR7402016A FR7402016A FR2258172A1 FR 2258172 A1 FR2258172 A1 FR 2258172A1 FR 7402016 A FR7402016 A FR 7402016A FR 7402016 A FR7402016 A FR 7402016A FR 2258172 A1 FR2258172 A1 FR 2258172A1
- Authority
- FR
- France
- Prior art keywords
- piperidines
- benzylaminoethyl
- tranquillizing
- spasmolytic
- local anaesthetic
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
- C07D295/125—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
- C07D295/13—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Hydrogenated Pyridines (AREA)
Abstract
1-(2-Aminoethyl)piperidines of formula (I): (where R is H or 1-4C alkyl; X is halogen, 1-4C alkyl, 1-4C alkoxy, or trihalomethyl) are coronary vasodilators, spasmolytics, local anaesthetics, tranquilizers and uricosuric agents.
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR7402016A FR2258172A1 (en) | 1974-01-22 | 1974-01-22 | 1-(2-Benzylaminoethyl) piperidines - with coronary vasodilator, spasmolytic, local anaesthetic, tranquillizing and uricosuric activity |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR7402016A FR2258172A1 (en) | 1974-01-22 | 1974-01-22 | 1-(2-Benzylaminoethyl) piperidines - with coronary vasodilator, spasmolytic, local anaesthetic, tranquillizing and uricosuric activity |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2258172A1 true FR2258172A1 (en) | 1975-08-18 |
FR2258172B1 FR2258172B1 (en) | 1978-02-03 |
Family
ID=9133779
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR7402016A Granted FR2258172A1 (en) | 1974-01-22 | 1974-01-22 | 1-(2-Benzylaminoethyl) piperidines - with coronary vasodilator, spasmolytic, local anaesthetic, tranquillizing and uricosuric activity |
Country Status (1)
Country | Link |
---|---|
FR (1) | FR2258172A1 (en) |
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0518216A2 (en) * | 1991-06-06 | 1992-12-16 | G.D. Searle & Co. | N-/Arylethyl/-N-alkyl-2-(1-pyrrolidinyl)ethylamine derivatives for CNS disorders |
US6787570B2 (en) | 1999-09-23 | 2004-09-07 | Pfizer, Inc. | Substituted N-cycloalkyl-N-benzyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity |
-
1974
- 1974-01-22 FR FR7402016A patent/FR2258172A1/en active Granted
Cited By (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0518216A2 (en) * | 1991-06-06 | 1992-12-16 | G.D. Searle & Co. | N-/Arylethyl/-N-alkyl-2-(1-pyrrolidinyl)ethylamine derivatives for CNS disorders |
WO1992022279A2 (en) * | 1991-06-06 | 1992-12-23 | G.D. Searle & Co. | N-[arylethyl]-n-alkyl-2-(1-pyrrolidinyl)ethylamine derivatives for cns disorders |
WO1992022279A3 (en) * | 1991-06-06 | 1993-03-04 | Searle & Co | N-[arylethyl]-n-alkyl-2-(1-pyrrolidinyl)ethylamine derivatives for cns disorders |
EP0518216A3 (en) * | 1991-06-06 | 1993-03-31 | G.D. Searle & Co. | N-/arylethyl/-n-alkyl-2-(1-pyrrolidinyl)ethylamine derivatives for cns disorders |
US6787570B2 (en) | 1999-09-23 | 2004-09-07 | Pfizer, Inc. | Substituted N-cycloalkyl-N-benzyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity |
Also Published As
Publication number | Publication date |
---|---|
FR2258172B1 (en) | 1978-02-03 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
TP | Transmission of property | ||
CD | Change of name or company name | ||
TP | Transmission of property | ||
ST | Notification of lapse |