FR2201080A1 - 2-imino-5-methylene-thiazolidine derivs - antiinflammatory antibacterial, antifungal and hypotensive - Google Patents

2-imino-5-methylene-thiazolidine derivs - antiinflammatory antibacterial, antifungal and hypotensive

Info

Publication number
FR2201080A1
FR2201080A1 FR7233711A FR7233711A FR2201080A1 FR 2201080 A1 FR2201080 A1 FR 2201080A1 FR 7233711 A FR7233711 A FR 7233711A FR 7233711 A FR7233711 A FR 7233711A FR 2201080 A1 FR2201080 A1 FR 2201080A1
Authority
FR
France
Prior art keywords
derivs
hypotensive
thiazolidine
imino
antifungal
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7233711A
Other languages
French (fr)
Other versions
FR2201080B1 (en
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
BASF SE
Original Assignee
BASF SE
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by BASF SE filed Critical BASF SE
Priority to FR7233711A priority Critical patent/FR2201080A1/en
Publication of FR2201080A1 publication Critical patent/FR2201080A1/en
Application granted granted Critical
Publication of FR2201080B1 publication Critical patent/FR2201080B1/fr
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
    • C07D277/42—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Title cpds. are of formula (I): (where R1 is lower alkyl, lower alkenyl, cycloalkyl, aryl or acyl; R2 and R3 are H or lower alkyl; R4 is H or 1-8C alkyl; or R3 + R4 can form a 4-6C spirocycloalkyl or 6-8C spirobicycloalkyl ring) and their salts, including the tautomeric 2-aminothiazoline form of (I; R2=H). They may be prepd. by (a) reacting R1NCS with R2NH-CR3R4-C triple bond CH to give R1NH-CS-NR2-CR3R4-C triple bond CH (II) and cyclising, or (b) reacting R1NH2 with SCN-CR3R4-C triple bond CH to give (IV; R2=H) and cyclising.
FR7233711A 1972-09-22 1972-09-22 2-imino-5-methylene-thiazolidine derivs - antiinflammatory antibacterial, antifungal and hypotensive Granted FR2201080A1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FR7233711A FR2201080A1 (en) 1972-09-22 1972-09-22 2-imino-5-methylene-thiazolidine derivs - antiinflammatory antibacterial, antifungal and hypotensive

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7233711A FR2201080A1 (en) 1972-09-22 1972-09-22 2-imino-5-methylene-thiazolidine derivs - antiinflammatory antibacterial, antifungal and hypotensive

Publications (2)

Publication Number Publication Date
FR2201080A1 true FR2201080A1 (en) 1974-04-26
FR2201080B1 FR2201080B1 (en) 1975-10-31

Family

ID=9104677

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7233711A Granted FR2201080A1 (en) 1972-09-22 1972-09-22 2-imino-5-methylene-thiazolidine derivs - antiinflammatory antibacterial, antifungal and hypotensive

Country Status (1)

Country Link
FR (1) FR2201080A1 (en)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2001019807A1 (en) * 1999-09-14 2001-03-22 Shionogi & Co., Ltd. 2-imino-1,3-thiazine derivatives

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
NEANT *

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2001019807A1 (en) * 1999-09-14 2001-03-22 Shionogi & Co., Ltd. 2-imino-1,3-thiazine derivatives
US6818640B1 (en) 1999-09-14 2004-11-16 Shionogi & Co., Ltd. 2-imino-1,3-thiazine derivatives
US7183275B2 (en) 1999-09-14 2007-02-27 Shionogi Co., Ltd. 2-imino-1,3-thiazine derivatives
US7420053B2 (en) 1999-09-14 2008-09-02 Shionogi & Co., Ltd. 2-imino-1,3-thiazine derivatives

Also Published As

Publication number Publication date
FR2201080B1 (en) 1975-10-31

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Legal Events

Date Code Title Description
ST Notification of lapse