FR2187356A1 - - Google Patents

Info

Publication number: FR2187356A1
Authority: FR; France
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Granted

Application number

FR7321443A

Other languages

French (fr)

Other versions

FR2187356B1 (en

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Merck and Co Inc

Original Assignee

Merck and Co Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1972-06-14

Filing date

1973-06-13

Publication date

1974-01-18

1973-06-13 Application filed by Merck and Co Inc filed Critical Merck and Co Inc

1974-01-18 Publication of FR2187356A1 publication Critical patent/FR2187356A1/fr

1977-01-28 Application granted granted Critical

1977-01-28 Publication of FR2187356B1 publication Critical patent/FR2187356B1/fr

Status Expired legal-status Critical Current

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/69—Two or more oxygen atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/61—Halogen atoms or nitro radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/63—One oxygen atom
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/79—Acids; Esters
- C07D213/80—Acids; Esters in position 3
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Pain & Pain Management (AREA)
Public Health (AREA)
Rheumatology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Pyridine Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

FR7321443A 1972-06-14 1973-06-13 Expired FR2187356B1 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US26289872A	1972-06-14	1972-06-14
BE147896A BE819177R (en)	1972-06-14	1974-08-26	OXAZOLO- AND THIAZOLOPYRIDINES

Publications (2)

Publication Number	Publication Date
FR2187356A1 true FR2187356A1 (en)	1974-01-18
FR2187356B1 FR2187356B1 (en)	1977-01-28

Family

ID=25648082

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
FR7321443A Expired FR2187356B1 (en)	1972-06-14	1973-06-13

Country Status (17)

Country	Link
JP (1)	JPS5943475B2 (en)
AR (1)	AR208500A1 (en)
AT (1)	AT333277B (en)
AU (1)	AU472528B2 (en)
BE (2)	BE800868A (en)
CA (1)	CA1019741A (en)
CS (1)	CS178889B2 (en)
DD (1)	DD105237A5 (en)
DE (1)	DE2330109A1 (en)
DK (1)	DK152050C (en)
FI (1)	FI57417C (en)
FR (1)	FR2187356B1 (en)
GB (1)	GB1421619A (en)
LU (1)	LU67786A1 (en)
NL (1)	NL184836C (en)
SE (2)	SE401675B (en)
ZA (1)	ZA733760B (en)

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2319354A1 (en) *	1975-07-29	1977-02-25	Merck & Co Inc	2-SUBSTITUTED OXAZOLOPYRIDINES
FR2406629A1 (en) *	1977-10-21	1979-05-18	Ishihara Mining & Chemical Co	5-TRIFLUOROMETHYLPYRIDINES SUBSTITUTED IN POSITION 2 AND THEIR PREPARATION PROCESS
FR2652085A1 (en) *	1989-09-20	1991-03-22	Science Organisation	NEW PROCESS FOR THE SYNTHESIS OF OXAZOLOPYRIDINE DERIVATIVES

Families Citing this family (29)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE2527321A1 (en) *	1975-06-19	1976-12-23	Merck & Co Inc	2-(Substd phenyl) oxazolo (4,5-b) pyridines - topical anti-inflammatories with very low systemic activity
JPS527992A (en) *	1975-07-04	1977-01-21	Merck & Co Inc	Oxazolo 455b* pyridines
NL187021C (en) *	1975-07-15	1991-05-01	Merck & Co Inc	PROCESS FOR THE PREPARATION OF A PHARMACEUTICAL PREPARATION WITH ANTI-INFLAMMATORY ACTION, AND A METHOD FOR PREPARING ANTI-INFLAMMATIC ACTIVITY 2-PHENYL-OXAZOLO-PID-BIDANE.
US4753673A (en) *	1977-07-22	1988-06-28	The Dow Chemical Company	Trifluoromethyl pyridinyloxyphenoxy and pyridinylthiophenoxy propanoic acids and propanols and derivatives thereof and methods of herbicidal use
EP0001473B1 (en) *	1977-08-12	1988-07-27	Imperial Chemical Industries Plc	Herbicidal halogenomethyl--pyridyloxy-phenoxy-alkanecarboxylic acids and derivatives, and processes of controlling unwanted plants therewith
JPS5461182A (en) *	1977-10-20	1979-05-17	Ishihara Sangyo Kaisha Ltd	2-phenoxy-5-trifluoromethylpyridine compounds
EP0003877B1 (en) *	1978-02-15	1988-02-03	Imperial Chemical Industries Plc	Herbicidal derivatives of 2-(4(2-pyridyloxy)phenoxy)propane, processes for preparing them, and herbicidal compositions containing them
JPS55130840U (en) *	1979-03-12	1980-09-16
JPS55124763A (en) *	1979-03-19	1980-09-26	Ishihara Sangyo Kaisha Ltd	5-trifluoromethyl-2-pyridone derivative
GB8333514D0 (en) *	1983-12-16	1984-01-25	Erba Farmitalia	Tetrahydrothiazolo(5 4-c)pyridine derivatives
PT937075E (en) *	1996-11-11	2004-05-31	Altana Pharma Ag	NEW IMIDAZO- AND OXAZOLO-PYRIDINES AS PHOSPHODIESTERESE INHIBITORS
SK18542000A3 (en) *	1998-06-04	2001-12-03	Abbott Laboratories	Cell adhesion-inhibiting anti-inflammatory compounds
US6232320B1 (en)	1998-06-04	2001-05-15	Abbott Laboratories	Cell adhesion-inhibiting antiinflammatory compounds
WO2000075145A1 (en) *	1999-06-03	2000-12-14	Abbott Laboratories	Cell adhesion-inhibiting antiinflammatory compounds
AU2002216649A1 (en) *	2000-10-31	2002-05-15	Lynn Bonham	Benzoxazole lpaat- beta inhibitors and uses thereof
US7855289B2 (en)	2005-08-04	2010-12-21	Sirtris Pharmaceuticals, Inc.	Sirtuin modulating compounds
US8093401B2 (en)	2005-08-04	2012-01-10	Sirtris Pharmaceuticals, Inc.	Sirtuin modulating compounds
US8088928B2 (en)	2005-08-04	2012-01-03	Sirtris Pharmaceuticals, Inc.	Sirtuin modulating compounds
WO2007019345A1 (en) *	2005-08-04	2007-02-15	Sirtris Pharmaceuticals, Inc.	Imidazopyridine derivatives as sirtuin modulating agents
TW200916472A (en)	2007-06-20	2009-04-16	Sirtris Pharmaceuticals Inc	Sirtuin modulating compounds
US8795630B2 (en) *	2008-08-29	2014-08-05	Treventis Corporation	Butyrylcholinesterase ligands as diagnostic tools and treatment for diseases of the nervous system
PE20120057A1 (en)	2008-12-19	2012-02-24	Sirtris Pharmaceuticals Inc	SIRTUINE MODULATING THIAZOLOPYRIDINE COMPOUNDS
EP2482660A4 (en) *	2009-09-30	2013-04-17	Sumitomo Chemical Co	Composition and method for controlling arthropod pests
KR20130051507A (en)	2010-09-15	2013-05-20	에프. 호프만-라 로슈 아게	Azabenzothiazole compounds, compositions and methods of use
BR112013016022B1 (en)	2010-12-24	2019-05-07	Sumitomo Chemical Company, Limited	Fused heterocyclic compound and use for same control.
WO2015200650A1 (en) *	2014-06-25	2015-12-30	Epizyme, Inc.	Substituted benzene and 6,5-fused bicyclic heteroaryl compounds
JP2017537909A (en)	2014-12-02	2017-12-21	バイエル・クロップサイエンス・アクチェンゲゼルシャフト	Bicyclic compounds as pest control agents The present application relates to novel bicyclic compounds, compositions containing these compounds, their use to control pests, and to prepare them And to intermediates.
WO2017127627A1 (en) *	2016-01-21	2017-07-27	The University Of North Carolina At Chapel Hill	Compounds for treatment of trypanosomes and neurological pathogens and uses thereof
KR102440762B1 (en) *	2016-07-07	2022-09-05	호도가야 가가쿠 고교 가부시키가이샤	A compound having a benzoazole ring structure and an organic electroluminescent device

1973
- 1973-03-12 AR AR248527A patent/AR208500A1/en active
- 1973-05-22 FI FI1657/73A patent/FI57417C/en active
- 1973-05-24 DK DK284973A patent/DK152050C/en not_active IP Right Cessation
- 1973-05-25 SE SE7307412A patent/SE401675B/en unknown
- 1973-05-30 NL NLAANVRAGE7307582,A patent/NL184836C/en not_active IP Right Cessation
- 1973-06-04 ZA ZA00733760A patent/ZA733760B/en unknown
- 1973-06-04 AU AU56511/73A patent/AU472528B2/en not_active Expired
- 1973-06-05 CA CA173,275A patent/CA1019741A/en not_active Expired
- 1973-06-08 AT AT508673A patent/AT333277B/en active
- 1973-06-11 GB GB2763273A patent/GB1421619A/en not_active Expired
- 1973-06-12 CS CS7300004243A patent/CS178889B2/en unknown
- 1973-06-12 DD DD171559A patent/DD105237A5/xx unknown
- 1973-06-13 LU LU67786A patent/LU67786A1/xx unknown
- 1973-06-13 BE BE132231A patent/BE800868A/en not_active IP Right Cessation
- 1973-06-13 FR FR7321443A patent/FR2187356B1/fr not_active Expired
- 1973-06-13 DE DE2330109A patent/DE2330109A1/en not_active Withdrawn
- 1973-06-14 JP JP48066453A patent/JPS5943475B2/en not_active Expired
1974
- 1974-08-26 BE BE147896A patent/BE819177R/en not_active IP Right Cessation
1976
- 1976-04-14 SE SE7604385A patent/SE432767B/en not_active IP Right Cessation

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
NEANT *

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2319354A1 (en) *	1975-07-29	1977-02-25	Merck & Co Inc	2-SUBSTITUTED OXAZOLOPYRIDINES
FR2406629A1 (en) *	1977-10-21	1979-05-18	Ishihara Mining & Chemical Co	5-TRIFLUOROMETHYLPYRIDINES SUBSTITUTED IN POSITION 2 AND THEIR PREPARATION PROCESS
FR2652085A1 (en) *	1989-09-20	1991-03-22	Science Organisation	NEW PROCESS FOR THE SYNTHESIS OF OXAZOLOPYRIDINE DERIVATIVES
EP0419348A1 (en) *	1989-09-20	1991-03-27	Science Et Organisation	Process for the synthesis of oxazolopyridinderivatives

Also Published As

Publication number	Publication date
NL184836B (en)	1989-06-16
SE7604385L (en)	1976-04-14
AT333277B (en)	1976-11-10
DK152050B (en)	1988-01-25
FI57417B (en)	1980-04-30
GB1421619A (en)	1976-01-21
LU67786A1 (en)	1973-08-16
SE432767B (en)	1984-04-16
AR208500A1 (en)	1977-02-15
BE800868A (en)	1973-12-13
JPS4961195A (en)	1974-06-13
ZA733760B (en)	1975-01-29
FR2187356B1 (en)	1977-01-28
AU472528B2 (en)	1976-05-27
JPS5943475B2 (en)	1984-10-22
ATA508673A (en)	1976-03-15
CS178889B2 (en)	1977-10-31
DK152050C (en)	1988-07-18
NL184836C (en)	1989-11-16
DD105237A5 (en)	1974-04-12
CA1019741A (en)	1977-10-25
BE819177R (en)	1975-02-26
AU5651173A (en)	1974-12-05
NL7307582A (en)	1973-12-18
FI57417C (en)	1980-08-11
DE2330109A1 (en)	1974-01-03
SE401675B (en)	1978-05-22

Legal Events

Date	Code	Title	Description
1993-04-30	ST	Notification of lapse

Publication	Publication Date	Title
FR2187356B1 (en)	1977-01-28
JPS4919878A (en)	1974-02-21
JPS48105333U (en)	1973-12-07
JPS4896535U (en)	1973-11-16
FR2194847A1 (en)	1974-03-01
JPS4890984A (en)	1973-11-27
JPS4953000U (en)	1974-05-10
JPS5146702Y2 (en)	1976-11-11
JPS5020410Y2 (en)	1975-06-20
HU169323B (en)	1976-11-28
JPS4987348U (en)	1974-07-29
JPS4955006U (en)	1974-05-15
JPS4919622U (en)	1974-02-19
BG27066A3 (en)	1979-08-15
CH591494A5 (en)	1977-09-30
BG17907A1 (en)	1974-03-05
BG18232A1 (en)	1974-10-25
BG20632A3 (en)	1975-12-05
BG21854A3 (en)	1976-09-20
BG21870A3 (en)	1976-09-20
CH574197A5 (en)	1976-03-31
NL7312059A (en)	1974-03-05
CH1336273A4 (en)	1975-02-28
CH1654373A4 (en)	1975-06-30
SE7103088L (en)	1972-03-10