FR1520743A - Nouvelles quinazolinones substituées et procédé de préparation - Google Patents

Nouvelles quinazolinones substituées et procédé de préparation

Info

Publication number
FR1520743A
FR1520743A FR97203A FR97203A FR1520743A FR 1520743 A FR1520743 A FR 1520743A FR 97203 A FR97203 A FR 97203A FR 97203 A FR97203 A FR 97203A FR 1520743 A FR1520743 A FR 1520743A
Authority
FR
France
Prior art keywords
preparation
novel substituted
substituted quinazolinones
quinazolinones
novel
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
FR97203A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Aventis France
Original Assignee
Roussel Uclaf SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to FR85985A priority Critical patent/FR6001M/fr
Application filed by Roussel Uclaf SA filed Critical Roussel Uclaf SA
Priority to FR97203A priority patent/FR1520743A/fr
Priority to FR106810A priority patent/FR6158M/fr
Priority to IL2899167A priority patent/IL28991A/xx
Priority to CH1645167A priority patent/CH482685A/fr
Priority to NL6716429A priority patent/NL6716429A/xx
Priority to DK603267A priority patent/DK127332B/da
Priority to DE1967R0047487 priority patent/DE1695656B2/de
Priority to GB55090/67A priority patent/GB1181570A/en
Application granted granted Critical
Publication of FR1520743A publication Critical patent/FR1520743A/fr
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/78Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 2
    • C07D239/80Oxygen atoms
    • C07D239/82Oxygen atoms with an aryl radical attached in position 4
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/78Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 2
    • C07D239/80Oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
FR97203A 1966-12-02 1967-03-02 Nouvelles quinazolinones substituées et procédé de préparation Expired FR1520743A (fr)

Priority Applications (9)

Application Number Priority Date Filing Date Title
FR85985A FR6001M (fr) 1966-12-02 1966-12-02
FR97203A FR1520743A (fr) 1966-12-02 1967-03-02 Nouvelles quinazolinones substituées et procédé de préparation
FR106810A FR6158M (fr) 1966-12-02 1967-05-18
IL2899167A IL28991A (en) 1966-12-02 1967-11-21 Substituted quinazolinones and process of preparation thereof
CH1645167A CH482685A (fr) 1966-12-02 1967-11-23 Procédé de préparation de nouvelles quinazolinones substituées
NL6716429A NL6716429A (fr) 1966-12-02 1967-12-01
DK603267A DK127332B (da) 1966-12-02 1967-12-01 Analogifremgangsmåde til fremstilling af terapeutisk virksomme 1-substituerede 2[1H]-quinazolinoner.
DE1967R0047487 DE1695656B2 (de) 1966-12-02 1967-12-01 l-Alkyl-4-aryl-2(lH)-chinazoIinone
GB55090/67A GB1181570A (en) 1966-12-02 1967-12-04 Substituted Quinazolinones

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
FR85985A FR6001M (fr) 1966-12-02 1966-12-02
FR97203A FR1520743A (fr) 1966-12-02 1967-03-02 Nouvelles quinazolinones substituées et procédé de préparation
FR106810A FR6158M (fr) 1966-12-02 1967-05-18
FR125422 1967-10-23

Publications (1)

Publication Number Publication Date
FR1520743A true FR1520743A (fr) 1968-04-12

Family

ID=27444746

Family Applications (3)

Application Number Title Priority Date Filing Date
FR85985A Expired FR6001M (fr) 1966-12-02 1966-12-02
FR97203A Expired FR1520743A (fr) 1966-12-02 1967-03-02 Nouvelles quinazolinones substituées et procédé de préparation
FR106810A Expired FR6158M (fr) 1966-12-02 1967-05-18

Family Applications Before (1)

Application Number Title Priority Date Filing Date
FR85985A Expired FR6001M (fr) 1966-12-02 1966-12-02

Family Applications After (1)

Application Number Title Priority Date Filing Date
FR106810A Expired FR6158M (fr) 1966-12-02 1967-05-18

Country Status (7)

Country Link
CH (1) CH482685A (fr)
DE (1) DE1695656B2 (fr)
DK (1) DK127332B (fr)
FR (3) FR6001M (fr)
GB (1) GB1181570A (fr)
IL (1) IL28991A (fr)
NL (1) NL6716429A (fr)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1932402A1 (de) * 1969-06-26 1970-03-05 Sandoz Ag Heterocyclische Verbindungen und Verfahren zu ihrer Herstellung
US3764600A (en) * 1970-10-06 1973-10-09 Sandoz Ag 1-substituted-quinazoline-2(1h)-thiones
USB252947I5 (fr) * 1968-07-18 1975-01-28
USB368862I5 (fr) * 1970-10-06 1975-01-28

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2118315C3 (de) * 1970-04-20 1975-04-03 Sumitomo Chemical Co., Ltd., Osaka (Japan) 2-(1H)-Chinazolinonderivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel
US4071516A (en) 1976-08-20 1978-01-31 Sandoz, Inc. 4-(Acyloxyphenyl)-quinazolin-2(1H)-ones
AR038658A1 (es) 2001-06-15 2005-01-26 Novartis Ag Derivados de 4-aril-2(1h) quinazolinona y 4-aril-quinazolina 2-sustituidas, un proceso para su preparacion, composiciones farmaceuticas y el uso de dichos derivados para la preparacion de un medicamento
GB0230015D0 (en) 2002-12-23 2003-01-29 Novartis Ag Organic compounds
CN104364237B (zh) * 2012-04-10 2016-08-24 安基生技新药股份有限公司 组蛋白去乙酰化酶(hdacs)抑制剂

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
USB252947I5 (fr) * 1968-07-18 1975-01-28
DE1932402A1 (de) * 1969-06-26 1970-03-05 Sandoz Ag Heterocyclische Verbindungen und Verfahren zu ihrer Herstellung
US3764600A (en) * 1970-10-06 1973-10-09 Sandoz Ag 1-substituted-quinazoline-2(1h)-thiones
USB368862I5 (fr) * 1970-10-06 1975-01-28
US3925549A (en) * 1970-10-06 1975-12-09 Sandoz Ag 1-Substituted-quinazoline-2(1H)-thiones in the treatment of inflammation

Also Published As

Publication number Publication date
IL28991A (en) 1972-11-28
FR6158M (fr) 1968-07-01
DK127332B (da) 1973-10-22
CH482685A (fr) 1969-12-15
FR6001M (fr) 1968-04-29
NL6716429A (fr) 1968-06-04
DE1695656C3 (fr) 1979-12-06
GB1181570A (en) 1970-02-18
DE1695656B2 (de) 1974-06-06
DE1695656A1 (de) 1972-04-13

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