FI972720A0 - Förfarande för framställning av lamotrigin - Google Patents

Förfarande för framställning av lamotrigin

Info

Publication number
FI972720A0
FI972720A0 FI972720A FI972720A FI972720A0 FI 972720 A0 FI972720 A0 FI 972720A0 FI 972720 A FI972720 A FI 972720A FI 972720 A FI972720 A FI 972720A FI 972720 A0 FI972720 A0 FI 972720A0
Authority
FI
Finland
Prior art keywords
preparing lamotrigine
lamotrigine
preparing
Prior art date
Application number
FI972720A
Other languages
English (en)
Finnish (fi)
Other versions
FI972720A (sv
Inventor
Grahame Roy Lee
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wellcome Found filed Critical Wellcome Found
Publication of FI972720A0 publication Critical patent/FI972720A0/sv
Publication of FI972720A publication Critical patent/FI972720A/sv

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D253/00Heterocyclic compounds containing six-membered rings having three nitrogen atoms as the only ring hetero atoms, not provided for by group C07D251/00
    • C07D253/02Heterocyclic compounds containing six-membered rings having three nitrogen atoms as the only ring hetero atoms, not provided for by group C07D251/00 not condensed with other rings
    • C07D253/061,2,4-Triazines
    • C07D253/0651,2,4-Triazines having three double bonds between ring members or between ring members and non-ring members
    • C07D253/071,2,4-Triazines having three double bonds between ring members or between ring members and non-ring members with hetero atoms, or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D253/075Two hetero atoms, in positions 3 and 5
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D253/00Heterocyclic compounds containing six-membered rings having three nitrogen atoms as the only ring hetero atoms, not provided for by group C07D251/00
    • C07D253/02Heterocyclic compounds containing six-membered rings having three nitrogen atoms as the only ring hetero atoms, not provided for by group C07D251/00 not condensed with other rings
    • C07D253/061,2,4-Triazines
    • C07D253/0651,2,4-Triazines having three double bonds between ring members or between ring members and non-ring members
    • C07D253/071,2,4-Triazines having three double bonds between ring members or between ring members and non-ring members with hetero atoms, or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FI972720A 1994-12-30 1997-06-24 Förfarande för framställning av lamotrigin FI972720A (sv)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9426448.8A GB9426448D0 (en) 1994-12-30 1994-12-30 Process
PCT/GB1995/003049 WO1996020935A1 (en) 1994-12-30 1995-12-29 Process for the preparation of lamotrigine

Publications (2)

Publication Number Publication Date
FI972720A0 true FI972720A0 (sv) 1997-06-24
FI972720A FI972720A (sv) 1997-08-27

Family

ID=10766744

Family Applications (1)

Application Number Title Priority Date Filing Date
FI972720A FI972720A (sv) 1994-12-30 1997-06-24 Förfarande för framställning av lamotrigin

Country Status (9)

Country Link
US (1) US5925755A (sv)
EP (1) EP0800521A1 (sv)
JP (1) JPH11507011A (sv)
AU (1) AU4311696A (sv)
FI (1) FI972720A (sv)
GB (1) GB9426448D0 (sv)
HU (1) HUT77347A (sv)
RU (1) RU2162081C2 (sv)
WO (1) WO1996020935A1 (sv)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9512854D0 (en) * 1995-06-23 1995-08-23 Wellcome Found Novel formulation
GB9726987D0 (en) 1997-12-22 1998-02-18 Glaxo Group Ltd Compounds
US6420354B1 (en) 1998-06-08 2002-07-16 Advanced Medicine, Inc. Sodium channel drugs and uses
GB9812413D0 (en) * 1998-06-10 1998-08-05 Glaxo Group Ltd Compound and its use
US6479498B1 (en) 1999-06-04 2002-11-12 Theravance, Inc. Sodium channel drugs and uses
AU763244B2 (en) * 2000-01-03 2003-07-17 Rpg Life Sciences Limited A process for the preparation of 6-(2,3-dichlorophenyl)-1,2,4-triazine-3,5-diamine, commonly known as lamotrigine
IL157608A0 (en) * 2001-02-27 2004-03-28 Teva Pharma New crystal forms of lamotrigine and processes for their preparations
BRPI0211844B8 (pt) 2001-08-10 2021-05-25 Nippon Chemiphar Co composto de ácido fenóxi-acético ou um de seus sais farmaceuticamente aceitáveis, e, composição farmacêutica
JP4276074B2 (ja) 2001-10-12 2009-06-10 日本ケミファ株式会社 ペルオキシソーム増殖剤応答性受容体δの活性化剤
CA2366521C (en) 2001-12-24 2007-03-06 Brantford Chemicals Inc. A new and efficient process for the preparation of lamotrigine and related 3,5-diamino-6-substituted-1,2,4-triazines
WO2003090693A2 (en) * 2002-04-23 2003-11-06 Teva Pharmaceutical Industries Ltd. Pharmaceutical composition containing lamotrigine particles of defined morphology
HU225667B1 (en) 2002-09-20 2007-05-29 Richter Gedeon Nyrt Method for producing high-purity 3,5-diamino-6-(2,3-dichlorophenyl)-1,2,4-triazine
JP5290749B2 (ja) 2006-04-18 2013-09-18 日本ケミファ株式会社 ペルオキシソーム増殖剤活性化受容体δの活性化剤
US20120142919A1 (en) 2006-08-02 2012-06-07 Medichem, S.A. Method for synthesizing lamotrigine
WO2009061513A1 (en) 2007-11-09 2009-05-14 Thar Pharmaceuticals Crystalline forms of lamotrigine
ES2683012T3 (es) 2008-04-15 2018-09-24 Nippon Chemiphar Co., Ltd. Agente activador para el receptor activado por proliferadores de peroxisomas

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU530999B2 (en) * 1979-06-01 1983-08-04 Wellcome Foundation Limited, The Substituted amino triazines and their use in treatment of cns disorders

Also Published As

Publication number Publication date
HUT77347A (hu) 1998-03-30
EP0800521A1 (en) 1997-10-15
RU2162081C2 (ru) 2001-01-20
US5925755A (en) 1999-07-20
FI972720A (sv) 1997-08-27
WO1996020935A1 (en) 1996-07-11
AU4311696A (en) 1996-07-24
JPH11507011A (ja) 1999-06-22
GB9426448D0 (en) 1995-03-01

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Legal Events

Date Code Title Description
FD Application lapsed