FI935700A0 - Antibakteriella azaspirokinoloner - Google Patents

Antibakteriella azaspirokinoloner

Info

Publication number
FI935700A0
FI935700A0 FI935700A FI935700A FI935700A0 FI 935700 A0 FI935700 A0 FI 935700A0 FI 935700 A FI935700 A FI 935700A FI 935700 A FI935700 A FI 935700A FI 935700 A0 FI935700 A0 FI 935700A0
Authority
FI
Finland
Prior art keywords
pct
antibacterial
azaspiroquinoloner
sec
date
Prior art date
Application number
FI935700A
Other languages
English (en)
Other versions
FI102900B1 (fi
FI102900B (fi
FI935700A (fi
Inventor
Bingwei Vera Yang
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI935700A0 publication Critical patent/FI935700A0/fi
Publication of FI935700A publication Critical patent/FI935700A/fi
Application granted granted Critical
Publication of FI102900B1 publication Critical patent/FI102900B1/fi
Publication of FI102900B publication Critical patent/FI102900B/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Materials For Medical Uses (AREA)
FI935700A 1991-06-19 1993-12-17 Menetelmä terapeuttisesti aktiivisten kinoliini- ja naftyridiinijohdan naisten valmistamiseksi FI102900B (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US71755291A 1991-06-19 1991-06-19
US71755291 1991-06-19
US9203453 1992-05-04
PCT/US1992/003453 WO1992022550A1 (en) 1991-06-19 1992-05-04 Azaspiro quinolone antibacterial agents

Publications (4)

Publication Number Publication Date
FI935700A0 true FI935700A0 (fi) 1993-12-17
FI935700A FI935700A (fi) 1993-12-17
FI102900B1 FI102900B1 (fi) 1999-03-15
FI102900B FI102900B (fi) 1999-03-15

Family

ID=24882485

Family Applications (2)

Application Number Title Priority Date Filing Date
FI935700A FI102900B (fi) 1991-06-19 1993-12-17 Menetelmä terapeuttisesti aktiivisten kinoliini- ja naftyridiinijohdan naisten valmistamiseksi
FI982097A FI982097A (fi) 1991-06-19 1998-09-29 Antibakteerisia atsaspirokinoloneja

Family Applications After (1)

Application Number Title Priority Date Filing Date
FI982097A FI982097A (fi) 1991-06-19 1998-09-29 Antibakteerisia atsaspirokinoloneja

Country Status (13)

Country Link
US (1) US5407943A (fi)
EP (1) EP0641339B1 (fi)
JP (1) JPH0678335B2 (fi)
AT (1) ATE184603T1 (fi)
CA (1) CA2111463C (fi)
DE (1) DE69230005T2 (fi)
DK (1) DK0641339T3 (fi)
ES (1) ES2136086T3 (fi)
FI (2) FI102900B (fi)
GR (1) GR3031701T3 (fi)
IE (1) IE921970A1 (fi)
PT (1) PT100597B (fi)
WO (1) WO1992022550A1 (fi)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6664271B1 (en) * 1999-05-21 2003-12-16 Eli Lilly And Company Immunopotentiator agents
US7902227B2 (en) 2007-07-27 2011-03-08 Janssen Pharmaceutica Nv. C-7 isoxazolinyl quinolone / naphthyridine derivatives useful as antibacterial agents
FR2941696B1 (fr) 2009-02-05 2011-04-15 Sanofi Aventis Derives d'azaspiranyl-alkylcarbamates d'heterocycles a 5 chainons, leur preparation et leur application en therapeutique
FR2945531A1 (fr) 2009-05-12 2010-11-19 Sanofi Aventis Derives de 7-aza-spiro°3,5!nonane-7-carboxylates, leur preparation et leur application en therapeutique
WO2012047703A2 (en) * 2010-10-04 2012-04-12 Schering Corporation Cyclopropyl-spiro-piperidines useful as sodium channel blockers

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4571396A (en) * 1984-04-16 1986-02-18 Warner-Lambert Company Antibacterial agents
JPH0676400B2 (ja) * 1987-08-25 1994-09-28 大日本製薬株式会社 新規ピリドンカルボン酸誘導体、そのエステルおよびその塩
MY105136A (en) * 1988-04-27 1994-08-30 Daiichi Seiyaku Co Optically active pyridonecarboxylic acid derivatives.
CA1336090C (en) * 1988-08-31 1995-06-27 Isao Hayakawa Spiro-substituted cyclic amines of quinolone derivatives
CA2012681A1 (en) * 1989-03-31 1990-09-30 Masayasu Okuhira Quinolone derivatives, preparation processes thereof, and antibacterial agents containing the same
HU219403B (hu) * 1989-08-16 2001-04-28 Pfizer Inc. Azabiciklo-csoporttal helyettesített kinolon- és naftiridon-karbonsavak és eljárás ezek előállítására

Also Published As

Publication number Publication date
FI982097A0 (fi) 1998-09-29
IE921970A1 (en) 1992-12-30
FI102900B1 (fi) 1999-03-15
FI982097A (fi) 1998-09-29
ES2136086T3 (es) 1999-11-16
ATE184603T1 (de) 1999-10-15
EP0641339A1 (en) 1995-03-08
EP0641339B1 (en) 1999-09-15
DE69230005T2 (de) 2000-01-05
JPH06503355A (ja) 1994-04-14
DE69230005D1 (de) 1999-10-21
DK0641339T3 (da) 1999-12-20
CA2111463A1 (en) 1992-12-23
US5407943A (en) 1995-04-18
GR3031701T3 (en) 2000-02-29
CA2111463C (en) 1997-08-26
FI102900B (fi) 1999-03-15
WO1992022550A1 (en) 1992-12-23
PT100597A (pt) 1993-09-30
FI935700A (fi) 1993-12-17
PT100597B (pt) 1999-07-30
JPH0678335B2 (ja) 1994-10-05

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Legal Events

Date Code Title Description
MA Patent expired