FI905225A0 - Menetelmä 1-//1-/2-(trifluorimetyyli)-4-pyrimidinyyli/-4-piperidinyyli/metyyli/-2-pyrrolidinonin valmistamiseksi suuressa mittakaavassa - Google Patents

Menetelmä 1-//1-/2-(trifluorimetyyli)-4-pyrimidinyyli/-4-piperidinyyli/metyyli/-2-pyrrolidinonin valmistamiseksi suuressa mittakaavassa

Info

Publication number
FI905225A0
FI905225A0 FI905225A FI905225A FI905225A0 FI 905225 A0 FI905225 A0 FI 905225A0 FI 905225 A FI905225 A FI 905225A FI 905225 A FI905225 A FI 905225A FI 905225 A0 FI905225 A0 FI 905225A0
Authority
FI
Finland
Prior art keywords
pyrrolidinone
piperidinyl
pyrimidinyl
trifluoromethyl
methyl
Prior art date
Application number
FI905225A
Other languages
English (en)
Swedish (sv)
Other versions
FI95467B (fi
FI95467C (fi
Inventor
Gary D Madding
Joseph L Minielli
Ronald J Mattson
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of FI905225A0 publication Critical patent/FI905225A0/fi
Publication of FI95467B publication Critical patent/FI95467B/fi
Application granted granted Critical
Publication of FI95467C publication Critical patent/FI95467C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Silicon Polymers (AREA)
  • Macromonomer-Based Addition Polymer (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Catalysts (AREA)
FI905225A 1989-10-27 1990-10-24 Menetelmä 1-//1-/2-(trifluorimetyyli)-4-pyrimidinyyli/-4-piperidinyyli/metyyli/-2-pyrrolidinonin valmistamiseksi suuressa mittakaavassa FI95467C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US07/427,546 US4963678A (en) 1989-10-27 1989-10-27 Process for large-scale production of BMY 21502
US42754689 1989-10-27

Publications (3)

Publication Number Publication Date
FI905225A0 true FI905225A0 (fi) 1990-10-24
FI95467B FI95467B (fi) 1995-10-31
FI95467C FI95467C (fi) 1996-02-12

Family

ID=23695332

Family Applications (1)

Application Number Title Priority Date Filing Date
FI905225A FI95467C (fi) 1989-10-27 1990-10-24 Menetelmä 1-//1-/2-(trifluorimetyyli)-4-pyrimidinyyli/-4-piperidinyyli/metyyli/-2-pyrrolidinonin valmistamiseksi suuressa mittakaavassa

Country Status (12)

Country Link
US (1) US4963678A (fi)
KR (1) KR910007917A (fi)
CN (1) CN1032916C (fi)
AT (1) AT397961B (fi)
EG (1) EG19764A (fi)
ES (1) ES2026059A6 (fi)
FI (1) FI95467C (fi)
GR (1) GR1001125B (fi)
HU (1) HU206878B (fi)
NO (1) NO177303C (fi)
PT (1) PT95711B (fi)
YU (1) YU203290A (fi)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI95468C (fi) * 1989-10-27 1996-02-12 Squibb Bristol Myers Co Parannettu menetelmä käyttökelpoisten piperidiinijohdannaisten valmistamiseksi
US4963678A (en) * 1989-10-27 1990-10-16 Bristol-Myers Squibb Co. Process for large-scale production of BMY 21502
US5098904A (en) * 1990-06-27 1992-03-24 Bristol-Myers Squibb Company Cerebral function enhancing pyrimidinyl derivatives
US5401744A (en) * 1993-10-04 1995-03-28 Bristol-Myers Squibb Company Useful hemi-hydrate form of a cerebral function enhancing agent
US5538985A (en) * 1994-01-27 1996-07-23 Mitsui Toatsu Chemicals, Inc. Pyrrolidinone derivatives
SK11422003A3 (sk) 2001-03-15 2004-04-06 Basf Aktiengesellschaft 5-Fenylpyrimidíny, spôsoby a medziprodukty na ich prípravu a ich použitie pri ničení škodlivých húb
US7073271B2 (en) * 2002-02-14 2006-07-11 Faro Technologies Inc. Portable coordinate measurement machine
CN106883185B (zh) * 2015-12-15 2021-07-09 重庆博腾制药科技股份有限公司 一种4-氯-2-三氟甲基嘧啶的制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ216720A (en) * 1985-07-08 1990-09-26 Bristol Myers Co Diazinylpiperidine derivatives and pharmaceutical compositions
US4826843A (en) * 1985-07-08 1989-05-02 Bristol-Myers Cerebral function enhancing diazinylpiperidine derivatives
DE3703103A1 (de) * 1987-02-03 1988-08-11 Bayer Ag Mittel gegen fischparsiten
US4963678A (en) * 1989-10-27 1990-10-16 Bristol-Myers Squibb Co. Process for large-scale production of BMY 21502

Also Published As

Publication number Publication date
GR1001125B (el) 1993-04-28
EG19764A (en) 1996-01-31
NO904587L (no) 1991-04-29
ES2026059A6 (es) 1992-04-01
FI95467B (fi) 1995-10-31
FI95467C (fi) 1996-02-12
PT95711B (pt) 1997-12-31
US4963678A (en) 1990-10-16
GR900100776A (en) 1992-03-20
CN1051175A (zh) 1991-05-08
CN1032916C (zh) 1996-10-02
NO177303B (no) 1995-05-15
ATA212290A (de) 1993-12-15
PT95711A (pt) 1991-09-13
HU910050D0 (en) 1991-08-28
HU206878B (en) 1993-01-28
NO904587D0 (no) 1990-10-24
KR910007917A (ko) 1991-05-30
AT397961B (de) 1994-08-25
NO177303C (no) 1995-08-23
YU203290A (sh) 1993-10-20

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Legal Events

Date Code Title Description
BB Publication of examined application
FG Patent granted

Owner name: BRISTOL-MYERS SQUIBB COMPANY