FI854862A0 - Nya pteridiner, foerfarande foer deras framstaellning och deras anvaendning saosom mellanprodukter eller saosom laekemedel. - Google Patents

Nya pteridiner, foerfarande foer deras framstaellning och deras anvaendning saosom mellanprodukter eller saosom laekemedel.

Info

Publication number
FI854862A0
FI854862A0 FI854862A FI854862A FI854862A0 FI 854862 A0 FI854862 A0 FI 854862A0 FI 854862 A FI854862 A FI 854862A FI 854862 A FI854862 A FI 854862A FI 854862 A0 FI854862 A0 FI 854862A0
Authority
FI
Finland
Prior art keywords
saosom
deras
pteridiner
nya
eller
Prior art date
Application number
FI854862A
Other languages
English (en)
Other versions
FI854862A (fi
FI82696C (fi
FI82696B (fi
Inventor
Josef Roch
Armin Heckel
Josef Nickl
Erich Mueller
Berthold Narr
Rainer Zimmermann
Johannes Weisenberger
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of FI854862A0 publication Critical patent/FI854862A0/fi
Publication of FI854862A publication Critical patent/FI854862A/fi
Application granted granted Critical
Publication of FI82696B publication Critical patent/FI82696B/fi
Publication of FI82696C publication Critical patent/FI82696C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D475/00Heterocyclic compounds containing pteridine ring systems
    • C07D475/06Heterocyclic compounds containing pteridine ring systems with a nitrogen atom directly attached in position 4
    • C07D475/08Heterocyclic compounds containing pteridine ring systems with a nitrogen atom directly attached in position 4 with a nitrogen atom directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Hematology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
FI854862A 1984-12-12 1985-12-10 Foerfarande foer framstaellning av farmakologiskt vaerdefulla pteridiner. FI82696C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19843445298 DE3445298A1 (de) 1984-12-12 1984-12-12 Neue pteridine, verfahren zu ihrer herstellung und deren verwendung als zwischenprodukte oder als arzneimittel
DE3445298 1984-12-12

Publications (4)

Publication Number Publication Date
FI854862A0 true FI854862A0 (fi) 1985-12-10
FI854862A FI854862A (fi) 1986-06-13
FI82696B FI82696B (fi) 1990-12-31
FI82696C FI82696C (fi) 1991-04-10

Family

ID=6252576

Family Applications (1)

Application Number Title Priority Date Filing Date
FI854862A FI82696C (fi) 1984-12-12 1985-12-10 Foerfarande foer framstaellning av farmakologiskt vaerdefulla pteridiner.

Country Status (15)

Country Link
EP (1) EP0185259A3 (fi)
JP (1) JPS61140585A (fi)
AU (1) AU576924B2 (fi)
CA (1) CA1252783A (fi)
DE (1) DE3445298A1 (fi)
DK (1) DK161327C (fi)
ES (1) ES8707238A1 (fi)
FI (1) FI82696C (fi)
GR (1) GR852996B (fi)
IL (1) IL77294A (fi)
NO (1) NO161373C (fi)
NZ (1) NZ214522A (fi)
PH (1) PH24451A (fi)
PT (1) PT81650B (fi)
ZA (1) ZA859462B (fi)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7276506B2 (en) 1998-12-28 2007-10-02 4 Aza Bioscience Nv Immunosuppressive effects of pteridine derivatives
EE200400042A (et) * 2001-06-28 2004-10-15 Essential Therapeutics, Inc. 8/17 heterotsüklilised ühendid ning nende kasutamine D-alanüül-D-alaniini ligaasi inhibiitoritena
DE10202468A1 (de) * 2002-01-23 2004-09-30 Faustus Forschungs Cie. Translational Cancer Research Gmbh Pteridinderivate, Verfahren zu deren Herstellung und ihre Verwendung
DE602004009696T2 (de) * 2003-08-29 2008-08-28 4 Aza Ip Nv Immunosuppressive wirkungen von pteridinderivativen
GB2407089A (en) * 2003-10-17 2005-04-20 4 Aza Bioscience Nv Pteridine derivatives
AU2004283479A1 (en) * 2003-10-17 2005-05-06 4 Aza Bioscience Nv Heterocycle-substituted pteridine derivatives and their use in therapy
CN1950081A (zh) * 2004-03-04 2007-04-18 神经能质公司 芳烷氨基取代的喹唑啉类似物
DE102004057618A1 (de) 2004-11-29 2006-06-01 Boehringer Ingelheim Pharma Gmbh & Co. Kg Substituierte Pteridine zur Behandlung von entzündlichen Erkrankungen
DE102004057595A1 (de) 2004-11-29 2006-06-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg Substituierte Pteridine zur Behandlung von entzündlichen Erkrankungen
DE102004057594A1 (de) * 2004-11-29 2006-06-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg Substitueirte Pteridine zur Behandlung von entzündlichen Erkrankungen
DE102004057645A1 (de) 2004-11-29 2006-06-01 Boehringer Ingelheim Pharma Gmbh & Co. Kg Substituierte Pteridine zur Behandlung von entzündlichen Erkrankungen
WO2007060404A1 (en) * 2005-11-22 2007-05-31 Kudos Pharmaceuticals Limited PYRIDO-,PYRAZO- AND PYRIMIDO-PYRIMIDINE DERIVATIVES AS mTOR INHIBITORS
RU2445315C2 (ru) * 2005-11-22 2012-03-20 Кудос Фармасьютиклз Лимитед ПРОИЗВОДНЫЕ ПИРИДО-, ПИРАЗО- И ПИРИМИДО-ПИРИМИДИНА И ИХ ПРИМЕНЕНИЕ В КАЧЕСТВЕ ИНГИБИТОРОВ mTOR
CA2652840C (en) 2006-05-24 2014-09-09 Boehringer Ingelheim International Gmbh 2-piperazino-6-chloro-pteridines as pde4-inhibitors for the treatment of inflammatory diseases
US10144736B2 (en) 2006-07-20 2018-12-04 Gilead Sciences, Inc. Substituted pteridines useful for the treatment and prevention of viral infections
LT2057156T (lt) 2006-08-23 2017-05-25 Kudos Pharmaceuticals Limited 2-metilmorfolino pirido-, pirazo- ir pirimidopirimidino dariniai kaip mtor slopikliai
MX2010014230A (es) 2008-06-20 2011-03-29 Astrazeneca Ab Composiciones que contienen pirido [2,3-d] pirimidinas sustituidas con metilmorfolina y proceso relacionado.
CU20180011A7 (es) 2015-03-04 2018-06-05 Gilead Sciences Inc Composiciones farmacéuticas que comprenden compuestos derivados de diaminopirido (3,2-d) como moduladores de receptor de tipo toll
WO2018045150A1 (en) 2016-09-02 2018-03-08 Gilead Sciences, Inc. 4,6-diamino-pyrido[3,2-d]pyrimidine derivaties as toll like receptor modulators
PL3507276T3 (pl) 2016-09-02 2022-02-21 Gilead Sciences, Inc. Związki modulatory receptorów toll-podobnych
TWI751517B (zh) 2019-04-17 2022-01-01 美商基利科學股份有限公司 類鐸受體調節劑之固體形式
TWI751516B (zh) 2019-04-17 2022-01-01 美商基利科學股份有限公司 類鐸受體調節劑之固體形式
TW202115056A (zh) 2019-06-28 2021-04-16 美商基利科學股份有限公司 類鐸受體調節劑化合物的製備方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3159628A (en) * 1962-05-28 1964-12-01 Smith Kline French Lab Pteridine-5-oxide derivatives
DE3323932A1 (de) * 1983-07-02 1985-01-10 Dr. Karl Thomae Gmbh, 7950 Biberach Neue 2-piperazino-pteridine, verfahren zu ihrer herstellung und diese verbindung enthaltende arzneimittel

Also Published As

Publication number Publication date
FI854862A (fi) 1986-06-13
NO161373B (no) 1989-05-02
ZA859462B (en) 1987-07-29
JPS61140585A (ja) 1986-06-27
CA1252783A (en) 1989-04-18
GR852996B (fi) 1986-04-16
EP0185259A3 (de) 1989-03-01
DK572685D0 (da) 1985-12-11
ES8707238A1 (es) 1987-07-16
DE3445298A1 (de) 1986-06-12
NZ214522A (en) 1988-07-28
DK572685A (da) 1986-06-13
DK161327C (da) 1991-12-09
IL77294A (en) 1989-02-28
PT81650B (pt) 1988-04-21
NO161373C (no) 1989-08-09
AU576924B2 (en) 1988-09-08
PT81650A (de) 1986-01-01
NO854965L (no) 1986-06-13
DK161327B (da) 1991-06-24
FI82696C (fi) 1991-04-10
PH24451A (en) 1990-06-25
FI82696B (fi) 1990-12-31
EP0185259A2 (de) 1986-06-25
ES549806A0 (es) 1987-07-16
AU5123285A (en) 1986-06-19

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Legal Events

Date Code Title Description
MM Patent lapsed

Owner name: DR. KARL THOMAE GESELLSCHAFT MIT