FI58136C - Foerfarande foer framstaellning av terapeutiskt anvaendbara 16-deacetoxi-16alfa-acyltiofusidinsyraderivat - Google Patents
Foerfarande foer framstaellning av terapeutiskt anvaendbara 16-deacetoxi-16alfa-acyltiofusidinsyraderivat Download PDFInfo
- Publication number
- FI58136C FI58136C FI772066A FI772066A FI58136C FI 58136 C FI58136 C FI 58136C FI 772066 A FI772066 A FI 772066A FI 772066 A FI772066 A FI 772066A FI 58136 C FI58136 C FI 58136C
- Authority
- FI
- Finland
- Prior art keywords
- compound
- deacetoxy
- acid
- formula
- ether
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
- C07J41/0027—Azides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J13/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17
- C07J13/007—Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17 with double bond in position 17 (20)
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
- C07J31/003—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring the S atom directly linked to a ring carbon atom of the cyclopenta(a)hydrophenanthrene skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
- C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J33/00—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C07J33/002—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J51/00—Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Communicable Diseases (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB2792176 | 1976-07-05 | ||
GB27921/76A GB1581335A (en) | 1976-07-05 | 1976-07-05 | 16-s-acyl derivatives of fusidic acid |
Publications (3)
Publication Number | Publication Date |
---|---|
FI772066A FI772066A (de) | 1978-01-06 |
FI58136B FI58136B (fi) | 1980-08-29 |
FI58136C true FI58136C (fi) | 1980-12-10 |
Family
ID=10267438
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI772066A FI58136C (fi) | 1976-07-05 | 1977-07-01 | Foerfarande foer framstaellning av terapeutiskt anvaendbara 16-deacetoxi-16alfa-acyltiofusidinsyraderivat |
Country Status (22)
Country | Link |
---|---|
US (1) | US4119717A (de) |
JP (1) | JPS535152A (de) |
AT (1) | AT354625B (de) |
AU (1) | AU516152B2 (de) |
BE (1) | BE856464A (de) |
CA (1) | CA1100941A (de) |
DE (1) | DE2730196C2 (de) |
DK (1) | DK148390B (de) |
FI (1) | FI58136C (de) |
FR (1) | FR2357574A1 (de) |
GB (1) | GB1581335A (de) |
GR (1) | GR63210B (de) |
IE (1) | IE45217B1 (de) |
IT (1) | IT1083082B (de) |
LU (1) | LU77683A1 (de) |
NL (1) | NL7707221A (de) |
NZ (1) | NZ184408A (de) |
PH (1) | PH14058A (de) |
PT (1) | PT66759B (de) |
SE (1) | SE436752B (de) |
YU (1) | YU165477A (de) |
ZA (1) | ZA773739B (de) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4162259A (en) * | 1975-12-03 | 1979-07-24 | Leo Pharmaceutical Products Ltd. A/S (Lovens Kemiske fabrik Produktionsaktienselskab) | Fusidic acid derivatives |
US4746508A (en) * | 1983-06-06 | 1988-05-24 | Beth Israel Hospital Assn. | Drug administration |
US4959358A (en) * | 1983-06-06 | 1990-09-25 | Beth Israel Hospital Assn. | Drug administration |
US4548922A (en) * | 1983-06-06 | 1985-10-22 | Beth Israel Hospital | Drug administration |
US4994439A (en) * | 1989-01-19 | 1991-02-19 | California Biotechnology Inc. | Transmembrane formulations for drug administration |
GB9518883D0 (en) * | 1995-09-15 | 1995-11-15 | Leo Pharm Prod Ltd | Chemical compounds |
MY140194A (en) * | 2003-07-16 | 2009-11-30 | Leo Pharma As | Novel fusidic acid derivatives |
ES2424395T3 (es) * | 2006-09-19 | 2013-10-01 | Abbott Products Gmbh | Derivados de estratrieno y sus usos como inhibidores de la 17-beta-hidroxiesteroide-deshidrogenasa |
PT106679B (pt) | 2012-11-27 | 2015-03-25 | Hovione Farmaciencia Sa | Formulações tópicas de tetraciclinas, sua preparação e usos |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1490852A (en) * | 1974-09-12 | 1977-11-02 | Leo Pharm Prod Ltd | Fusidic acid derivatives |
GR60362B (en) * | 1975-06-25 | 1978-05-19 | Leo Pharm Prod Ltd | Preparation process of new 16-ethers of fusidic acid derivatives |
US4060606A (en) * | 1975-06-25 | 1977-11-29 | Leo Pharmaceutical Products Ltd. A/S | 16-Ethers of fusidic acid derivatives |
-
1976
- 1976-07-05 GB GB27921/76A patent/GB1581335A/en not_active Expired
-
1977
- 1977-06-14 US US05/806,376 patent/US4119717A/en not_active Expired - Lifetime
- 1977-06-14 IE IE1209/77A patent/IE45217B1/en unknown
- 1977-06-16 NZ NZ184408A patent/NZ184408A/xx unknown
- 1977-06-22 ZA ZA00773739A patent/ZA773739B/xx unknown
- 1977-06-24 AU AU26438/77A patent/AU516152B2/en not_active Expired
- 1977-06-28 AT AT455777A patent/AT354625B/de not_active IP Right Cessation
- 1977-06-29 NL NL7707221A patent/NL7707221A/xx not_active Application Discontinuation
- 1977-07-01 DK DK294177AA patent/DK148390B/da unknown
- 1977-07-01 FI FI772066A patent/FI58136C/fi not_active IP Right Cessation
- 1977-07-04 CA CA281,930A patent/CA1100941A/en not_active Expired
- 1977-07-04 JP JP7976377A patent/JPS535152A/ja active Granted
- 1977-07-04 IT IT68550/77A patent/IT1083082B/it active
- 1977-07-04 LU LU77683A patent/LU77683A1/xx unknown
- 1977-07-04 GR GR53871A patent/GR63210B/el unknown
- 1977-07-04 FR FR7720523A patent/FR2357574A1/fr active Granted
- 1977-07-04 PT PT66759A patent/PT66759B/pt unknown
- 1977-07-04 SE SE7707749A patent/SE436752B/xx unknown
- 1977-07-04 DE DE2730196A patent/DE2730196C2/de not_active Expired
- 1977-07-04 BE BE179074A patent/BE856464A/xx not_active IP Right Cessation
- 1977-07-05 PH PH19958A patent/PH14058A/en unknown
- 1977-07-05 YU YU01654/77A patent/YU165477A/xx unknown
Also Published As
Publication number | Publication date |
---|---|
AU2643877A (en) | 1979-01-04 |
PH14058A (en) | 1980-12-29 |
US4119717A (en) | 1978-10-10 |
AT354625B (de) | 1979-01-25 |
BE856464A (fr) | 1978-01-04 |
AU516152B2 (en) | 1981-05-21 |
SE7707749L (sv) | 1978-01-06 |
SE436752B (sv) | 1985-01-21 |
DE2730196A1 (de) | 1978-01-19 |
FR2357574A1 (fr) | 1978-02-03 |
FI58136B (fi) | 1980-08-29 |
JPS535152A (en) | 1978-01-18 |
ZA773739B (en) | 1978-05-30 |
IE45217B1 (en) | 1982-07-14 |
LU77683A1 (de) | 1978-01-31 |
NZ184408A (en) | 1980-04-28 |
PT66759B (en) | 1978-12-14 |
GB1581335A (en) | 1980-12-10 |
DK148390B (da) | 1985-06-24 |
ATA455777A (de) | 1979-06-15 |
DK294177A (da) | 1978-01-06 |
DE2730196C2 (de) | 1987-03-05 |
CA1100941A (en) | 1981-05-12 |
IE45217L (en) | 1978-01-05 |
JPS6238360B2 (de) | 1987-08-17 |
PT66759A (en) | 1977-08-01 |
GR63210B (en) | 1979-10-08 |
YU165477A (en) | 1982-06-30 |
FR2357574B1 (de) | 1979-07-20 |
IT1083082B (it) | 1985-05-21 |
FI772066A (de) | 1978-01-06 |
NL7707221A (nl) | 1978-01-09 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM | Patent lapsed |
Owner name: LEO PHARMACEUTICAL PRODUCTS LTD A/S (LOEVENS KEMIS |