FI56013B - Foerfarande foer framstaellning av nya farmakologiskt aktiva triazolo(4 3-b)pyridaziner - Google Patents

Foerfarande foer framstaellning av nya farmakologiskt aktiva triazolo(4 3-b)pyridaziner

Info

Publication number
FI56013B
FI56013B FI2656/74A FI265674A FI56013B FI 56013 B FI56013 B FI 56013B FI 2656/74 A FI2656/74 A FI 2656/74A FI 265674 A FI265674 A FI 265674A FI 56013 B FI56013 B FI 56013B
Authority
FI
Finland
Prior art keywords
pyridaziner
pharmaceutical form
pharmacological active
triazolo
active triazolo
Prior art date
Application number
FI2656/74A
Other languages
English (en)
Other versions
FI56013C (fi
FI265674A (fi
Inventor
Elvio Bellasio
Ambrogio Campi
Original Assignee
Lepetit Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lepetit Spa filed Critical Lepetit Spa
Publication of FI265674A publication Critical patent/FI265674A/fi
Application granted granted Critical
Publication of FI56013B publication Critical patent/FI56013B/fi
Publication of FI56013C publication Critical patent/FI56013C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pulmonology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FI2656/74A 1973-09-21 1974-09-11 Foerfarande foer framstaellning av nya farmakologiskt aktiva triazolo(4,3-b)-pyridatsiner FI56013C (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US399661A US3915968A (en) 1973-09-21 1973-09-21 Triazolopyridazines

Publications (3)

Publication Number Publication Date
FI265674A FI265674A (fi) 1975-03-22
FI56013B true FI56013B (fi) 1979-07-31
FI56013C FI56013C (fi) 1979-11-12

Family

ID=23580450

Family Applications (1)

Application Number Title Priority Date Filing Date
FI2656/74A FI56013C (fi) 1973-09-21 1974-09-11 Foerfarande foer framstaellning av nya farmakologiskt aktiva triazolo(4,3-b)-pyridatsiner

Country Status (25)

Country Link
US (1) US3915968A (fi)
JP (1) JPS537439B2 (fi)
AR (2) AR206514A1 (fi)
AT (1) AT336604B (fi)
BE (1) BE820163A (fi)
CA (1) CA1034948A (fi)
CH (2) CH599212A5 (fi)
DD (1) DD113543A5 (fi)
DE (1) DE2444322C3 (fi)
DK (1) DK138692B (fi)
ES (2) ES430277A1 (fi)
FI (1) FI56013C (fi)
FR (1) FR2244519B1 (fi)
GB (1) GB1480621A (fi)
HU (1) HU171789B (fi)
IE (1) IE40651B1 (fi)
IL (1) IL45654A (fi)
LU (1) LU70949A1 (fi)
NL (1) NL7411849A (fi)
NO (1) NO141717C (fi)
PL (1) PL91748B1 (fi)
RO (1) RO64487A (fi)
SE (1) SE419990B (fi)
SU (2) SU576940A3 (fi)
ZA (1) ZA745482B (fi)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3994898A (en) * 1975-10-16 1976-11-30 E. R. Squibb & Sons, Inc. 1,2,4-Triazolo (4,3-b) pyridazin-3-ones
GR70309B (fi) * 1979-10-29 1982-09-08 Dow Chemical Co
US4526890A (en) * 1979-10-29 1985-07-02 The Dow Chemical Company 3,6,7,8-Substituted-s-triazolo[4,3-b]pyridazines as bronchodilators
US4260756A (en) * 1979-11-15 1981-04-07 American Cyanamid Company 6- And 8-heteroaryl-1,2,4-triazolo[4,3-b]pyridazines
US4293554A (en) * 1980-02-21 1981-10-06 American Cyanamid Company Method of treating asthma
US4487930A (en) * 1982-09-07 1984-12-11 The Dow Chemical Company 6-[(Cyclic amino)alkylamino]-tetrahydrotriazolo[3,4-a]phthalazines
DE3311753A1 (de) * 1983-03-31 1984-10-04 Hoechst Ag, 6230 Frankfurt Substituierte 6-aryl-1,2,4-triazolo(4,3-b)pyridazine - ihre herstellung und verwendung -
US4578464A (en) * 1983-11-22 1986-03-25 Merrell Dow Pharmaceuticals Inc. 6-Hydroxyalkylamino-8-methyl-1,2,4-triazolo-[4,3-b]pyridazine and related compounds
ZA873934B (en) * 1986-06-05 1987-12-02 Merrell Dow Pharmaceuticals Inc. 2,3-dihydro-1-(8-methyl-1,2,4-triazolo(4,3-b)pyridazin-6-yl)-4(1h)-pyridinone
US5011835A (en) * 1990-02-07 1991-04-30 Merrell Dow Pharmaceuticals Inc. Substituted triazolopyridazines, pharmaceutical compositions and use
FR2668151A1 (fr) * 1990-10-23 1992-04-24 Rhone Poulenc Agrochimie Composes a groupe triazolopyridazine leurs preparations et compositions herbicides les contenant.
LT3200B (en) 1992-03-18 1995-03-27 Takeda Chemical Industries Ltd Triazolopyridazine methodfor production thereof and use
ATE168376T1 (de) * 1993-04-12 1998-08-15 Takeda Chemical Industries Ltd Triazolopyridazin-derivate, ihre herstellung und verwendung
KR20040087335A (ko) 2002-03-01 2004-10-13 야마노우치세이야쿠 가부시키가이샤 질소 함유 복소환 화합물
CA2498237A1 (en) * 2002-09-13 2004-03-25 Merck & Co., Inc. Fused heterobicyclo substituted phenyl metabotropic glutamate-5 modulators
US9422290B2 (en) 2012-11-13 2016-08-23 Boehringer Ingelheim International Gmbh Triazolopyridazine
US9266891B2 (en) 2012-11-16 2016-02-23 Boehringer Ingelheim International Gmbh Substituted [1,2,4]triazolo[4,3-A]pyrazines that are BRD4 inhibitors
GB201321745D0 (en) * 2013-12-09 2014-01-22 Ucb Pharma Sa Therapeutic agents
CN112142744A (zh) * 2019-06-28 2020-12-29 上海瑛派药业有限公司 取代的稠合杂芳双环化合物作为激酶抑制剂及其应用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1248409A (fr) * 1957-06-13 1960-12-16 Bellon Labor Sa Roger Perfectionnements aux procédés de préparation de dérivés de la triazolo [4-3,b]pyridazine
DE2161586A1 (de) * 1971-12-11 1973-06-14 Boehringer Mannheim Gmbh Nitrofuryl-triazolo eckige klammer auf 4,3-b eckige klammer zu pyridazin-derivate

Also Published As

Publication number Publication date
FI56013C (fi) 1979-11-12
CH599212A5 (fi) 1978-05-12
CH595382A5 (fi) 1978-02-15
SE7411888L (fi) 1975-03-24
DK138692C (fi) 1979-03-19
CA1034948A (en) 1978-07-18
IL45654A (en) 1977-07-31
NL7411849A (nl) 1975-03-25
BE820163A (fr) 1975-01-16
AR206643A1 (es) 1976-08-06
ES430277A1 (es) 1976-12-16
ES432243A1 (es) 1977-04-16
JPS5058092A (fi) 1975-05-20
PL91748B1 (fi) 1977-03-31
FI265674A (fi) 1975-03-22
IE40651B1 (en) 1979-07-18
GB1480621A (en) 1977-07-20
ATA755074A (de) 1976-09-15
SE419990B (sv) 1981-09-07
FR2244519A1 (fi) 1975-04-18
DK138692B (da) 1978-10-16
RO64487A (fr) 1979-06-15
DE2444322C3 (de) 1981-03-19
FR2244519B1 (fi) 1978-07-21
US3915968A (en) 1975-10-28
SU576940A3 (ru) 1977-10-15
AR206514A1 (es) 1976-07-30
DE2444322B2 (de) 1980-08-07
JPS537439B2 (fi) 1978-03-17
DK496374A (fi) 1975-05-20
NO141717B (no) 1980-01-21
NO743140L (fi) 1975-04-14
AT336604B (de) 1977-05-10
ZA745482B (en) 1975-09-24
NO141717C (no) 1980-04-30
SU545261A3 (ru) 1977-01-30
IE40651L (en) 1975-03-21
DD113543A5 (fi) 1975-06-12
DE2444322A1 (de) 1975-03-27
AU7305374A (en) 1976-03-11
LU70949A1 (fi) 1975-03-06
IL45654A0 (en) 1974-11-29
HU171789B (hu) 1978-03-28

Similar Documents

Publication Publication Date Title
FI56013B (fi) Foerfarande foer framstaellning av nya farmakologiskt aktiva triazolo(4 3-b)pyridaziner
NO141163C (no) Analogifremgangsmaate for fremstilling av farmakologisk aktive pyrimidiner
SE423720B (sv) Framstellning av nya peptidantibiotika
SE386445B (sv) Forfaranden for framstellning av nya bensotiadiazoler
NO145056C (no) (s)-1-aryloksy-2-propanolderivater for fremstilling av terapeutisk aktive (s)-1-aryloksy-3-amino-2-propanolderivater
SE418184B (sv) Forfarande for framstellning av nya penicillin- och cefalosporinforeningar
SE382060B (sv) Forfarande for framstellning av nya substituerade piperidinoalkanonoximderivat
SE424994B (sv) Forfarande for framstellning av nya pseudotrisackarider
SE416731B (sv) Forfarande for framstellning av nya penicilliner
NO137782C (no) Analogifremgangsmaate for fremstilling av nye farmakologisk aktive amino-fenyl-etanolaminer
SE7700442L (sv) Forfarande for framstellning av 6-aminopenicillansyra
SE385698B (sv) Forfarande for framstellning av kinolinettiksyraderivat
SE405477B (sv) Forfarande for framstellning av tetrazolyl-kinaldinsyraderivat med farmakologisk verkan
NO740327L (no) Analogifremgangsmåte for fremstilling av farmakologisk aktive imidazopyridiner.
FI55843B (fi) Foerfarande foer framstaellning av nya terapeutiskt anvaendbara 9 10-dihydro-9- eller -10-hydroxi-imino-4-(1-alkyl-4-piperidyliden-4h-benso(4 5)cyklohepta(1 2-b)tiofenderivat och deras syraadditionssalter
SE418085B (sv) Forfarande for framstellning av nya sulfamoylbensoesyraamider
NO741744L (no) Analogifremgangsmåte for fremstilling av nye terapeutisk aktive derivater av naftyridin.
SE399708B (sv) Forfarande for framstellning av tioxanton-2-karboxylsyraderivat
NO142712C (no) Analogifremgangsmaater for fremstilling av farmakologisk virksomme 9-desoksy-prosta-5,9,(10),13-tripelargonsyrederivater
SE404801B (sv) Forfaranden for framstellning av nya tiazolderivat
NO143499C (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive indanderivater
FI54309B (fi) Foerfarande foer framstaellning av nya farmakologiskt aktiva 8-substituerade 10-piperazino-10,11-dihydrodibenso(b,f) tiepiner
SE434402B (sv) Forfarande for framstellning av nya cefalosporinderivat
SE393801B (sv) Forfarande for framstellning av tiokarbaminsyraderivat med antifungistatisk lekemedelsverken
NO144344C (no) Fremgangsmaate for fremstilling av terapeutisk aktive n-arylsulfonyl n`-(3-azabicykloalkyl)urinstoffer