FI53704C - Foerfarande foer framstaellning av nya histaminolytiskt verkande i 2-staellning basiskt substituerade bentsylftalazonderivater och deras salter - Google Patents

Foerfarande foer framstaellning av nya histaminolytiskt verkande i 2-staellning basiskt substituerade bentsylftalazonderivater och deras salter

Info

Publication number
FI53704C
FI53704C FI160/72A FI16072A FI53704C FI 53704 C FI53704 C FI 53704C FI 160/72 A FI160/72 A FI 160/72A FI 16072 A FI16072 A FI 16072A FI 53704 C FI53704 C FI 53704C
Authority
FI
Finland
Prior art keywords
framework
bentylftalazonderivater
histaminolytic
substitutes
windows
Prior art date
Application number
FI160/72A
Other languages
English (en)
Other versions
FI53704B (fi
Inventor
Dietrich Vogelsang
Gerhard Scheffler
Norbert Brock
Dieter Lenke
Original Assignee
Asta Werke Ag Chem Fab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Asta Werke Ag Chem Fab filed Critical Asta Werke Ag Chem Fab
Publication of FI53704B publication Critical patent/FI53704B/fi
Application granted granted Critical
Publication of FI53704C publication Critical patent/FI53704C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D451/00Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
FI160/72A 1971-01-22 1972-01-21 Foerfarande foer framstaellning av nya histaminolytiskt verkande i 2-staellning basiskt substituerade bentsylftalazonderivater och deras salter FI53704C (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH101271A CH572914A5 (fi) 1971-01-22 1971-01-22

Publications (2)

Publication Number Publication Date
FI53704B FI53704B (fi) 1978-03-31
FI53704C true FI53704C (fi) 1978-07-10

Family

ID=4200381

Family Applications (1)

Application Number Title Priority Date Filing Date
FI160/72A FI53704C (fi) 1971-01-22 1972-01-21 Foerfarande foer framstaellning av nya histaminolytiskt verkande i 2-staellning basiskt substituerade bentsylftalazonderivater och deras salter

Country Status (21)

Country Link
AR (1) AR197293A1 (fi)
AT (1) AT313288B (fi)
AU (1) AU3767472A (fi)
BE (1) BE778269A (fi)
CA (1) CA1010041A (fi)
CH (1) CH572914A5 (fi)
DE (1) DE2164058C3 (fi)
DK (1) DK136981B (fi)
ES (1) ES398949A1 (fi)
FI (1) FI53704C (fi)
FR (1) FR2122517B1 (fi)
GB (1) GB1377231A (fi)
HK (1) HK62577A (fi)
HU (1) HU163979B (fi)
IL (1) IL38496A (fi)
NL (1) NL177116C (fi)
OA (1) OA04087A (fi)
PL (1) PL88930B1 (fi)
SE (1) SE404604B (fi)
YU (1) YU35361B (fi)
ZA (1) ZA718712B (fi)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3575135D1 (de) * 1984-09-14 1990-02-08 Asta Pharma Ag Substituierte benzylphthalazinon-derivate.
PT88984B (pt) * 1987-11-13 1993-01-29 Asta Medica Ag Processo para a preparação de embonato de azelastina e de composições earmacâutxcas que 0 contêm como ingrediente activo
EP0316633B1 (de) * 1987-11-13 1993-01-27 ASTA Medica Aktiengesellschaft Azelastin enthaltende Arzneimittel zur Anwendung in der Nase und/oder am Auge
EP0316639B1 (de) * 1987-11-13 1994-06-08 ASTA Medica Aktiengesellschaft Azelastin-Embonat, Verfahren zu seiner Herstellung und pharmazeutische Zubereitungen, die als Wirkstoff Azelastin-Embonat enthalten
DE3836579A1 (de) * 1987-11-13 1989-05-24 Asta Pharma Ag Azelastin enthaltende arzneimittel zur anwendung in der nase und/oder am auge
DE3912292A1 (de) * 1988-04-20 1989-11-09 Asta Pharma Ag Azelastin enthaltende arzneimittel mit kontrollierter wirkstoffabgabe
US5110814A (en) * 1989-01-11 1992-05-05 Asta Pharma Ag Azelastine and its salts used to combat psoriasis
EP0396069B1 (de) * 1989-05-05 1994-06-22 ASTA Medica Aktiengesellschaft Salze des Azelastins mit verbesserter Löslichkeit
DE4207234A1 (de) * 1992-03-07 1993-09-09 Asta Medica Ag Neue aminocarbonsaeure-derivate mit antiallergischer/antiasthmatischer wirkung und verfahren zu deren herstellung
DE4345224C2 (de) * 1993-12-18 1999-07-01 Asta Medica Ag Verfahren zur Herstellung von Säureadditionssalzen des Azelastins und Flezelastins
DE4343409C2 (de) * 1993-12-18 1997-03-20 Asta Medica Ag Verbessertes Verfahren zur Herstellung von Hexahydroazepinonen und Hexahydroazepinolen
GB2389530B (en) 2002-06-14 2007-01-10 Cipla Ltd Pharmaceutical compositions
US20070020330A1 (en) 2004-11-24 2007-01-25 Medpointe Healthcare Inc. Compositions comprising azelastine and methods of use thereof
DK2377557T3 (en) 2004-11-24 2017-02-06 Meda Pharmaceuticals Inc Compositions comprising azelastine and methods for its use
US8758816B2 (en) 2004-11-24 2014-06-24 Meda Pharmaceuticals Inc. Compositions comprising azelastine and methods of use thereof
BRPI0710156A2 (pt) * 2006-04-20 2012-06-05 Glaxo Group Ltd composto ou um sal do mesno, composição, combinação, e, uso de um composto.

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1046625B (de) * 1957-08-15 1958-12-18 Hydrierwerk Rodleben Veb Verfahren zur Herstellung basisch substituierter Phthalazone
GB1100911A (en) * 1963-08-20 1968-01-24 Benger Lab Ltd Phthalazine derivatives
FR1512879A (fr) * 1966-10-28 1968-02-09 Hydrierwerk Rodleben Veb Procédé pour la fabrication de phtalazones avec substituants basiques

Also Published As

Publication number Publication date
GB1377231A (en) 1974-12-11
AT313288B (de) 1974-02-11
ES398949A1 (es) 1975-06-01
CH572914A5 (fi) 1976-02-27
NL7200400A (fi) 1972-07-25
AR197293A1 (es) 1974-03-29
NL177116B (nl) 1985-03-01
SE404604B (sv) 1978-10-16
DE2164058A1 (de) 1972-07-27
DK136981C (fi) 1978-06-05
ZA718712B (en) 1972-09-27
FR2122517B1 (fi) 1975-08-01
YU11272A (en) 1980-06-30
IL38496A0 (en) 1972-03-28
FR2122517A1 (fi) 1972-09-01
BE778269A (fr) 1972-07-19
DE2164058B2 (de) 1980-10-23
FI53704B (fi) 1978-03-31
OA04087A (fr) 1979-10-30
IL38496A (en) 1975-05-22
PL88930B1 (fi) 1976-10-30
HU163979B (fi) 1973-12-28
NL177116C (nl) 1985-08-01
DE2164058C3 (de) 1981-08-13
DK136981B (da) 1977-12-27
SU440838A3 (fi) 1974-08-25
YU35361B (en) 1980-12-31
AU3767472A (en) 1973-07-12
CA1010041A (en) 1977-05-10
HK62577A (en) 1977-12-30

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