FI112227B - Menetelmä farmakologisesti aktiivisten pyridiinijohdannaisten valmistamiseksi - Google Patents

Menetelmä farmakologisesti aktiivisten pyridiinijohdannaisten valmistamiseksi Download PDF

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Publication number
FI112227B
FI112227B FI952607A FI952607A FI112227B FI 112227 B FI112227 B FI 112227B FI 952607 A FI952607 A FI 952607A FI 952607 A FI952607 A FI 952607A FI 112227 B FI112227 B FI 112227B
Authority
FI
Finland
Prior art keywords
pyridyl
formula
pyrimidinamine
compound
amino
Prior art date
Application number
FI952607A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI952607A0 (fi
FI952607A (fi
Inventor
Juerg Zimmermann
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of FI952607A0 publication Critical patent/FI952607A0/fi
Publication of FI952607A publication Critical patent/FI952607A/fi
Application granted granted Critical
Publication of FI112227B publication Critical patent/FI112227B/fi

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/28—Compounds containing heavy metals
    • A61K31/305—Mercury compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/04—Immunostimulants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Dermatology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Vascular Medicine (AREA)
  • Rheumatology (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Medicinal Preparation (AREA)
FI952607A 1993-10-01 1995-05-29 Menetelmä farmakologisesti aktiivisten pyridiinijohdannaisten valmistamiseksi FI112227B (fi)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
CH296993 1993-10-01
CH296993 1993-10-01
CH228194 1994-07-18
CH228194 1994-07-18
EP9403151 1994-09-21
PCT/EP1994/003151 WO1995009853A1 (fr) 1993-10-01 1994-09-21 Derives pyridine pharmacologiquement actifs ainsi que leurs procedes de preparation

Publications (3)

Publication Number Publication Date
FI952607A0 FI952607A0 (fi) 1995-05-29
FI952607A FI952607A (fi) 1995-05-29
FI112227B true FI112227B (fi) 2003-11-14

Family

ID=25690002

Family Applications (1)

Application Number Title Priority Date Filing Date
FI952607A FI112227B (fi) 1993-10-01 1995-05-29 Menetelmä farmakologisesti aktiivisten pyridiinijohdannaisten valmistamiseksi

Country Status (21)

Country Link
US (1) US5728708A (fr)
EP (1) EP0672041B1 (fr)
JP (1) JP2983636B2 (fr)
KR (1) KR100330553B1 (fr)
CN (1) CN1047776C (fr)
AT (1) ATE208772T1 (fr)
AU (1) AU691834B2 (fr)
CA (1) CA2148928C (fr)
CZ (1) CZ290681B6 (fr)
DE (1) DE69429078T2 (fr)
DK (1) DK0672041T3 (fr)
ES (1) ES2167377T3 (fr)
FI (1) FI112227B (fr)
HU (1) HU228172B1 (fr)
IL (1) IL111077A (fr)
NO (1) NO308794B1 (fr)
NZ (1) NZ273617A (fr)
PL (1) PL179417B1 (fr)
PT (1) PT672041E (fr)
RU (1) RU2135491C1 (fr)
WO (1) WO1995009853A1 (fr)

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Also Published As

Publication number Publication date
AU691834B2 (en) 1998-05-28
HU228172B1 (en) 2013-01-28
HU9501953D0 (en) 1995-09-28
DE69429078D1 (de) 2001-12-20
HUT72609A (en) 1996-05-28
RU2135491C1 (ru) 1999-08-27
ES2167377T3 (es) 2002-05-16
PL309225A1 (en) 1995-10-02
PL179417B1 (en) 2000-09-29
CA2148928C (fr) 2005-10-18
JPH08504215A (ja) 1996-05-07
PT672041E (pt) 2002-04-29
NO952132L (no) 1995-05-30
FI952607A0 (fi) 1995-05-29
AU7697794A (en) 1995-05-01
CN1047776C (zh) 1999-12-29
IL111077A0 (en) 1994-11-28
US5728708A (en) 1998-03-17
CA2148928A1 (fr) 1995-04-13
EP0672041B1 (fr) 2001-11-14
IL111077A (en) 1999-10-28
KR950704296A (ko) 1995-11-17
DK0672041T3 (da) 2002-02-25
DE69429078T2 (de) 2002-07-11
ATE208772T1 (de) 2001-11-15
JP2983636B2 (ja) 1999-11-29
CN1115982A (zh) 1996-01-31
CZ290681B6 (cs) 2002-09-11
NO952132D0 (no) 1995-05-30
WO1995009853A1 (fr) 1995-04-13
CZ172295A3 (en) 1996-03-13
KR100330553B1 (ko) 2002-11-27
EP0672041A1 (fr) 1995-09-20
NO308794B1 (no) 2000-10-30
FI952607A (fi) 1995-05-29
NZ273617A (en) 1996-11-26

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