FI104950B - Menetelmä glipitsidiä sisältävän annosmuodon valmistamiseksi - Google Patents

Menetelmä glipitsidiä sisältävän annosmuodon valmistamiseksi Download PDF

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Publication number
FI104950B
FI104950B FI920956A FI920956A FI104950B FI 104950 B FI104950 B FI 104950B FI 920956 A FI920956 A FI 920956A FI 920956 A FI920956 A FI 920956A FI 104950 B FI104950 B FI 104950B
Authority
FI
Finland
Prior art keywords
glipizide
dosage form
compound
wall
molecular weight
Prior art date
Application number
FI920956A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI920956A0 (fi
Inventor
Patrick S-L Wong
Atul Devdatt Ayer
Anthony L Kuczynski
Original Assignee
Alza Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Alza Corp filed Critical Alza Corp
Publication of FI920956A0 publication Critical patent/FI920956A0/fi
Application granted granted Critical
Publication of FI104950B publication Critical patent/FI104950B/fi

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/64Sulfonylureas, e.g. glibenclamide, tolbutamide, chlorpropamide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0002Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0004Osmotic delivery systems; Sustained release driven by osmosis, thermal energy or gas
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2031Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Investigating Or Analysing Biological Materials (AREA)
  • Ultra Sonic Daignosis Equipment (AREA)
  • Lubrication Of Internal Combustion Engines (AREA)
FI920956A 1989-09-05 1992-03-04 Menetelmä glipitsidiä sisältävän annosmuodon valmistamiseksi FI104950B (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US07/402,314 US5024843A (en) 1989-09-05 1989-09-05 Oral hypoglycemic glipizide granulation
US40231489 1989-09-05
PCT/US1990/004981 WO1991003247A1 (en) 1989-09-05 1990-08-31 Dosage form for administering oral hypoglycemic glipizide
US9004981 1990-08-31

Publications (2)

Publication Number Publication Date
FI920956A0 FI920956A0 (fi) 1992-03-04
FI104950B true FI104950B (fi) 2000-05-15

Family

ID=23591411

Family Applications (1)

Application Number Title Priority Date Filing Date
FI920956A FI104950B (fi) 1989-09-05 1992-03-04 Menetelmä glipitsidiä sisältävän annosmuodon valmistamiseksi

Country Status (20)

Country Link
US (2) US5024843A (pt)
EP (1) EP0490991B1 (pt)
JP (1) JP2919964B2 (pt)
KR (1) KR0157640B1 (pt)
AT (1) ATE94393T1 (pt)
AU (1) AU632859B2 (pt)
CA (1) CA2024502C (pt)
DE (1) DE69003392T2 (pt)
DK (1) DK0490991T3 (pt)
ES (1) ES2060199T3 (pt)
FI (1) FI104950B (pt)
GR (1) GR1000932B (pt)
HK (1) HK116897A (pt)
IE (1) IE62594B1 (pt)
MX (1) MX171191B (pt)
NO (1) NO303963B1 (pt)
NZ (1) NZ235127A (pt)
PT (1) PT95169B (pt)
WO (1) WO1991003247A1 (pt)
ZA (1) ZA906972B (pt)

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US5208037A (en) * 1991-04-22 1993-05-04 Alza Corporation Dosage forms comprising polymers comprising different molecular weights
US6726930B1 (en) * 1993-09-09 2004-04-27 Penwest Pharmaceuticals Co. Sustained release heterodisperse hydrogel systems for insoluble drugs
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ES2322405T3 (es) * 1996-07-08 2009-06-19 Penwest Pharmaceuticals Co. Matriz de liberacion controlada para farmacos insolubles en dosis elevadas.
ES2255103T3 (es) * 1996-10-25 2006-06-16 Shire Laboratories Inc. Sistema osmotico de administracion de dosis en forma soluble.
US6361796B1 (en) 1996-10-25 2002-03-26 Shire Laboratories, Inc. Soluble form osmotic dose delivery system
US6919373B1 (en) 1996-11-12 2005-07-19 Alza Corporation Methods and devices for providing prolonged drug therapy
DE69735848T2 (de) * 1996-11-25 2006-12-28 Alza Corp., Palo Alto Dosisform mit ansteigender dosisfreisetzung
ZA979605B (en) * 1996-11-25 1998-05-21 Alza Corp Ascending-dose dosage form.
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US6056977A (en) 1997-10-15 2000-05-02 Edward Mendell Co., Inc. Once-a-day controlled release sulfonylurea formulation
US8524277B2 (en) 1998-03-06 2013-09-03 Alza Corporation Extended release dosage form
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US6703045B2 (en) 2001-08-21 2004-03-09 Council Of Scientific & Industrial Research Composition and method for maintaining blood glucose level
CA2461693A1 (en) * 2001-09-28 2003-04-03 Sun Pharmaceutical Industries Limited Dosage form for treatment of diabetes mellitus
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US20050232995A1 (en) 2002-07-29 2005-10-20 Yam Nyomi V Methods and dosage forms for controlled delivery of paliperidone and risperidone
US20040052844A1 (en) * 2002-09-16 2004-03-18 Fang-Hsiung Hsiao Time-controlled, sustained release, pharmaceutical composition containing water-soluble resins
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US7611728B2 (en) * 2003-09-05 2009-11-03 Supernus Pharmaceuticals, Inc. Osmotic delivery of therapeutic compounds by solubility enhancement
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CN100571783C (zh) * 2006-10-30 2009-12-23 北京红林制药有限公司 格列吡嗪控释片及其制备方法
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CA2765876A1 (en) * 2009-06-19 2010-12-23 Knopp Neurosciences, Inc. Compositions and methods for treating amyotrophic lateral sclerosis
CN101940578B (zh) * 2010-08-25 2012-07-25 山东新华制药股份有限公司 一种用于治疗2型糖尿病的药物组合物及其制备方法
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Also Published As

Publication number Publication date
DE69003392D1 (de) 1993-10-21
PT95169B (pt) 1998-06-30
HK116897A (en) 1997-09-05
AU6417590A (en) 1991-04-08
KR920703066A (ko) 1992-12-17
EP0490991A1 (en) 1992-06-24
GR900100659A (en) 1992-01-20
DK0490991T3 (da) 1993-11-29
EP0490991B1 (en) 1993-09-15
NO920740D0 (no) 1992-02-25
CA2024502A1 (en) 1991-03-06
GR1000932B (el) 1993-03-16
DE69003392T2 (de) 1994-01-13
US5545413A (en) 1996-08-13
MX171191B (es) 1993-10-06
WO1991003247A1 (en) 1991-03-21
ATE94393T1 (de) 1993-10-15
IE903166A1 (en) 1991-03-13
NO303963B1 (no) 1998-10-05
JPH05500222A (ja) 1993-01-21
NZ235127A (en) 1993-02-25
ZA906972B (en) 1991-06-26
CA2024502C (en) 1991-03-06
US5024843A (en) 1991-06-18
IE62594B1 (en) 1995-02-08
KR0157640B1 (ko) 1998-11-16
PT95169A (pt) 1991-05-22
JP2919964B2 (ja) 1999-07-19
FI920956A0 (fi) 1992-03-04
ES2060199T3 (es) 1994-11-16
NO920740L (no) 1992-02-25
AU632859B2 (en) 1993-01-14

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