ES557723A0 - Procedimiento para la produccion de tiazoles - Google Patents
Procedimiento para la produccion de tiazolesInfo
- Publication number
- ES557723A0 ES557723A0 ES557723A ES557723A ES557723A0 ES 557723 A0 ES557723 A0 ES 557723A0 ES 557723 A ES557723 A ES 557723A ES 557723 A ES557723 A ES 557723A ES 557723 A0 ES557723 A0 ES 557723A0
- Authority
- ES
- Spain
- Prior art keywords
- tiazoles
- procedure
- production
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/42—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE3522351 | 1985-06-22 | ||
DE3522353 | 1985-06-22 | ||
DE3522354 | 1985-06-22 | ||
DE3605868 | 1986-02-24 |
Publications (2)
Publication Number | Publication Date |
---|---|
ES8802045A1 ES8802045A1 (es) | 1988-03-16 |
ES557723A0 true ES557723A0 (es) | 1988-03-16 |
Family
ID=27433378
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES556363A Expired ES8802154A1 (es) | 1985-06-22 | 1986-06-20 | Procedimiento para la produccion de tiazoles., |
ES557723A Expired ES8802045A1 (es) | 1985-06-22 | 1987-09-15 | Procedimiento para la produccion de tiazoles |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES556363A Expired ES8802154A1 (es) | 1985-06-22 | 1986-06-20 | Procedimiento para la produccion de tiazoles., |
Country Status (17)
Country | Link |
---|---|
US (2) | US4737500A (es) |
AU (1) | AU5894086A (es) |
BE (1) | BE904945A (es) |
CH (1) | CH668426A5 (es) |
DK (1) | DK292986A (es) |
ES (2) | ES8802154A1 (es) |
FI (1) | FI862644A (es) |
FR (1) | FR2587342A1 (es) |
GB (1) | GB2177395B (es) |
GR (1) | GR861601B (es) |
HU (1) | HUT43600A (es) |
IL (1) | IL79178A0 (es) |
IT (1) | IT1203806B (es) |
LU (1) | LU86487A1 (es) |
NL (1) | NL8601494A (es) |
PH (1) | PH23389A (es) |
SE (1) | SE8602723L (es) |
Families Citing this family (45)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4804663A (en) * | 1985-03-27 | 1989-02-14 | Janssen Pharmaceutica N.V. | 3-piperidinyl-substituted 1,2-benzisoxazoles and 1,2-benzisothiazoles |
HUT43600A (en) * | 1985-06-22 | 1987-11-30 | Sandoz Ag | Process for production of new thiazole derivatives and medical compound containing those |
MX173362B (es) * | 1987-03-02 | 1994-02-23 | Pfizer | Compuestos de piperazinil heterociclicos y procedimiento para su preparacion |
FR2612187B1 (fr) * | 1987-03-12 | 1989-07-21 | Sanofi Sa | Derives du thiazole actifs sur le systeme cholinergique, leur procede de preparation et compositions pharmaceutiques en contenant |
US4804751A (en) * | 1987-06-30 | 1989-02-14 | American Home Products Corporation | Polycyclic hydrocarbon succinimides with psychotropic activity |
ES2053748T3 (es) * | 1987-09-10 | 1994-08-01 | Merck Sharp & Dohme | Oxazoles y tiazoles para el tratamiento de la demencia senil. |
US4883795A (en) * | 1988-01-22 | 1989-11-28 | Pfizer Inc. | Piperazinyl-heterocyclic compounds |
EP0350145A3 (en) * | 1988-04-28 | 1990-07-04 | Yamanouchi Pharmaceutical Co. Ltd. | Pyridylthiazolidine carboxamide derivatives and their intermediates and production of both |
US4935424A (en) * | 1988-05-27 | 1990-06-19 | Warner-Lambert Company | 4 or 5-(substituted piperazinylalkyl)-2-aminothiazoles as antipsychotic agents |
US5015740A (en) * | 1988-08-05 | 1991-05-14 | Janssen Pharmaceutica N.V. | Antipsychotic 3-piperazinylbenzazole derivatives |
US4957916A (en) * | 1988-08-05 | 1990-09-18 | Janssen Pharmaceutica N.V. | Antipsychotic 3-piperazinylbenzazole derivatives |
US5077295A (en) * | 1988-09-16 | 1991-12-31 | Pfizer Inc. | Antipsychoic 4-(4-(3-benzisothiazolyl)-1-piperazinyl)buytl bridged bicycle imides |
US4954503A (en) * | 1989-09-11 | 1990-09-04 | Hoechst-Roussel Pharmaceuticals, Inc. | 3-(1-substituted-4-piperazinyl)-1H-indazoles |
US5194436A (en) * | 1991-01-10 | 1993-03-16 | Hoechst-Roussel Pharmaceuticals Inc. | 1-piperazinyl-2-butenes and -2-butynes |
US5130315A (en) * | 1991-01-10 | 1992-07-14 | Raymond R. Wittekind | 1-piperazinyl-2-butenes and -2-butynes |
IT1251144B (it) * | 1991-07-30 | 1995-05-04 | Boehringer Ingelheim Italia | Derivati del benzimidazolone |
NZ276088A (en) | 1993-11-19 | 1999-07-29 | Janssen Pharmaceutica Nv | [(1,2-benzisoxazol-3-yl)-1-piperidinyl-alkyl-6,7,8,9-tetrahydro-4h- pyrido[1,2-a]-pyrimidin-4-one derivatives (ie risperidone) |
US5889010A (en) * | 1995-05-18 | 1999-03-30 | Pfizer Inc. | Benzimidazole derivatives having dopaminergic activity |
DE19746612A1 (de) | 1997-10-22 | 1999-04-29 | Basf Ag | 2-Substituierte 1,2-Benzisothiazol-Derivate, ihre Herstellung und Verwendung |
US7183410B2 (en) | 2001-08-02 | 2007-02-27 | Bidachem S.P.A. | Stable polymorph of flibanserin |
US20030060475A1 (en) * | 2001-08-10 | 2003-03-27 | Boehringer Ingelheim Pharma Kg | Method of using flibanserin for neuroprotection |
US10675280B2 (en) | 2001-10-20 | 2020-06-09 | Sprout Pharmaceuticals, Inc. | Treating sexual desire disorders with flibanserin |
UA78974C2 (en) | 2001-10-20 | 2007-05-10 | Boehringer Ingelheim Pharma | Use of flibanserin for treating disorders of sexual desire |
MXPA06012059A (es) * | 2004-04-22 | 2007-01-25 | Boehringer Ingelheim Int | Nuevas composiciones farmaceuticas para el tratamiento de los trastornos sexuales ii. |
US20050239798A1 (en) * | 2004-04-22 | 2005-10-27 | Boehringer Ingelheim Pharmaceuticals, Inc. | Method for the treatment of premenstrual and other female sexual disorders |
US20060025420A1 (en) * | 2004-07-30 | 2006-02-02 | Boehringer Ingelheimn International GmbH | Pharmaceutical compositions for the treatment of female sexual disorders |
JP2008511569A (ja) * | 2004-09-03 | 2008-04-17 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 注意欠如活動過多障害の治療方法 |
WO2006096439A2 (en) * | 2005-03-04 | 2006-09-14 | Boehringer Ingelheim International Gmbh | Pharmaceutical compositions for the treatment and/or prevention of schizophrenia and related diseases |
EP1858515A2 (en) * | 2005-03-04 | 2007-11-28 | Boehringer Ingelheim International Gmbh | Pharmaceutical compositions for the treatment and/or prevention of anxiety disorders |
CA2599721A1 (en) * | 2005-03-04 | 2006-09-14 | Boehringer Ingelheim International Gmbh | Pharmaceutical compositions for the treatment and/or prevention of depression |
CA2608249A1 (en) * | 2005-05-06 | 2006-11-16 | Boehringer Ingelheim International Gmbh | Method for the treatment of drug abuse with flibanserin |
CA2608363A1 (en) * | 2005-05-19 | 2006-11-23 | Boehringer Ingelheim International Gmbh | Method for the treatment of drug-induced sexual dysfunction |
JP2009503020A (ja) | 2005-08-03 | 2009-01-29 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 肥満症の治療におけるフリバンセリンの使用 |
US20070123540A1 (en) * | 2005-10-29 | 2007-05-31 | Angelo Ceci | Sexual desire enhancing medicaments comprising benzimidazolone derivatives |
WO2007048803A1 (en) | 2005-10-29 | 2007-05-03 | Boehringer Ingelheim International Gmbh | Benzimidazolone derivatives for the treatment of premenstrual and other female sexual disorders |
US20070105869A1 (en) * | 2005-11-08 | 2007-05-10 | Stephane Pollentier | Use of flibanserin for the treatment of pre-menopausal sexual desire disorders |
WO2007128802A2 (en) * | 2006-05-09 | 2007-11-15 | Boehringer Ingelheim International Gmbh | Use of flibanserin for the treatment of post-menopausal sexual desire disorders |
JP2009541443A (ja) | 2006-06-30 | 2009-11-26 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 尿失禁及び関連疾患の治療のためのフリバンセリン |
CA2657043A1 (en) * | 2006-07-14 | 2008-01-17 | Boehringer Ingelheim International Gmbh | Use of flibanserin for the treatment of sexual disorders in females |
CL2007002214A1 (es) | 2006-08-14 | 2008-03-07 | Boehringer Ingelheim Int | Composicion farmaceutica en la forma de comprimido, donde al menos la longitud del comprimido en el estado anterior de la aplicacion es al menos 7/12 del diametro pilorico del paciente y despues de ingerirlo en estado alimentado, la longitud del comp |
EA200900264A1 (ru) | 2006-08-14 | 2009-08-28 | Бёрингер Ингельхайм Интернациональ Гмбх | Композиции флибансерина и способ их приготовления |
EA200900270A1 (ru) | 2006-08-25 | 2009-08-28 | Бёрингер Ингельхайм Интернациональ Гмбх | Системы регулируемого высвобождения и способ их приготовления |
PT2159226T (pt) * | 2007-03-29 | 2016-12-16 | Joint-Stock Company Obninsk Chemical Pharmaceutical Company | Agente anti-histamínico e antialérgico e um método para a produção do mesmo |
PE20091188A1 (es) | 2007-09-12 | 2009-08-31 | Boehringer Ingelheim Int | Compuesto 1-[2-(4-(3-trifluorometil-fenil)piperazin-1-il)etil]-2,3-dihidro-1h-benzimidazol-2-ona (flibanserina), sus sales de adicion y composiciones farmaceuticas que los contienen |
CA2686480A1 (en) | 2008-12-15 | 2010-06-15 | Boehringer Ingelheim International Gmbh | New salts |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BE637271A (es) * | 1963-04-04 | 1900-01-01 | ||
DE1595923A1 (de) * | 1965-02-20 | 1969-11-27 | Merck Ag E | 1-Aralkyl-4-(thiazolyl-2)-piperazine und Verfahren zu ihrer Herstellung |
BE759371A (fr) * | 1969-11-24 | 1971-05-24 | Bristol Myers Co | Azaspirodecanediones heterocycliques et procedes pour leur preparation |
JPS5246935B1 (es) * | 1971-04-06 | 1977-11-29 | ||
BE787059A (fr) * | 1971-08-03 | 1973-02-01 | Wander Ag Dr A | Nouveaux derives du thiazole, leur preparation et leur application comme medicaments |
CH583232A5 (es) * | 1973-02-02 | 1976-12-31 | Wander Ag Dr A | |
US4182763A (en) * | 1978-05-22 | 1980-01-08 | Mead Johnson & Company | Buspirone anti-anxiety method |
US4423049A (en) * | 1981-12-28 | 1983-12-27 | Mead Johnson & Company | 2-[4-[(4,4-Dialkyl-2,6-piperidinedion-1-yl)butyl]-1-piperazinyl]pyrimidines |
DE3321969A1 (de) * | 1983-06-18 | 1984-12-20 | Troponwerke GmbH & Co KG, 5000 Köln | 2-pyrimidinyl-1-piperazin-derivate, verfahren zu ihrer herstellung und diese enthaltende arzneimittel |
HUT43600A (en) * | 1985-06-22 | 1987-11-30 | Sandoz Ag | Process for production of new thiazole derivatives and medical compound containing those |
-
1986
- 1986-06-09 HU HU862433A patent/HUT43600A/hu unknown
- 1986-06-09 NL NL8601494A patent/NL8601494A/nl not_active Application Discontinuation
- 1986-06-12 CH CH2373/86A patent/CH668426A5/de not_active IP Right Cessation
- 1986-06-18 FR FR8608893A patent/FR2587342A1/fr active Pending
- 1986-06-18 BE BE1/011508A patent/BE904945A/fr not_active IP Right Cessation
- 1986-06-18 SE SE8602723A patent/SE8602723L/xx not_active Application Discontinuation
- 1986-06-19 GB GB8614974A patent/GB2177395B/en not_active Expired
- 1986-06-19 FI FI862644A patent/FI862644A/fi not_active IP Right Cessation
- 1986-06-20 PH PH33910A patent/PH23389A/en unknown
- 1986-06-20 DK DK292986A patent/DK292986A/da not_active Application Discontinuation
- 1986-06-20 IT IT48157/86A patent/IT1203806B/it active
- 1986-06-20 US US06/876,617 patent/US4737500A/en not_active Expired - Fee Related
- 1986-06-20 ES ES556363A patent/ES8802154A1/es not_active Expired
- 1986-06-20 GR GR861601A patent/GR861601B/el unknown
- 1986-06-20 AU AU58940/86A patent/AU5894086A/en not_active Abandoned
- 1986-06-20 LU LU86487A patent/LU86487A1/fr unknown
- 1986-06-20 IL IL79178A patent/IL79178A0/xx unknown
-
1987
- 1987-09-15 ES ES557723A patent/ES8802045A1/es not_active Expired
-
1988
- 1988-02-02 US US07/151,349 patent/US4892879A/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
US4892879A (en) | 1990-01-09 |
ES8802045A1 (es) | 1988-03-16 |
PH23389A (en) | 1989-07-26 |
LU86487A1 (fr) | 1987-01-13 |
FI862644A0 (fi) | 1986-06-19 |
CH668426A5 (de) | 1988-12-30 |
ES8802154A1 (es) | 1988-04-01 |
US4737500A (en) | 1988-04-12 |
NL8601494A (nl) | 1987-01-16 |
SE8602723D0 (sv) | 1986-06-18 |
DK292986D0 (da) | 1986-06-20 |
HUT43600A (en) | 1987-11-30 |
GR861601B (en) | 1986-10-20 |
GB2177395B (en) | 1989-04-26 |
DK292986A (da) | 1986-12-23 |
IT1203806B (it) | 1989-02-23 |
FI862644A (fi) | 1986-12-23 |
FR2587342A1 (fr) | 1987-03-20 |
GB2177395A (en) | 1987-01-21 |
SE8602723L (sv) | 1986-12-23 |
ES556363A0 (es) | 1988-04-01 |
GB8614974D0 (en) | 1986-07-23 |
IL79178A0 (en) | 1986-09-30 |
AU5894086A (en) | 1986-12-24 |
IT8648157A0 (it) | 1986-06-20 |
BE904945A (fr) | 1986-12-18 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
ES557723A0 (es) | Procedimiento para la produccion de tiazoles | |
ES556927A0 (es) | Procedimiento para la produccion de derivados de la 13-betamilbemicina | |
ES557231A0 (es) | Procedimiento para la preparacion de 3-ariluracilos | |
ES551625A0 (es) | Procedimiento para la preparacion de 13-alquil-ll b -fenil-gonamos | |
ES2016244B3 (es) | Procedimiento para produccion de placas de conexion | |
IT1190018B (it) | Procedimento per la produzione di beta-allumina | |
ES551071A0 (es) | Procedimiento para la fabricacion de nuevos antibioticos de b-lactama | |
ES556313A0 (es) | Procedimiento para la produccion de gamma-butirolactona. | |
ES555434A0 (es) | Procedimiento para la preparacion de benzoil-ureas | |
ES556533A0 (es) | Procedimiento para la obtencion de determinadas parejas de enantiomeros de permetrinato de l-ciano-3-fenoxi-4-fluorbencilo | |
ES557428A0 (es) | Procedimiento para la fabricacion de derivados nucleosidos | |
MX3681A (es) | Procedimiento para la produccion de gamma-carbolinas antipsicoticas y compuestos obtenidos. | |
ES552935A0 (es) | Procedimiento para la produccion de d-l-amino acidos | |
ES533735A0 (es) | Procedimiento para la produccion de espirosuccinimidas | |
MX162552A (es) | Procedimiento para la preparacion de benzoil-ureas | |
ES554942A0 (es) | Procedimiento para la obtencion de nuevos compuestos de piridazinio | |
ES552282A0 (es) | Procedimiento para la obtencion de cefalosporinas | |
MX162939B (es) | Procedimiento mejorado para la preparacion de monoterbutiltolueno-diamina | |
ES553986A0 (es) | Procedimiento para la obtencion de compuestos de heterociclil-penem | |
MX157830A (es) | Procedimiento para la produccion de beta-fenilserina | |
ES555278A0 (es) | Procedimiento para la obtencion de derivados de diclorociclopropilalquilhidroxialquil-azol | |
ES557233A0 (es) | Procedimiento para la preparacion de 3-ariluracilos | |
ES545451A0 (es) | Procedimiento para la fabricacion de derivados de pirrolidi-na | |
ES539586A0 (es) | Procedimiento para la produccion de derivados de bencimida- zol | |
ES539587A0 (es) | Procedimiento para la produccion de derivados de bencimida- zol |