ES460411A2 - Procedimiento de preparacion de derivados arilamino-pirimi- dinicos. - Google Patents
Procedimiento de preparacion de derivados arilamino-pirimi- dinicos.Info
- Publication number
- ES460411A2 ES460411A2 ES460411A ES460411A ES460411A2 ES 460411 A2 ES460411 A2 ES 460411A2 ES 460411 A ES460411 A ES 460411A ES 460411 A ES460411 A ES 460411A ES 460411 A2 ES460411 A2 ES 460411A2
- Authority
- ES
- Spain
- Prior art keywords
- preparation
- derivatives
- arylaminopyrimidine
- therapeutics
- application
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/32—One oxygen, sulfur or nitrogen atom
- C07D239/42—One nitrogen atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Neurology (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Neurosurgery (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Biomedical Technology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hospice & Palliative Care (AREA)
- Cardiology (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Liquid Crystal Substances (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Mejoras introducidas en el objeto de la patente principal Nº 429.869, concedida el 27 de Marzo de 1976: Procedimiento de preparación de derivados arilamino-pirimidínicos¿¿, refiriéndose dichas mejoras a un procedimiento de preparación de los compuestos que responden a la fórmula ***
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR7620775A FR2357252A2 (fr) | 1976-07-07 | 1976-07-07 | Nouveaux derives arylaminopyrimidiniques, leur procede de preparation et leur application en therapeutique |
FR7718471A FR2394543A2 (fr) | 1977-06-16 | 1977-06-16 | Nouveaux derives arylaminopyrimidiniques, leur procede de preparation et leur application en therapeutique |
Publications (1)
Publication Number | Publication Date |
---|---|
ES460411A2 true ES460411A2 (es) | 1978-10-01 |
Family
ID=26219529
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES460411A Expired ES460411A2 (es) | 1976-07-07 | 1977-07-05 | Procedimiento de preparacion de derivados arilamino-pirimi- dinicos. |
Country Status (11)
Country | Link |
---|---|
JP (1) | JPS5312877A (es) |
AU (1) | AU2680877A (es) |
CH (1) | CH611283A5 (es) |
DE (1) | DE2729360A1 (es) |
ES (1) | ES460411A2 (es) |
GB (1) | GB1548858A (es) |
IT (1) | IT1114810B (es) |
LU (1) | LU77660A1 (es) |
NL (1) | NL7707531A (es) |
SE (1) | SE7707880L (es) |
SU (1) | SU679143A3 (es) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8455489B2 (en) | 2003-11-10 | 2013-06-04 | Exelixis, Inc. | Substituted pyrimidine compositions and methods of use |
-
1977
- 1977-06-21 GB GB25894/77A patent/GB1548858A/en not_active Expired
- 1977-06-22 CH CH765677A patent/CH611283A5/xx not_active IP Right Cessation
- 1977-06-24 IT IT25031/77A patent/IT1114810B/it active
- 1977-06-29 DE DE19772729360 patent/DE2729360A1/de not_active Ceased
- 1977-06-30 LU LU77660A patent/LU77660A1/xx unknown
- 1977-07-05 ES ES460411A patent/ES460411A2/es not_active Expired
- 1977-07-06 NL NL7707531A patent/NL7707531A/xx not_active Application Discontinuation
- 1977-07-06 SU SU772499407A patent/SU679143A3/ru active
- 1977-07-06 JP JP8090477A patent/JPS5312877A/ja active Pending
- 1977-07-06 AU AU26808/77A patent/AU2680877A/en active Pending
- 1977-07-06 SE SE7707880A patent/SE7707880L/xx unknown
Also Published As
Publication number | Publication date |
---|---|
JPS5312877A (en) | 1978-02-04 |
SU679143A3 (ru) | 1979-08-05 |
NL7707531A (nl) | 1978-01-10 |
IT1114810B (it) | 1986-01-27 |
LU77660A1 (es) | 1978-01-27 |
SE7707880L (sv) | 1978-01-08 |
CH611283A5 (en) | 1979-05-31 |
AU2680877A (en) | 1979-01-11 |
DE2729360A1 (de) | 1978-01-12 |
GB1548858A (en) | 1979-07-18 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FD2A | Announcement of lapse in spain |
Effective date: 20170706 |