ES424851A1 - Un procedimiento para preparar derivados de piperazina. - Google Patents

Un procedimiento para preparar derivados de piperazina.

Info

Publication number
ES424851A1
ES424851A1 ES424851A ES424851A ES424851A1 ES 424851 A1 ES424851 A1 ES 424851A1 ES 424851 A ES424851 A ES 424851A ES 424851 A ES424851 A ES 424851A ES 424851 A1 ES424851 A1 ES 424851A1
Authority
ES
Spain
Prior art keywords
formula
translation
procedure
machine
group
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES424851A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Dainippon Pharmaceutical Co Ltd
Original Assignee
Dainippon Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP3845373A external-priority patent/JPS5546400B2/ja
Priority claimed from JP5654473A external-priority patent/JPS565753B2/ja
Priority claimed from JP6446473A external-priority patent/JPS565755B2/ja
Application filed by Dainippon Pharmaceutical Co Ltd filed Critical Dainippon Pharmaceutical Co Ltd
Publication of ES424851A1 publication Critical patent/ES424851A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
ES424851A 1973-04-03 1974-04-02 Un procedimiento para preparar derivados de piperazina. Expired ES424851A1 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP3845373A JPS5546400B2 (es) 1973-04-03 1973-04-03
JP5654473A JPS565753B2 (es) 1973-05-21 1973-05-21
JP6446473A JPS565755B2 (es) 1973-06-07 1973-06-07

Publications (1)

Publication Number Publication Date
ES424851A1 true ES424851A1 (es) 1976-06-01

Family

ID=27289838

Family Applications (1)

Application Number Title Priority Date Filing Date
ES424851A Expired ES424851A1 (es) 1973-04-03 1974-04-02 Un procedimiento para preparar derivados de piperazina.

Country Status (11)

Country Link
AR (2) AR204003A1 (es)
AT (1) AT340931B (es)
CA (1) CA1066701A (es)
CH (1) CH593281A5 (es)
ES (1) ES424851A1 (es)
FI (1) FI56011C (es)
IE (1) IE39102B1 (es)
NL (1) NL186087C (es)
NO (1) NO142221C (es)
PH (2) PH10529A (es)
SE (1) SE416051B (es)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1209163B (it) * 1979-12-21 1989-07-10 Unibios S P A Trecate Novara Procedimento per la fabbricazione di: 6-alcossicarbonil-8-etil-5-oxo-5,8diidro-aperta par. quadrata 2,3-dchiusa par. quadrata-primidine 2-sostituite ed acidi libri corrispondenti.
SI2448938T1 (sl) 2009-06-29 2014-08-29 Incyte Corporation Experimental Station Pirimidinoni kot zaviralci pi3k
US8759359B2 (en) 2009-12-18 2014-06-24 Incyte Corporation Substituted heteroaryl fused derivatives as PI3K inhibitors
AR079529A1 (es) 2009-12-18 2012-02-01 Incyte Corp Derivados arilo y heteroarilo sustituidos y fundidos como inhibidores de la pi3k
US9096600B2 (en) 2010-12-20 2015-08-04 Incyte Corporation N-(1-(substituted-phenyl)ethyl)-9H-purin-6-amines as PI3K inhibitors
EP3513793B1 (en) 2011-09-02 2021-03-10 Incyte Holdings Corporation Heterocyclylamines as pi3k inhibitors
AR090548A1 (es) 2012-04-02 2014-11-19 Incyte Corp Azaheterociclobencilaminas biciclicas como inhibidores de pi3k
WO2015191677A1 (en) 2014-06-11 2015-12-17 Incyte Corporation Bicyclic heteroarylaminoalkyl phenyl derivatives as pi3k inhibitors
CN117736209A (zh) 2015-02-27 2024-03-22 因赛特控股公司 Pi3k抑制剂的盐及其制备方法
US9988401B2 (en) 2015-05-11 2018-06-05 Incyte Corporation Crystalline forms of a PI3K inhibitor
WO2016183060A1 (en) 2015-05-11 2016-11-17 Incyte Corporation Process for the synthesis of a phosphoinositide 3-kinase inhibitor

Also Published As

Publication number Publication date
NO142221C (no) 1980-07-16
AR204003A1 (es) 1975-11-12
CA1066701A (en) 1979-11-20
NL7401509A (es) 1974-10-07
CH593281A5 (en) 1977-11-30
FI56011B (fi) 1979-07-31
ATA277774A (de) 1977-05-15
IE39102B1 (en) 1978-08-02
NO740349L (no) 1974-10-04
NO142221B (no) 1980-04-08
FI56011C (fi) 1979-11-12
AR204660A1 (es) 1976-02-20
PH10529A (en) 1977-05-30
NL186087B (nl) 1990-04-17
IE39102L (en) 1974-10-03
NL186087C (nl) 1990-09-17
SE416051B (sv) 1980-11-24
AT340931B (de) 1978-01-10
PH10984A (en) 1977-10-18

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