ES2120885A1 - New thienopyrimidones with antifungal activity - Google Patents
New thienopyrimidones with antifungal activityInfo
- Publication number
- ES2120885A1 ES2120885A1 ES09600646A ES9600646A ES2120885A1 ES 2120885 A1 ES2120885 A1 ES 2120885A1 ES 09600646 A ES09600646 A ES 09600646A ES 9600646 A ES9600646 A ES 9600646A ES 2120885 A1 ES2120885 A1 ES 2120885A1
- Authority
- ES
- Spain
- Prior art keywords
- thienopyrimidones
- new
- antifungal activity
- halogen
- compounds
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Abstract
Compounds of formula I and their salts and solvates in which Ar is a phenyl group optionally substituted by one or more halogen and/or trifluoromethyl groups, R1 is a C1- C4 alkyl group, R2 is hydrogen or a C1-C4 alkyl group, or R1 together with R2 form a C2-C4 polymethylene chain, R3 represents cyano, halogen, C1-C4 haloalkyl or C1-C4 haloalkoxy, and R4 represents hydrogen or C1-C4 alkyl. These compounds are useful as antifungal agents. Processes for obtaining them and pharmaceutical compositions containing them are also described. <IMAGE>
Priority Applications (17)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ES9600646A ES2120885B1 (en) | 1996-03-15 | 1996-03-15 | NEW TIENOPIRIMIDONAS WITH ANTIFUNGAL ACTIVITY. |
DE69611512T DE69611512T2 (en) | 1995-08-02 | 1996-08-02 | PYRIMIDONE DERIVATIVES WITH ANTIFUNGAL EFFECT |
EP96929201A EP0783501B9 (en) | 1995-08-02 | 1996-08-02 | pyrimidone derivatives with antifungal activity |
KR1019970701515A KR100423590B1 (en) | 1995-08-02 | 1996-08-02 | New pyrimidone derivatives with antifungal activity |
MX9702382A MX9702382A (en) | 1995-08-02 | 1996-08-02 | New pyrimidone derivatives with antifungal activity. |
BR9606547A BR9606547A (en) | 1995-08-02 | 1996-08-02 | New pyrimidone derivatives with fungicidal activity |
AU68703/96A AU6870396A (en) | 1995-08-02 | 1996-08-02 | New pyrimidone derivatives with antifungal activity |
CA002201477A CA2201477C (en) | 1995-08-02 | 1996-08-02 | New pyrimidone derivatives with antifungal activity |
PT96929201T PT783501E (en) | 1995-08-02 | 1996-08-02 | PYRIMIDONE DERIVATIVES WITH ANTIFUNGAL ACTIVITY |
JP50725497A JP4049207B2 (en) | 1995-08-02 | 1996-08-02 | Novel pyrimidone derivatives with antifungal activity |
ES96929201T ES2153975T3 (en) | 1995-08-02 | 1996-08-02 | DERIVATIVES OF PIRIMIDONA WITH ANTIFUNGIC ACTIVITY. |
AT96929201T ATE198593T1 (en) | 1995-08-02 | 1996-08-02 | PYRIMIDONE DERIVATIVES WITH ANTI-FUNGAL EFFECT |
PCT/EP1996/003420 WO1997005130A1 (en) | 1995-08-02 | 1996-08-02 | New pyrimidone derivatives with antifungal activity |
US08/809,967 US5807854A (en) | 1995-08-02 | 1996-08-02 | Pyrimidone derivatives with antifungal activity |
DK96929201T DK0783501T3 (en) | 1995-08-02 | 1996-08-02 | Pyrimidone derivatives with anti-fungal activity |
NO19971470A NO312898B1 (en) | 1995-08-02 | 1997-04-01 | New pyrimidone derivatives with fungicidal activity |
GR20010400466T GR3035621T3 (en) | 1995-08-02 | 2001-03-23 | New pyrimidone derivatives with antifungal activity |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ES9600646A ES2120885B1 (en) | 1996-03-15 | 1996-03-15 | NEW TIENOPIRIMIDONAS WITH ANTIFUNGAL ACTIVITY. |
Publications (2)
Publication Number | Publication Date |
---|---|
ES2120885A1 true ES2120885A1 (en) | 1998-11-01 |
ES2120885B1 ES2120885B1 (en) | 1999-06-16 |
Family
ID=8294213
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES9600646A Expired - Fee Related ES2120885B1 (en) | 1995-08-02 | 1996-03-15 | NEW TIENOPIRIMIDONAS WITH ANTIFUNGAL ACTIVITY. |
Country Status (1)
Country | Link |
---|---|
ES (1) | ES2120885B1 (en) |
Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES2024336A6 (en) * | 1990-10-16 | 1992-02-16 | Uriach & Cia Sa J | Process for obtaining new thiazole derivatives |
EP0567982A1 (en) * | 1992-04-28 | 1993-11-03 | Takeda Chemical Industries, Ltd. | Azole compounds, their production and use |
-
1996
- 1996-03-15 ES ES9600646A patent/ES2120885B1/en not_active Expired - Fee Related
Patent Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES2024336A6 (en) * | 1990-10-16 | 1992-02-16 | Uriach & Cia Sa J | Process for obtaining new thiazole derivatives |
EP0567982A1 (en) * | 1992-04-28 | 1993-11-03 | Takeda Chemical Industries, Ltd. | Azole compounds, their production and use |
Also Published As
Publication number | Publication date |
---|---|
ES2120885B1 (en) | 1999-06-16 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
EC2A | Search report published |
Date of ref document: 19981101 Kind code of ref document: A1 Effective date: 19981101 |
|
FD1A | Patent lapsed |
Effective date: 20020404 |