EP3723761A4 - Forme pharmaceutique orale solide comprenant de la linagliptine - Google Patents
Forme pharmaceutique orale solide comprenant de la linagliptine Download PDFInfo
- Publication number
- EP3723761A4 EP3723761A4 EP18914956.0A EP18914956A EP3723761A4 EP 3723761 A4 EP3723761 A4 EP 3723761A4 EP 18914956 A EP18914956 A EP 18914956A EP 3723761 A4 EP3723761 A4 EP 3723761A4
- Authority
- EP
- European Patent Office
- Prior art keywords
- linagliptin
- dosage form
- oral dosage
- solid oral
- solid
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- LTXREWYXXSTFRX-QGZVFWFLSA-N Linagliptin Chemical compound N=1C=2N(C)C(=O)N(CC=3N=C4C=CC=CC4=C(C)N=3)C(=O)C=2N(CC#CC)C=1N1CCC[C@@H](N)C1 LTXREWYXXSTFRX-QGZVFWFLSA-N 0.000 title 1
- 229960002397 linagliptin Drugs 0.000 title 1
- 239000006186 oral dosage form Substances 0.000 title 1
- 239000007787 solid Substances 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
- A61K31/52—Purines, e.g. adenine
- A61K31/522—Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
TR2017/20515A TR201720515A2 (tr) | 2017-12-15 | 2017-12-15 | Li̇nagli̇pti̇n i̇çeren bi̇r kati oral dozaj formu |
PCT/TR2018/050812 WO2019203755A2 (fr) | 2017-12-15 | 2018-12-14 | Forme pharmaceutique orale solide comprenant de la linagliptine |
Publications (2)
Publication Number | Publication Date |
---|---|
EP3723761A2 EP3723761A2 (fr) | 2020-10-21 |
EP3723761A4 true EP3723761A4 (fr) | 2021-06-30 |
Family
ID=67900883
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EP18914956.0A Pending EP3723761A4 (fr) | 2017-12-15 | 2018-12-14 | Forme pharmaceutique orale solide comprenant de la linagliptine |
Country Status (4)
Country | Link |
---|---|
EP (1) | EP3723761A4 (fr) |
CA (1) | CA3085455C (fr) |
TR (1) | TR201720515A2 (fr) |
WO (1) | WO2019203755A2 (fr) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2022173406A1 (fr) * | 2021-02-15 | 2022-08-18 | Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi | Procédé pour formulations de linagliptine ou d'un sel pharmaceutiquement acceptable de celle-ci |
WO2024136773A1 (fr) * | 2022-12-21 | 2024-06-27 | Santa Farma Ilac Sanayii A.S. | Composition pharmaceutique stable comprenant de la linagliptine |
Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2010092124A1 (fr) * | 2009-02-13 | 2010-08-19 | Boehringer Ingelheim International Gmbh | Composition pharmaceutique contenant de la linagliptine et facultativement un inhibiteur sglt-2, et ses utilisations |
US20140100236A1 (en) * | 2012-10-09 | 2014-04-10 | Boehringer Ingelheim International Gmbh | Use of selectively moisture-adjusted tabletting material in the production of mechanically stable tablets which contain at least one hydrate-forming active substance and/or adjuvant relevant to the mechanical stability of the tablets, particularly arginine-containing tablets |
WO2014080383A1 (fr) * | 2012-11-26 | 2014-05-30 | Ranbaxy Laboratories Limited | Composition pharmaceutique d'inhibiteurs de la dipeptidyl-peptidase-iv (dpp-iv) en association avec d'autres antidiabétiques |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2013128379A2 (fr) | 2012-02-27 | 2013-09-06 | Dr. Reddy's Laboratories Limited | Formes polymorphes cristallines de linagliptine |
WO2014080384A1 (fr) | 2012-11-26 | 2014-05-30 | Ranbaxy Laboratories Limited | Composition pharmaceutique de linagliptine |
CN106138059A (zh) * | 2015-03-27 | 2016-11-23 | 天津汉瑞药业有限公司 | 一种稳定的利格列汀药物组合物 |
EP3156048A1 (fr) * | 2015-10-13 | 2017-04-19 | Galenicum Health S.L. | Composition pharmaceutique stable de linagliptine sous forme de comprimé à libération immédiate |
-
2017
- 2017-12-15 TR TR2017/20515A patent/TR201720515A2/tr unknown
-
2018
- 2018-12-14 CA CA3085455A patent/CA3085455C/fr active Active
- 2018-12-14 WO PCT/TR2018/050812 patent/WO2019203755A2/fr unknown
- 2018-12-14 EP EP18914956.0A patent/EP3723761A4/fr active Pending
Patent Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2010092124A1 (fr) * | 2009-02-13 | 2010-08-19 | Boehringer Ingelheim International Gmbh | Composition pharmaceutique contenant de la linagliptine et facultativement un inhibiteur sglt-2, et ses utilisations |
US20140100236A1 (en) * | 2012-10-09 | 2014-04-10 | Boehringer Ingelheim International Gmbh | Use of selectively moisture-adjusted tabletting material in the production of mechanically stable tablets which contain at least one hydrate-forming active substance and/or adjuvant relevant to the mechanical stability of the tablets, particularly arginine-containing tablets |
WO2014080383A1 (fr) * | 2012-11-26 | 2014-05-30 | Ranbaxy Laboratories Limited | Composition pharmaceutique d'inhibiteurs de la dipeptidyl-peptidase-iv (dpp-iv) en association avec d'autres antidiabétiques |
Also Published As
Publication number | Publication date |
---|---|
EP3723761A2 (fr) | 2020-10-21 |
CA3085455A1 (fr) | 2019-10-24 |
WO2019203755A3 (fr) | 2020-01-16 |
CA3085455C (fr) | 2022-08-16 |
WO2019203755A2 (fr) | 2019-10-24 |
TR201720515A2 (tr) | 2019-07-22 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
STAA | Information on the status of an ep patent application or granted ep patent |
Free format text: STATUS: THE INTERNATIONAL PUBLICATION HAS BEEN MADE |
|
PUAI | Public reference made under article 153(3) epc to a published international application that has entered the european phase |
Free format text: ORIGINAL CODE: 0009012 |
|
STAA | Information on the status of an ep patent application or granted ep patent |
Free format text: STATUS: REQUEST FOR EXAMINATION WAS MADE |
|
17P | Request for examination filed |
Effective date: 20200714 |
|
AK | Designated contracting states |
Kind code of ref document: A2 Designated state(s): AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR |
|
AX | Request for extension of the european patent |
Extension state: BA ME |
|
DAV | Request for validation of the european patent (deleted) | ||
DAX | Request for extension of the european patent (deleted) | ||
A4 | Supplementary search report drawn up and despatched |
Effective date: 20210601 |
|
RIC1 | Information provided on ipc code assigned before grant |
Ipc: A61K 31/522 20060101AFI20210526BHEP Ipc: A61K 47/00 20060101ALI20210526BHEP Ipc: A61P 3/10 20060101ALI20210526BHEP |
|
TPAC | Observations filed by third parties |
Free format text: ORIGINAL CODE: EPIDOSNTIPA |
|
P01 | Opt-out of the competence of the unified patent court (upc) registered |
Effective date: 20230708 |
|
STAA | Information on the status of an ep patent application or granted ep patent |
Free format text: STATUS: EXAMINATION IS IN PROGRESS |
|
17Q | First examination report despatched |
Effective date: 20231108 |