EP2429290A4 - Compounds and methods for treating aids and hiv infections - Google Patents
Compounds and methods for treating aids and hiv infectionsInfo
- Publication number
- EP2429290A4 EP2429290A4 EP10775430A EP10775430A EP2429290A4 EP 2429290 A4 EP2429290 A4 EP 2429290A4 EP 10775430 A EP10775430 A EP 10775430A EP 10775430 A EP10775430 A EP 10775430A EP 2429290 A4 EP2429290 A4 EP 2429290A4
- Authority
- EP
- European Patent Office
- Prior art keywords
- compounds
- methods
- hiv infections
- treating aids
- aids
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
- C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
- C07D493/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D515/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen, oxygen, and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D515/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen, oxygen, and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D515/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US17708609P | 2009-05-11 | 2009-05-11 | |
| PCT/US2010/034437 WO2010132494A1 (en) | 2009-05-11 | 2010-05-11 | Compounds and methods for treating aids and hiv infections |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| EP2429290A1 EP2429290A1 (en) | 2012-03-21 |
| EP2429290A4 true EP2429290A4 (en) | 2012-11-07 |
| EP2429290B1 EP2429290B1 (en) | 2014-01-01 |
Family
ID=43085303
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EP20100775430 Not-in-force EP2429290B1 (en) | 2009-05-11 | 2010-05-11 | Compounds and methods for treating aids and hiv infections |
Country Status (3)
| Country | Link |
|---|---|
| US (2) | US8921349B2 (en) |
| EP (1) | EP2429290B1 (en) |
| WO (1) | WO2010132494A1 (en) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2010132494A1 (en) | 2009-05-11 | 2010-11-18 | Ghosh Arun K | Compounds and methods for treating aids and hiv infections |
| WO2012075122A2 (en) | 2010-11-30 | 2012-06-07 | Purdue Research Foundation | Processes and intermediates for preparing substituted hexahydrofuro [2,3-b] furans |
| WO2019006335A1 (en) * | 2017-06-30 | 2019-01-03 | Ghosh Arun K | Macrocyclic hiv-1 protease inhibitors and uses thereof |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2003049746A2 (en) * | 2001-12-12 | 2003-06-19 | Tibotec Pharmaceuticals Ltd. | Combination of cytochome p450 dependent protease inhibitors |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EE9800115A (en) * | 1995-11-14 | 1998-10-15 | The Du Pont Merck Pharmaceutical Company | Novel macrocyclic compounds as metalloprotease inhibitors |
| WO1999067254A2 (en) | 1998-06-23 | 1999-12-29 | The United States Of America Represented By The Secretary, Department Of Health And Human Services | Multi-drug resistant retroviral protease inhibitors and use thereof |
| US7157489B2 (en) * | 2002-03-12 | 2007-01-02 | The Board Of Trustees Of The University Of Illinois | HIV protease inhibitors |
| WO2010132494A1 (en) | 2009-05-11 | 2010-11-18 | Ghosh Arun K | Compounds and methods for treating aids and hiv infections |
-
2010
- 2010-05-11 WO PCT/US2010/034437 patent/WO2010132494A1/en active Application Filing
- 2010-05-11 EP EP20100775430 patent/EP2429290B1/en not_active Not-in-force
- 2010-05-11 US US13/319,973 patent/US8921349B2/en active Active
-
2014
- 2014-10-21 US US14/520,099 patent/US9617276B2/en active Active
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2003049746A2 (en) * | 2001-12-12 | 2003-06-19 | Tibotec Pharmaceuticals Ltd. | Combination of cytochome p450 dependent protease inhibitors |
Non-Patent Citations (2)
| Title |
|---|
| GHOSH A K ET AL: "Design and synthesis of novel HIV-1 protease inhibitors incorporating oxyindoles as the P2<'>-ligands", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, PERGAMON, ELSEVIER SCIENCE, GB, vol. 16, no. 7, 1 April 2006 (2006-04-01), pages 1869 - 1873, XP027966355, ISSN: 0960-894X, [retrieved on 20060401] * |
| See also references of WO2010132494A1 * |
Also Published As
| Publication number | Publication date |
|---|---|
| US20150111962A1 (en) | 2015-04-23 |
| US9617276B2 (en) | 2017-04-11 |
| EP2429290B1 (en) | 2014-01-01 |
| US8921349B2 (en) | 2014-12-30 |
| WO2010132494A1 (en) | 2010-11-18 |
| EP2429290A1 (en) | 2012-03-21 |
| US20120059161A1 (en) | 2012-03-08 |
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| RIC1 | Information provided on ipc code assigned before grant |
Ipc: C07D 493/04 20060101ALI20121002BHEP Ipc: A61K 31/16 20060101ALI20121002BHEP Ipc: C07D 519/00 20060101ALI20121002BHEP Ipc: A61K 31/195 20060101ALI20121002BHEP Ipc: C07D 515/04 20060101ALI20121002BHEP Ipc: A01N 37/44 20060101AFI20121002BHEP |
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