EE03239B1 - 7-hüdroksütaksaani valmistamise meetod - Google Patents

7-hüdroksütaksaani valmistamise meetod

Info

Publication number
EE03239B1
EE03239B1 EE9600141A EE9600141A EE03239B1 EE 03239 B1 EE03239 B1 EE 03239B1 EE 9600141 A EE9600141 A EE 9600141A EE 9600141 A EE9600141 A EE 9600141A EE 03239 B1 EE03239 B1 EE 03239B1
Authority
EE
Estonia
Prior art keywords
radical
pct
general formula
optionally substituted
image
Prior art date
Application number
EE9600141A
Other languages
English (en)
Inventor
Bastart Jean-Pierre
Bourzat Jean-Dominique
Commer�on Alain
Leconte Jean-Pierre
Original Assignee
Rh�Ne-Poulenc Rorer S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rh�Ne-Poulenc Rorer S.A. filed Critical Rh�Ne-Poulenc Rorer S.A.
Publication of EE03239B1 publication Critical patent/EE03239B1/et

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D305/00Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Epoxy Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
EE9600141A 1994-04-05 1995-04-03 7-hüdroksütaksaani valmistamise meetod EE03239B1 (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9403980A FR2718135B1 (fr) 1994-04-05 1994-04-05 Procédé de préparation d'hydroxy-7 taxanes.
PCT/FR1995/000420 WO1995026961A1 (fr) 1994-04-05 1995-04-03 Procede de preparation d'hydroxy-7 taxanes

Publications (1)

Publication Number Publication Date
EE03239B1 true EE03239B1 (et) 1999-12-15

Family

ID=9461748

Family Applications (1)

Application Number Title Priority Date Filing Date
EE9600141A EE03239B1 (et) 1994-04-05 1995-04-03 7-hüdroksütaksaani valmistamise meetod

Country Status (31)

Country Link
US (1) US5750738A (et)
EP (1) EP0754181B1 (et)
JP (1) JPH09511245A (et)
KR (1) KR970702269A (et)
CN (1) CN1066144C (et)
AT (1) ATE168109T1 (et)
AU (1) AU691916B2 (et)
BG (1) BG62731B1 (et)
BR (1) BR9507443A (et)
CA (1) CA2186917A1 (et)
CZ (1) CZ284725B6 (et)
DE (1) DE69503366T2 (et)
DK (1) DK0754181T3 (et)
EE (1) EE03239B1 (et)
ES (1) ES2118592T3 (et)
FI (1) FI964002A0 (et)
FR (1) FR2718135B1 (et)
GE (1) GEP19991535B (et)
HU (1) HU214157B (et)
LT (1) LT4186B (et)
LV (1) LV11685B (et)
NO (1) NO314145B1 (et)
NZ (1) NZ284491A (et)
PL (1) PL316589A1 (et)
RO (1) RO115727B1 (et)
RU (1) RU2127730C1 (et)
SK (1) SK281075B6 (et)
TW (1) TW285669B (et)
UA (1) UA45332C2 (et)
WO (1) WO1995026961A1 (et)
ZA (1) ZA952732B (et)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2732968B1 (fr) * 1995-04-14 1997-05-16 Rhone Poulenc Rorer Sa Nouveaux taxoides, leur preparation et les compositions pharmaceutiques qui les contiennent
FR2750989B1 (fr) * 1996-07-09 1998-09-25 Rhone Poulenc Rorer Sa Procede de monoacylation d'hydroxy taxanes
AU761389B2 (en) * 1999-05-17 2003-06-05 Bristol-Myers Squibb Company Novel reaction conditions for the cleavage of silyl ethers in the preparation of paclitaxel (taxol) and paclitaxel analogues
CA2385528C (en) 1999-10-01 2013-12-10 Immunogen, Inc. Compositions and methods for treating cancer using immunoconjugates and chemotherapeutic agents
PT3351558T (pt) 2009-11-13 2020-04-09 Daiichi Sankyo Europe Gmbh Material e métodos para tratamento ou prevenção de doenças associadas a her-3
JP2013540694A (ja) 2010-08-06 2013-11-07 ウー3・フアルマ・ゲー・エム・ベー・ハー Her3結合剤の前立腺治療における使用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2629818B1 (fr) * 1988-04-06 1990-11-16 Centre Nat Rech Scient Procede de preparation du taxol
FR2678930B1 (fr) * 1991-07-10 1995-01-13 Rhone Poulenc Rorer Sa Procede de preparation de derives de la baccatine iii et de la desacetyl-10 baccatine iii.

Also Published As

Publication number Publication date
BG62731B1 (bg) 2000-06-30
NO964104D0 (no) 1996-09-27
HU9602736D0 (en) 1996-11-28
HU214157B (hu) 1998-01-28
CN1145070A (zh) 1997-03-12
CN1066144C (zh) 2001-05-23
UA45332C2 (uk) 2002-04-15
GEP19991535B (en) 1999-03-05
LT96138A (en) 1997-02-25
LV11685A (lv) 1997-02-20
HUT75690A (en) 1997-05-28
NZ284491A (en) 1998-01-26
BG100887A (en) 1998-01-30
FI964002A (fi) 1996-10-04
NO964104L (no) 1996-09-27
PL316589A1 (en) 1997-01-20
CA2186917A1 (fr) 1995-10-12
RO115727B1 (ro) 2000-05-30
LT4186B (en) 1997-07-25
LV11685B (en) 1997-06-20
ATE168109T1 (de) 1998-07-15
FI964002A0 (fi) 1996-10-04
CZ284725B6 (cs) 1999-02-17
ES2118592T3 (es) 1998-09-16
WO1995026961A1 (fr) 1995-10-12
US5750738A (en) 1998-05-12
BR9507443A (pt) 1997-09-16
TW285669B (et) 1996-09-11
DK0754181T3 (da) 1998-11-16
SK281075B6 (sk) 2000-11-07
MX9604465A (es) 1997-07-31
EP0754181B1 (fr) 1998-07-08
FR2718135B1 (fr) 1996-04-26
ZA952732B (en) 1996-01-09
AU691916B2 (en) 1998-05-28
SK126496A3 (en) 1997-05-07
EP0754181A1 (fr) 1997-01-22
NO314145B1 (no) 2003-02-03
DE69503366T2 (de) 1999-01-21
FR2718135A1 (fr) 1995-10-06
KR970702269A (ko) 1997-05-13
RU2127730C1 (ru) 1999-03-20
DE69503366D1 (de) 1998-08-13
AU2309795A (en) 1995-10-23
CZ289996A3 (en) 1997-01-15
JPH09511245A (ja) 1997-11-11

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DK0663905T3 (da) Ny fremgangsmåde dtil forestring af baccatin III og 10-desacetylbaccatin III
EE03239B1 (et) 7-hüdroksütaksaani valmistamise meetod
BR9507444A (pt) Processo de preparação de trialcoilsilil 7 bacatina III
BR9510235A (pt) Taxóides seu processo de preparação e composição farmacêutica que os contêm
NO951840L (no) Fremgangsmåte for fremstilling av 1,3-oksazolidin-5-karboksylsyre
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Legal Events

Date Code Title Description
KB4A Valid patent at the end of a year

Effective date: 20021231

MM4A Lapsed by not paying the annual fees

Effective date: 20030403