EA201690655A1 - Новые соединения в качестве модуляторов протеинкиназ - Google Patents
Новые соединения в качестве модуляторов протеинкиназInfo
- Publication number
- EA201690655A1 EA201690655A1 EA201690655A EA201690655A EA201690655A1 EA 201690655 A1 EA201690655 A1 EA 201690655A1 EA 201690655 A EA201690655 A EA 201690655A EA 201690655 A EA201690655 A EA 201690655A EA 201690655 A1 EA201690655 A1 EA 201690655A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- modulators
- proteinkinase
- new connections
- methods
- kinase
- Prior art date
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
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- C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
- C07D473/32—Nitrogen atom
- C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
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- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
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- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Abstract
В настоящем изобретении представлены модуляторы протеинкиназы PI3K, способы их получения, фармацевтические композиции, содержащие их, а также способы лечения, предупреждения и/или улучшения с их помощью киназа-опосредованных заболеваний или расстройств.
Applications Claiming Priority (1)
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IN81CH2012 | 2012-01-09 |
Publications (2)
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EA201690655A1 true EA201690655A1 (ru) | 2017-01-30 |
EA039266B1 EA039266B1 (ru) | 2021-12-24 |
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EA201690655A EA039266B1 (ru) | 2012-01-09 | 2012-05-04 | Производные 4н-хромен-4-она в качестве модуляторов протеинкиназ |
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JPS62201882A (ja) * | 1985-11-18 | 1987-09-05 | Yamanouchi Pharmaceut Co Ltd | イソフラボン誘導体 |
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