EA201690655A1 - Новые соединения в качестве модуляторов протеинкиназ - Google Patents

Новые соединения в качестве модуляторов протеинкиназ

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Publication number
EA201690655A1
EA201690655A1 EA201690655A EA201690655A EA201690655A1 EA 201690655 A1 EA201690655 A1 EA 201690655A1 EA 201690655 A EA201690655 A EA 201690655A EA 201690655 A EA201690655 A EA 201690655A EA 201690655 A1 EA201690655 A1 EA 201690655A1
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EA
Eurasian Patent Office
Prior art keywords
modulators
proteinkinase
new connections
methods
kinase
Prior art date
Application number
EA201690655A
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English (en)
Other versions
EA039266B1 (ru
Inventor
Дханапалан Нагаратхнам
Сваруп Кумар В.С. Ваккаланка
Мейяппан Мутуппаланиаппан
Срикант Висванадха
Говиндараджулу Бабу
Прашант Кашинат Бхавар
Original Assignee
Ризен Фармасьютикалз Са
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Application filed by Ризен Фармасьютикалз Са filed Critical Ризен Фармасьютикалз Са
Publication of EA201690655A1 publication Critical patent/EA201690655A1/ru
Publication of EA039266B1 publication Critical patent/EA039266B1/ru

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    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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Abstract

В настоящем изобретении представлены модуляторы протеинкиназы PI3K, способы их получения, фармацевтические композиции, содержащие их, а также способы лечения, предупреждения и/или улучшения с их помощью киназа-опосредованных заболеваний или расстройств.
EA201690655A 2012-01-09 2012-05-04 Производные 4н-хромен-4-она в качестве модуляторов протеинкиназ EA039266B1 (ru)

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EA201690655A1 true EA201690655A1 (ru) 2017-01-30
EA039266B1 EA039266B1 (ru) 2021-12-24

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* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS62201882A (ja) * 1985-11-18 1987-09-05 Yamanouchi Pharmaceut Co Ltd イソフラボン誘導体

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