EA201591192A1 - Антибактериальные соединения - Google Patents
Антибактериальные соединенияInfo
- Publication number
- EA201591192A1 EA201591192A1 EA201591192A EA201591192A EA201591192A1 EA 201591192 A1 EA201591192 A1 EA 201591192A1 EA 201591192 A EA201591192 A EA 201591192A EA 201591192 A EA201591192 A EA 201591192A EA 201591192 A1 EA201591192 A1 EA 201591192A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- antibacterial
- connections
- compounds
- relates
- present
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/82—Nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
- A61K31/423—Oxazoles condensed with carbocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/428—Thiazoles condensed with carbocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A61P31/06—Antibacterial agents for tuberculosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
- C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
- C07D263/58—Benzoxazoles; Hydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Communicable Diseases (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Oncology (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Настоящее изобретение относится к следующим соединениям для применения в лечении бактериальной инфекциигде целые числа определены в описании. Настоящее изобретение также относится к соединениям для применения в качестве лекарственных препаратов, фармацевтическим композициям и некоторым новым соединениям.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP12199026 | 2012-12-21 | ||
PCT/EP2013/077565 WO2014096300A2 (en) | 2012-12-21 | 2013-12-20 | Antibacterial compounds |
Publications (2)
Publication Number | Publication Date |
---|---|
EA201591192A1 true EA201591192A1 (ru) | 2015-11-30 |
EA038333B1 EA038333B1 (ru) | 2021-08-11 |
Family
ID=47519922
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA201591192A EA038333B1 (ru) | 2012-12-21 | 2013-12-20 | Антибактериальные соединения |
Country Status (22)
Country | Link |
---|---|
US (3) | US9428474B2 (ru) |
EP (1) | EP2934498B1 (ru) |
JP (1) | JP6441229B2 (ru) |
KR (1) | KR102233199B1 (ru) |
CN (1) | CN104981238B (ru) |
AP (1) | AP2015008503A0 (ru) |
AU (1) | AU2013366572B2 (ru) |
BR (1) | BR112015014145B1 (ru) |
CA (1) | CA2892899C (ru) |
CL (1) | CL2015001781A1 (ru) |
EA (1) | EA038333B1 (ru) |
ES (1) | ES2659953T3 (ru) |
HK (1) | HK1210954A1 (ru) |
MX (1) | MX2015008036A (ru) |
MY (1) | MY173280A (ru) |
NZ (1) | NZ708742A (ru) |
PE (1) | PE20151165A1 (ru) |
PH (1) | PH12015501428B1 (ru) |
SA (1) | SA515360628B1 (ru) |
SG (1) | SG11201504873RA (ru) |
UA (1) | UA117672C2 (ru) |
WO (1) | WO2014096300A2 (ru) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP2934498B1 (en) | 2012-12-21 | 2017-11-15 | Janssen Sciences Ireland UC | Antibacterial compounds |
US9801909B2 (en) | 2015-04-06 | 2017-10-31 | The Penn State Research Foundation | Compositions and methods for combating bacterial infections by killing persister cells with mitomycin C |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BE744970A (fr) * | 1969-01-28 | 1970-07-27 | Lilly Co Eli | Agents antiviraux et immuno-depresseurs |
US4028374A (en) | 1975-11-03 | 1977-06-07 | Morton-Norwich Products, Inc. | Antibacterial thiocyanatobenzothiazoles |
GB8816519D0 (en) | 1987-07-23 | 1988-08-17 | Ici Plc | Antibiotic compounds |
GB9107341D0 (en) | 1991-04-08 | 1991-05-22 | Ici Plc | Antibiotic compounds |
WO2000056725A1 (en) * | 1999-03-19 | 2000-09-28 | Du Pont Pharmaceuticals Company | N-adamant-1-yl-n'-[4-chlorobenzothiazol-2-yl] urea useful in the treatment of inflammation and as an anticancer radiosensitizing agent |
DK2301544T3 (da) | 2002-07-25 | 2013-01-02 | Janssen Pharmaceutica Nv | Quinolinderivater som mellemprodukter til mykobakterielle inhibitorer |
NZ543372A (en) | 2003-05-30 | 2008-11-28 | Hoffmann La Roche | Benzothiazole derivatives and use thereof in the treatment of diseases related to the adenoside A2A receptor |
CA2572750A1 (en) | 2003-09-10 | 2005-03-17 | Anil Koul | Heterobicyclic compounds as pharmaceutically active agents |
EP1680431A1 (en) * | 2003-10-17 | 2006-07-19 | Rigel Pharmaceuticals, Inc. | Benzothiazole and thiazole'5,5-b!pyridine compositions and their use as ubiquitin ligase inhibitors |
EP2024349B1 (en) | 2006-05-31 | 2017-08-02 | AbbVie Inc. | Compounds as cannabinoid receptor ligands and uses thereof |
GB0724342D0 (en) | 2007-12-13 | 2008-01-30 | Prolysis Ltd | Anitbacterial compositions |
EP2934498B1 (en) * | 2012-12-21 | 2017-11-15 | Janssen Sciences Ireland UC | Antibacterial compounds |
-
2013
- 2013-12-20 EP EP13814926.5A patent/EP2934498B1/en active Active
- 2013-12-20 EA EA201591192A patent/EA038333B1/ru unknown
- 2013-12-20 SG SG11201504873RA patent/SG11201504873RA/en unknown
- 2013-12-20 NZ NZ708742A patent/NZ708742A/en not_active IP Right Cessation
- 2013-12-20 MY MYPI2015001584A patent/MY173280A/en unknown
- 2013-12-20 UA UAA201507312A patent/UA117672C2/uk unknown
- 2013-12-20 WO PCT/EP2013/077565 patent/WO2014096300A2/en active Application Filing
- 2013-12-20 AU AU2013366572A patent/AU2013366572B2/en active Active
- 2013-12-20 JP JP2015548614A patent/JP6441229B2/ja active Active
- 2013-12-20 BR BR112015014145-5A patent/BR112015014145B1/pt active IP Right Grant
- 2013-12-20 CA CA2892899A patent/CA2892899C/en active Active
- 2013-12-20 CN CN201380067207.4A patent/CN104981238B/zh active Active
- 2013-12-20 US US14/654,186 patent/US9428474B2/en active Active
- 2013-12-20 PE PE2015001057A patent/PE20151165A1/es active IP Right Grant
- 2013-12-20 AP AP2015008503A patent/AP2015008503A0/xx unknown
- 2013-12-20 MX MX2015008036A patent/MX2015008036A/es unknown
- 2013-12-20 ES ES13814926.5T patent/ES2659953T3/es active Active
- 2013-12-20 KR KR1020157018199A patent/KR102233199B1/ko active IP Right Grant
-
2015
- 2015-06-18 SA SA515360628A patent/SA515360628B1/ar unknown
- 2015-06-19 PH PH12015501428A patent/PH12015501428B1/en unknown
- 2015-06-19 CL CL2015001781A patent/CL2015001781A1/es unknown
- 2015-12-01 HK HK15111776.0A patent/HK1210954A1/xx unknown
-
2016
- 2016-08-08 US US15/231,389 patent/US9758497B2/en active Active
-
2017
- 2017-09-08 US US15/699,770 patent/US9951032B2/en active Active
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
EA201890201A1 (ru) | Антибактериальные соединения | |
EA201500536A1 (ru) | Триазолопиразин | |
EA201992133A1 (ru) | Производные пиперидино-пиримидина для лечения вирусных инфекций | |
JO3357B1 (ar) | مركبات إيميدازوبيروليدينون | |
EA201491412A1 (ru) | Соединения для лечения спинальной мышечной атрофии | |
UA116648C2 (uk) | Фумарати як проліки та їх застосування при лікуванні різних захворювань | |
EA201491766A1 (ru) | Соединения для лечения спинальной мышечной атрофии | |
EA201390274A1 (ru) | Борсодержащие малые молекулы | |
EA201591166A1 (ru) | Ингибиторы аутотаксина | |
EA201590931A1 (ru) | Гетероциклические замещенные производные 2-амино-хиназолина для лечения вирусных инфекций | |
EA201201661A1 (ru) | Новые аминопиразолохиназолины | |
PH12015501609A1 (en) | Phenicol antibacterials | |
EA201500383A1 (ru) | Производные 1,2,4-триазина для лечения вирусных инфекций | |
EA201590667A1 (ru) | Ациламинопиримидиновые производные для лечения вирусных инфекций и других заболеваний | |
EA201400976A1 (ru) | Бензодиоксаны в комбинации с другими активными средствами для ингибирования продуцирования лейкотриена | |
EA201591451A1 (ru) | Модуляторы flap | |
EA201590787A1 (ru) | Замещенные пиридопиразины в качестве ингибиторов syk | |
EA201590475A1 (ru) | Тетрациклиновые соединения | |
MX367309B (es) | Nuevos compuestos antibacterianos. | |
MX2015001835A (es) | Nuevos compuestos antibacterianos. | |
EA201591192A1 (ru) | Антибактериальные соединения | |
MX2015015251A (es) | Derivados de la quinolona. | |
BR112015006220A2 (pt) | agentes antibacterianos de tetrahidroquinolina tricíclica | |
EA201390764A1 (ru) | Фармацевтические композиции | |
WO2014006601A3 (en) | Nanoparticle compositions of antibacterial compounds and other uses thereof |