EA201270253A1 - Производные n1-ацил-5-фторпиримидинона - Google Patents

Производные n1-ацил-5-фторпиримидинона

Info

Publication number
EA201270253A1
EA201270253A1 EA201270253A EA201270253A EA201270253A1 EA 201270253 A1 EA201270253 A1 EA 201270253A1 EA 201270253 A EA201270253 A EA 201270253A EA 201270253 A EA201270253 A EA 201270253A EA 201270253 A1 EA201270253 A1 EA 201270253A1
Authority
EA
Eurasian Patent Office
Prior art keywords
acyl
derivatives
ftorpyrimidinona
fluoropyrimidinones
fungicides
Prior art date
Application number
EA201270253A
Other languages
English (en)
Other versions
EA023411B1 (ru
Inventor
Тимоти Бебель
Кристи Брайан
Бет Лорсбах
Тимоти Мартин
В. Оуэн
Марк Побанс
Скотт Торнберг
Джеффри Вебстер
Чэнлинь Яо
Original Assignee
ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535292&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA201270253(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи filed Critical ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи
Publication of EA201270253A1 publication Critical patent/EA201270253A1/ru
Publication of EA023411B1 publication Critical patent/EA023411B1/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Настоящее изобретение относится к области N1-ацил-5-фторпиримидинонов и их производных и к применению этих соединений в качестве фунгицидов.
EA201270253A 2009-08-07 2010-08-05 Производные n1-ацил-5-фторпиримидинона EA023411B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23222309P 2009-08-07 2009-08-07
PCT/US2010/044576 WO2011017538A1 (en) 2009-08-07 2010-08-05 N1-acyl-5-fluoropyrimidinone derivatives

Publications (2)

Publication Number Publication Date
EA201270253A1 true EA201270253A1 (ru) 2012-07-30
EA023411B1 EA023411B1 (ru) 2016-06-30

Family

ID=43535292

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201270253A EA023411B1 (ru) 2009-08-07 2010-08-05 Производные n1-ацил-5-фторпиримидинона

Country Status (34)

Country Link
US (1) US8470839B2 (ru)
EP (1) EP2519512B1 (ru)
JP (1) JP5748754B2 (ru)
KR (1) KR101792285B1 (ru)
CN (1) CN102548981B (ru)
AU (1) AU2010279402B2 (ru)
BR (1) BR112012002810B1 (ru)
CA (1) CA2768510C (ru)
CL (1) CL2012000316A1 (ru)
CO (1) CO6491117A2 (ru)
CR (1) CR20120030A (ru)
CY (1) CY1122115T1 (ru)
DK (1) DK2519512T3 (ru)
EA (1) EA023411B1 (ru)
EC (1) ECSP12011653A (ru)
ES (1) ES2728966T3 (ru)
HK (1) HK1172894A1 (ru)
HN (1) HN2012000269A (ru)
HR (1) HRP20190919T1 (ru)
HU (1) HUE045290T2 (ru)
IL (1) IL217952A (ru)
IN (1) IN2012DN00539A (ru)
LT (1) LT2519512T (ru)
MX (1) MX2012001620A (ru)
NI (1) NI201200022A (ru)
NZ (1) NZ597570A (ru)
PE (1) PE20120688A1 (ru)
PL (1) PL2519512T3 (ru)
PT (1) PT2519512T (ru)
SI (1) SI2519512T1 (ru)
TR (1) TR201908180T4 (ru)
UA (1) UA106889C2 (ru)
WO (1) WO2011017538A1 (ru)
ZA (1) ZA201200819B (ru)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2769073C (en) * 2009-08-07 2018-07-24 Dow Agrosciences Llc N1-sulfonyl-5-fluoropyrimidinone derivatives
JP6128658B2 (ja) * 2011-08-17 2017-05-17 アダマ・マクテシム・リミテッド ５−フルオロ−４−イミノ−３−（置換）−３，４−ジヒドロピリミジン−２−（１ｈ）−オン誘導体
RU2015131149A (ru) 2012-12-28 2017-02-03 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи N-(замещенные)-5-фтор-4-имино-3-метил-2-оксо-3,4-дигидропиримидин-1(2н)-карбоксамидные производные
MX2015008441A (es) 2012-12-28 2015-09-23 Dow Agrosciences Llc Derivados de n-(sustituido)-5-fluoro-4-imino-3-metil-2-oxo-3, 4-dihidropirimidin-1 (2h)-carboxilato.
CN104994859B (zh) * 2012-12-28 2018-10-26 阿达玛马克西姆股份有限公司 1-(取代的苯甲酰基)-5-氟-4-亚氨基-3-甲基-3,4-二氢嘧啶-2(1h)-酮衍生物
MX2015008565A (es) 2012-12-31 2015-09-07 Dow Agrosciences Llc Derivados de 3-alquil-5-fluoro-4-sustituido-imino-3,4-dihidropirim idin-2(1h)-ona como fungicidas.
WO2015103142A1 (en) 2013-12-31 2015-07-09 Dow Agrosciences Llc 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1- (arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
UA124962C2 (uk) 2013-12-31 2021-12-22 Адама Махтешім Лтд. Синергічні фунгіцидні суміші та композиції для контролю грибків
CN107001397B (zh) 2014-09-26 2020-10-13 科慕埃弗西有限公司 异氰酸酯衍生的有机硅烷
BR112020000953A2 (pt) 2017-07-17 2020-07-14 Adama Makhteshim Ltd. polimorfos de 5-fluoro-4-imino-3-metil-1-tosil-3,4-di-hidropirimidin-2-ona

Family Cites Families (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH421973A (de) * 1962-05-01 1966-10-15 Hoffmann La Roche Verfahren zur Herstellung eines Cytosin-Derivates
US3309359A (en) 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3868373A (en) 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (ru) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
EP0139613A1 (de) 1983-08-29 1985-05-02 Ciba-Geigy Ag N-(2-Nitrophenyl)-4-aminopyrimidin-Derivate, deren Herstellung und Verwendung
US4845081A (en) 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
DE58908159D1 (de) 1988-03-09 1994-09-15 Ciba Geigy Ag Mittel zum Schutz von Pflanzen gegen Krankheiten.
DE3821711A1 (de) 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
JP3217191B2 (ja) 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
PL324486A1 (en) 1995-07-05 1998-05-25 Du Pont Fungicidal pyrimidinones
CN1213373A (zh) 1996-03-11 1999-04-07 诺瓦提斯公司 农药用嘧啶－4－酮衍生物
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
WO2003018051A1 (en) 2001-08-27 2003-03-06 Vic Jira Anti-fungal composition
JPWO2005095419A1 (ja) 2004-04-01 2008-02-21 武田薬品工業株式会社 チアゾロピリミジン誘導体
EP2044086A2 (en) 2006-06-30 2009-04-08 Janssen Pharmaceutica N.V. Thiazolopyrimidine modulators of trpv1
US9174970B2 (en) 2008-01-22 2015-11-03 Dow Agrosciences Llc 5-fluoro pyrimidine derivatives
US20100029482A1 (en) 2008-08-01 2010-02-04 Benko Zoltan L Use of 5-fluorocytosine as a fungicide
CA2750413C (en) 2009-01-23 2016-06-21 Northlake Biosciences Llc Hydroxamic acid derivatives
CA2769073C (en) 2009-08-07 2018-07-24 Dow Agrosciences Llc N1-sulfonyl-5-fluoropyrimidinone derivatives

Also Published As

Publication number Publication date
NI201200022A (es) 2012-05-22
HRP20190919T1 (hr) 2019-09-20
US20110034490A1 (en) 2011-02-10
CO6491117A2 (es) 2012-07-31
NZ597570A (en) 2014-04-30
JP5748754B2 (ja) 2015-07-15
MX2012001620A (es) 2012-04-11
IL217952A (en) 2017-11-30
LT2519512T (lt) 2019-07-25
ES2728966T3 (es) 2019-10-29
EP2519512A1 (en) 2012-11-07
CN102548981A (zh) 2012-07-04
AU2010279402A1 (en) 2012-02-02
HUE045290T2 (hu) 2019-12-30
CL2012000316A1 (es) 2014-06-27
KR20120041786A (ko) 2012-05-02
EP2519512B1 (en) 2019-03-20
WO2011017538A1 (en) 2011-02-10
AU2010279402B2 (en) 2015-04-16
CA2768510A1 (en) 2011-02-10
BR112012002810A2 (pt) 2015-09-15
PE20120688A1 (es) 2012-06-06
EA023411B1 (ru) 2016-06-30
CN102548981B (zh) 2015-05-13
TR201908180T4 (tr) 2019-06-21
UA106889C2 (uk) 2014-10-27
ZA201200819B (en) 2013-05-29
JP2013501723A (ja) 2013-01-17
ECSP12011653A (es) 2012-03-30
SI2519512T1 (sl) 2019-09-30
HN2012000269A (es) 2015-04-27
HK1172894A1 (en) 2013-05-03
IN2012DN00539A (ru) 2015-06-12
DK2519512T3 (da) 2019-05-27
CA2768510C (en) 2018-05-15
PT2519512T (pt) 2019-06-04
CY1122115T1 (el) 2020-11-25
IL217952A0 (en) 2012-03-29
EP2519512A4 (en) 2013-01-16
PL2519512T3 (pl) 2019-09-30
US8470839B2 (en) 2013-06-25
KR101792285B1 (ko) 2017-10-31
CR20120030A (es) 2012-03-28
BR112012002810B1 (pt) 2018-12-11

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Legal Events

Date Code Title Description
PC4A Registration of transfer of a eurasian patent by assignment
MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): AM AZ BY KZ KG MD TJ TM RU